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2-[3-(2-hydroxyethyl)-4-(3-phenylpropyl)piperazine-1-carbonyl]phenol
1-[(2-ethylpyrimidin-5-yl)methyl]-8-[5-(trifluoromethyl)pyridin-2-yl]-1,8-diazaspiro[4.5]decane
5-acetyl-N-(6-methoxy-1,3-benzothiazol-2-yl)thiophene-3-carboxamide
1-{5-propyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-yl}-4-(1H-pyrazol-1-yl)butan-1-one
6-ethyl-2-(1-methyl-1H-pyrazol-4-yl)-4-(4-methylpiperidine-1-carbonyl)quinoline
N-[(1,3-dimethyl-1H-pyrazol-5-yl)methyl]-5-fluoroquinazolin-4-amine
N,1,3-trimethyl-N-[2-(oxan-4-yl)ethyl]-1H-pyrazolo[3,4-d][1,3]thiazol-5-amine
{5-[2-(1H-1,3-benzodiazol-2-yl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-5-carbonyl]furan-2-yl}methanol
3-({[2-(2-methylphenyl)-1,3-thiazol-5-yl]methyl}amino)-2,3-dihydro-1λ6-thiophene-1,1-dione
6-fluoro-2-{[4-(pyridin-4-ylmethyl)piperazin-1-yl]methyl}quinolin-4-ol
4-(4-chlorophenyl)-1-{[5-(4-fluorophenyl)-2-hydroxyphenyl]methyl}piperidin-4-ol
3-{[(1H-1,3-benzodiazol-2-ylmethyl)(methyl)amino]methyl}-1-(2,2-dimethylpropyl)-3-hydroxypiperidin-2-one
3-(2-{7-cyclopentyl-6-oxo-2,7-diazaspiro[4.5]decan-2-yl}-2-oxoethyl)imidazolidine-2,4-dione
N-(2-methoxyethyl)-1,3-dimethyl-N-[(1-methyl-1H-pyrazol-4-yl)methyl]-1H-pyrazolo[3,4-d][1,3]thiazol-5-amine
N,N-dimethyl-2-[(naphthalen-1-ylformamido)methyl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-5-carboxamide
3,5-dichloro-4-methyl-N-[2-(pyrrolidine-1-sulfonyl)ethyl]benzamide
3-{[2-(furan-3-yl)-1H-imidazol-1-yl]methyl}-4-(2-methoxyethyl)-4H-1,2,4-triazole
N-{1-[5-(2,4-difluorophenoxymethyl)-1,2-oxazole-3-carbonyl]pyrrolidin-3-yl}acetamide
1-{4-[4-(2-aminopropan-2-yl)-1H-1,2,3-triazol-1-yl]piperidin-1-yl}-2,2-dimethylpropan-1-one
4-phenoxy-1-{thieno[2,3-d]pyrimidin-4-yl}piperidine-4-carboxylic acid
N6-(3-methoxypropyl)-N5-methyl-N5-(2-phenoxyethyl)-[1,2,5]oxadiazolo[3,4-b]pyrazine-5,6-diamine
3-ethyl-N-[(3R,4S)-1-(oxan-4-yl)-4-propylpyrrolidin-3-yl]-1,2-oxazole-5-carboxamide
methyl({[1-(2-methylpropyl)-2-(oxolan-2-ylmethanesulfonyl)-1H-imidazol-5-yl]methyl})(thiophen-2-ylmethyl)amine
5-(3-methoxypropanoyl)-1-(pyridin-2-ylmethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylic acid
3-{[(dimethyl-1,3-thiazol-2-yl)methyl]sulfamoyl}-N-propylbenzamide
3-{[2-(4-fluorophenyl)pyrrolidin-1-yl]methyl}pyridin-2-amine
1-[2-(cyclopent-2-en-1-yl)acetyl]-4-(1H-pyrazol-1-yl)piperidine-4-carboxylic acid
5-(3-cyclopropyl-1-phenyl-1H-1,2,4-triazol-5-yl)-N-ethylpyrimidin-2-amine
N-[(2S,4R,6S)-2-(2-butyl-1H-imidazol-4-yl)-6-(2-methylpropyl)oxan-4-yl]acetamide
(4S,4aS,8aS)-4-phenyl-1-[1-(propan-2-yl)-1H-pyrazole-4-carbonyl]-decahydroquinolin-4-ol
2-[4-(4-benzyl-5-oxo-4,5-dihydro-1H-1,2,4-triazol-3-yl)piperidin-1-yl]pyridine-4-carbonitrile
4-[(4,6-dimethylpyrimidin-2-yl)amino]-1-(2-methoxyphenyl)pyrrolidin-2-one
3-[1-(cyclohex-1-ene-1-carbonyl)piperidin-3-yl]-N-methyl-N-[2-(pyridin-2-yl)ethyl]propanamide
3-({6-tert-butyl-1-methyl-1H-pyrazolo[3,4-d]pyrimidin-4-yl}amino)-2,3-dihydro-1λ6-thiophene-1,1-dione
2-[4-(2-amino-6-methylpyrimidin-4-yl)-6-hydroxy-1,4-diazepan-1-yl]-1-(piperazin-1-yl)ethan-1-one
1-benzyl-4-(1-ethyl-1H-pyrazole-4-carbonyl)-6-(pyridin-3-ylmethoxy)-1,4-diazepan-2-one
4-phenyl-3-({1-[2-(1,2,3,6-tetrahydropyridin-4-yl)acetyl]piperidin-4-yl}methyl)-4,5-dihydro-1H-1,2,4-triazol-5-one
(3S,4S)-4-(2H-1,3-benzodioxol-5-yl)-1-(6-ethyl-2-methylpyrimidin-4-yl)piperidin-3-ol
N-[(5-{[(2-chlorophenyl)methyl]sulfanyl}-4-(2-methylpropyl)-4H-1,2,4-triazol-3-yl)methyl]furan-3-carboxamide
methyl 2-[benzyl(methyl)sulfamoyl]-6-(3-methylbenzoyl)-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
(2R)-1-{[5-(4-chloro-2-fluorophenyl)furan-2-yl]methyl}pyrrolidine-2-carboxamide
4-ethyl-3-{1-[(4-methyl-2-oxo-2H-chromen-7-yl)methyl]piperidin-4-yl}-4,5-dihydro-1H-1,2,4-triazol-5-one
N-methyl-N-[(4-methyl-1H-imidazol-2-yl)methyl]-3-phenoxybenzamide
1-(2-{[5-(methoxymethyl)furan-2-yl]formamido}ethyl)piperidine-3-carboxamide
(3S,4R)-3-methoxy-1-[2-(1H-1,2,4-triazol-1-yl)benzoyl]piperidin-4-amine
1-[3-(4-benzyl-1H-pyrazol-5-yl)piperidin-1-yl]-4-methylpentane-1,2-dione
2-(2H-1,3-benzodioxol-5-yl)-N-(2,3,4,9-tetrahydro-1H-carbazol-6-ylmethyl)acetamide
2-{[(5-tert-butyl-1H-pyrazol-3-yl)methyl](thiophen-3-ylmethyl)amino}butan-1-ol
(3S)-3-ethyl-4-[(2E)-3-(4-methoxyphenyl)prop-2-en-1-yl]morpholine
3-(1-ethyl-1H-imidazol-2-yl)-1-[1-(2-methoxyphenyl)-1H-pyrazole-4-carbonyl]piperidine