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[2-(azepan-1-yl)ethyl](ethyl)[(2-ethyl-4-methyl-1H-imidazol-5-yl)methyl]amine
N-[1-(1-{5,7-dimethylpyrazolo[1,5-a]pyrimidine-2-carbonyl}piperidin-4-yl)-2-(3-methoxyphenyl)ethyl]-N-methylcyclopropanecarboxamide
2-[(1R,5R)-6-benzyl-3,6-diazabicyclo[3.2.2]nonan-3-yl]pyridine-3-carboxamide
2-methyl-N-{[2-(4-methylpiperazin-1-yl)pyridin-3-yl]methyl}-1H-1,3-benzodiazole-4-carboxamide
N-{[4-(3-methoxypropyl)-4H-1,2,4-triazol-3-yl]methyl}-5-methylpyrazolo[1,5-a]pyrimidin-7-amine
(2R,6S)-4-(1-{1-[(2,6-difluorophenyl)methyl]-1H-1,2,3-triazole-4-carbonyl}piperidin-4-yl)-2,6-dimethylmorpholine
1-{[1-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}-3-[4-(propan-2-yl)-1H-pyrazol-5-yl]piperidine
N-methyl-5-{[2-(2-methyl-1-benzothiophen-3-yl)-1H-imidazol-1-yl]methyl}furan-2-carboxamide
2-{3-[3-(1H-imidazol-2-yl)piperidine-1-carbonyl]phenyl}-5,6-dimethyl-2,3-dihydro-1H-isoindole
N-[2-(dimethylamino)ethyl]-2-hydroxy-N-[(5-methylthiophen-2-yl)methyl]pyridine-3-carboxamide
8-(2-fluoro-2-phenylacetyl)-2-(2-methylpropyl)-2,8-diazaspiro[4.5]decan-3-one
3-(3-benzyl-1H-1,2,4-triazol-5-yl)-4,5,6,7-tetrahydro-1,2-benzoxazole
N-methyl-3-(4-methyl-4H-1,2,4-triazol-3-yl)-N-{3-[(4-methylphenyl)sulfanyl]propyl}propanamide
N-methyl-N-[(4-oxo-3,4-dihydroquinazolin-2-yl)methyl]-4-(1H-1,2,4-triazol-1-yl)butanamide
1-benzyl-4-oxo-N-(propan-2-yl)-5-(1,2,3,4-tetrahydroisoquinoline-2-carbonyl)-1,4-dihydropyridine-3-carboxamide
1-[6-hydroxy-4-(pyrimidin-2-ylmethyl)-1,4-diazepan-1-yl]-2-[(2-methoxyethyl)(methyl)amino]ethan-1-one
2-(4-{[5-(hydroxymethyl)furan-2-yl]methyl}-1-(thiophen-3-ylmethyl)piperazin-2-yl)ethan-1-ol
N-{[4-amino-6-(dimethylamino)-1,3,5-triazin-2-yl]methyl}-5-(2-chlorophenyl)furan-2-carboxamide
(4aR,7aS)-1-acetyl-4-{[1-(3-methylphenyl)-1H-pyrazol-4-yl]methyl}-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
3-[(3R,4S)-1-(3,5-dichloropyridin-2-yl)-4-(4-methylpiperazin-1-yl)piperidin-3-yl]propanoic acid
N-({2-methylimidazo[2,1-b][1,3]thiazol-6-yl}methyl)-2-(pyrrolidin-1-yl)-6-(thiophen-2-yl)pyridine-3-carboxamide
methyl 5-(cyclobutylamino)-3-(oxolane-2-amido)-1-(3-phenylpropyl)-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
3-{2-[(4-methyl-1,2,5-oxadiazol-3-yl)oxy]ethyl}-1-{4-[(5-methyl-4H-1,2,4-triazol-3-yl)methyl]phenyl}urea
2-(5-acetylthiophen-3-yl)-1-[(3R,4R)-3-{[(2R,6S)-2,6-dimethylmorpholin-4-yl]methyl}-4-(hydroxymethyl)pyrrolidin-1-yl]ethan-1-one
