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6-{1-[5-(1H-imidazol-1-ylmethyl)furan-2-carbonyl]piperidin-3-yl}-2-methylpyrimidin-4-ol
5-ethyl-N4-{[1-(2-methylphenyl)pyrrolidin-3-yl]methyl}pyrimidine-2,4-diamine
(3R,4R)-1-[1-(4-fluoro-2-methylphenyl)piperidin-4-yl]-4-(2-methoxyethyl)-3-methylpiperidin-4-ol
4-ethyl-4-[({[1-(4-methylpiperazin-1-yl)cyclohexyl]methyl}amino)methyl]hexanenitrile
3-propyl-N-{2-[3-(trifluoromethyl)phenyl]ethyl}-1H-pyrazole-5-carboxamide
4-[2-(2-fluorophenyl)ethyl]-3-[1-(1H-pyrazol-1-yl)ethyl]-4,5-dihydro-1H-1,2,4-triazol-5-one
1-(4-oxo-4,5,6,7-tetrahydro-1-benzofuran-3-carbonyl)-4-{[3-(trifluoromethyl)phenyl]methyl}-1,4-diazepan-5-one
N-({3-methyl-7-[4-(1H-pyrazol-1-yl)benzoyl]-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl}methyl)-2-(thiophen-2-yl)acetamide
N-[2-(2,3-dihydro-1,4-benzodioxin-2-yl)ethyl]-6-(3-oxopiperazin-1-yl)pyridine-3-carboxamide
1-{[4-(1H-imidazol-1-yl)phenyl]methyl}-4-(pyridin-3-ylmethyl)-1,4-diazepane
6-[4-(4-benzyl-1H-1,2,3-triazol-1-yl)piperidin-1-yl]-9H-purine
1-[(3,4-difluorophenyl)methyl]-3-hydroxy-3-({methyl[(3-methyl-1,2-oxazol-5-yl)methyl]amino}methyl)piperidin-2-one
N-{[4-(cyclobutylmethoxy)phenyl]methyl}-N-cyclopropyl-2-(dimethyl-1,2-oxazol-4-yl)acetamide
1-[3-(3-methoxyphenoxymethyl)piperidin-1-yl]-2-(1H-pyrazol-1-yl)ethan-1-one
3-({1-[(2E)-3-(furan-2-yl)prop-2-en-1-yl]piperidin-4-yl}oxy)-N-(pyridin-3-ylmethyl)benzamide
3-({dimethyl-[1,3]oxazolo[5,4-d]pyrimidin-7-yl}amino)-2-(thiophen-3-ylmethyl)propan-1-ol
N-[(4-fluorophenyl)methyl]-3-[1-(1H-pyrazole-4-sulfonyl)piperidin-4-yl]propanamide
N-[2-(2-fluorophenyl)ethyl]-3-(2-hydroxyphenyl)-1H-pyrazole-5-carboxamide
1-{[2-chloro-3-(3,4-dimethoxyphenoxy)phenyl]methyl}pyrrolidine
3-{3-[(dimethylamino)methyl]-1,2,4-oxadiazol-5-yl}-N-[(4-fluorophenyl)methyl]aniline
1-{[1-(2-methoxyethyl)-2-(3-methylbutanesulfonyl)-1H-imidazol-5-yl]methyl}-4-phenylpiperazine
3-[1-({5,7-dimethylpyrazolo[1,5-a]pyrimidin-3-yl}methyl)piperidin-2-yl]pyridine
2-methyl-8-(5-propylpyrimidin-4-yl)-2,8-diazaspiro[4.5]decane-3-carboxylic acid
2-amino-4-(2,6-dimethoxyphenyl)-6-(2-methoxyphenyl)pyridine-3-carbonitrile
8-{2-[(dimethylamino)methyl]-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-5-yl}-3,7-dimethyl-2,3,6,7-tetrahydro-1H-purine-2,6-dione
(3R,5S)-5-[3-(naphthalen-1-yl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridine-5-carbonyl]pyrrolidin-3-ol
N-{[5-(methoxymethyl)-1H-pyrazol-3-yl]methyl}-N-methyl-2-(trifluoromethyl)-1H-1,3-benzodiazole-5-carboxamide
5-{1-[(2Z)-2-chloro-3-phenylprop-2-en-1-yl]-4-hydroxypiperidin-4-yl}-N-(oxolan-2-ylmethyl)-1-benzofuran-2-carboxamide
1-(2-methoxyacetyl)-N-{[4-(5-methyl-1,2,4-oxadiazol-3-yl)phenyl]methyl}piperidine-4-carboxamide
8-[3-(5-methyl-1H-1,2,3,4-tetrazol-1-yl)propyl]-3-(2-phenylethyl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
4-{4-[(4-hydroxybutyl)amino]-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-2-yl}benzamide
N-[2-(dimethylsulfamoyl)ethyl]-3-(6-methyl-2-oxo-1,2-dihydropyridin-1-yl)propanamide
4-{[2-(cyclohex-1-en-1-yl)ethyl]amino}-5-methyl-N-(pyridin-2-ylmethyl)thieno[2,3-d]pyrimidine-6-carboxamide
3-{3-[({2H,4H,5H,6H-cyclopenta[c]pyrazol-3-ylmethyl}(methyl)amino)methyl]-1H-indol-1-yl}propanamide
2-(4-chlorophenyl)-N-(3-cyanophenyl)morpholine-4-carboxamide
(2S,4S)-4-(4-cyanobenzamido)-N-ethyl-1-(oxan-4-yl)pyrrolidine-2-carboxamide
1-methyl-2-oxo-8-[3-(1H-1,2,3,4-tetrazol-1-yl)propanoyl]-1,8-diazaspiro[4.5]decane-4-carboxylic acid
N-(prop-2-en-1-yl)-2-{4-[2-(pyridin-4-yl)ethyl]piperazine-1-carbonyl}aniline
N-(6-methoxy-2-methylquinolin-4-yl)quinoxaline-6-carboxamide
5-methyl-3-[2-(piperazin-1-yl)ethyl]-3H,4H-thieno[2,3-d]pyrimidin-4-one
N-[1-(3-ethyl-1,2-oxazol-5-yl)ethyl]imidazo[1,2-a]pyridine-6-carboxamide
4-({1-[(4-fluorophenyl)methanesulfonyl]piperidin-2-yl}methyl)morpholine
4-[5-(morpholin-4-ylmethyl)-1H-1,2,3,4-tetrazol-1-yl]-N-(prop-2-en-1-yl)-N-(prop-2-yn-1-yl)butanamide
N-[4-(morpholin-4-yl)phenyl]-3-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}propanamide
1-(5-chloropyridin-2-yl)-4-[(3-ethyl-4-methyl-1H-pyrazol-5-yl)methyl]piperazine
N,8-dimethyl-N-[1-(3-methylpyridin-2-yl)propan-2-yl]-2-(pyrimidin-5-yl)quinoline-4-carboxamide
5-methyl-4-{[2-(piperidin-1-yl)ethyl]amino}-N-[2-(thiophen-2-yl)ethyl]thieno[2,3-d]pyrimidine-6-carboxamide
1-(5-hydroxypyrazine-2-carbonyl)-3-propylpiperidine-3-carboxylic acid
N4-[(5-ethylpyridin-2-yl)methyl]-N4-methyl-6-(pyrrolidin-1-yl)pyrimidine-2,4-diamine
N-[3-(1H-imidazol-1-yl)propyl]-2-{[1-(pyridin-2-ylmethyl)piperidin-4-yl]oxy}benzamide