1-[4-(dimethylamino)-2-(pyridin-4-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl]-2-(2-hydroxyphenyl)ethan-1-one
3-propyl-5-[2-(trifluoromethyl)pyrrolidine-1-carbonyl]-1H-pyrazole
4-(2,4-difluorobenzoyl)-6-(pyrrolidin-1-ylmethyl)-1,4-oxazepan-6-ol
2-(2,5-dioxoimidazolidin-1-yl)-N-[3-(2-methyl-1H-imidazol-1-yl)-1-phenylpropyl]acetamide
6-({3-[2-(2-methylphenyl)ethyl]piperidin-1-yl}methyl)-1,2,3,4-tetrahydropyrimidine-2,4-dione
N-cyclopropyl-N-[(1-methyl-1H-imidazol-2-yl)methyl]-2-[1-(3-methylbutyl)-3-oxopiperazin-2-yl]acetamide
methyl({[4-(2-methylphenyl)phenyl]methyl}){[5-(methylsulfanyl)-4-(oxolan-2-ylmethyl)-4H-1,2,4-triazol-3-yl]methyl}amine
6-[3-(2-chlorophenoxy)azetidin-1-yl]-2-methylpyrimidin-4-amine
N-benzyl-1-(2-hydroxyethyl)-5-[(1-methyl-1H-indol-3-yl)methyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
1-[(3R,4R)-4-cyclobutyl-4-hydroxy-3-methylpiperidin-1-yl]-3-(2-hydroxy-4,6-dimethylpyrimidin-5-yl)propan-1-one
N-(1-{1-[2-(cyclohex-1-en-1-yl)acetyl]piperidin-4-yl}-2-phenylethyl)-2-(dimethylamino)-N-methylacetamide
1-{5-hydroxy-1-oxa-9-azaspiro[5.5]undecan-9-yl}-3-(4-methyl-1,3-thiazol-5-yl)propan-1-one
1-{3-[(4-methoxyphenyl)amino]piperidin-1-yl}-2-(pyridin-4-ylsulfanyl)ethan-1-one
2-{[5-(cyclohexylsulfanyl)furan-2-yl]methyl}-2,7-diazaspiro[4.5]decan-6-one
3-[(1S,4R)-2-azabicyclo[2.2.1]heptan-2-yl]-1-{4-[3-(propan-2-yl)-1H-pyrazol-5-yl]piperidin-1-yl}propan-1-one
4-methoxy-N-({1-[2-(methylsulfanyl)acetyl]piperidin-3-yl}methyl)benzene-1-sulfonamide
2-cyclopropyl-9-(2-hydroxyacetyl)-4-phenyl-2,9-diazaspiro[5.5]undecan-3-one
2-(2-methylpropyl)-6-{6-methylthieno[2,3-d]pyrimidin-4-yl}-5H,6H,7H-pyrrolo[3,4-d]pyrimidine
2,6-dihydroxy-N-({1-[(4-methylpiperazin-1-yl)methyl]cyclopropyl}methyl)benzamide
ethyl 4-({4-[(2-fluoro-4-methoxyphenyl)methyl]-3-(2-hydroxyethyl)piperazin-1-yl}methyl)-1H-pyrazole-3-carboxylate
(2S)-2-(methylamino)-1-{8-[(4-methylpiperazin-1-yl)sulfonyl]-1,2,3,4-tetrahydroisoquinolin-2-yl}propan-1-one
4-(4-{[2-(propan-2-yl)pyrimidin-4-yl]methyl}piperazin-1-yl)quinazoline
N-methyl-3-({3-[2-(pyridin-4-yl)pyridin-4-yl]pyrrolidin-1-yl}methyl)pyridin-2-amine
1-(4-{2,3-dimethyl-5-phenylpyrazolo[1,5-a]pyrimidin-7-yl}piperazin-1-yl)ethan-1-one
N-[3-(1H-1,2,3-benzotriazol-1-yl)propyl]-2-ethyl-4-methyl-1,3-thiazole-5-carboxamide
3-(2-{[3-(2-aminoethyl)piperidin-1-yl]methyl}-1H-pyrrol-1-yl)benzonitrile