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9-(2-methoxyethyl)-1-methyl-4-[3-(methylsulfanyl)propyl]-1,4,9-triazaspiro[5.6]dodecan-10-one
4-[4-(pyrrolidine-1-carbonyl)piperidin-1-yl]-10-oxa-5,7-diazatricyclo[9.4.0.03,8]pentadeca-1(11),3,5,7,12,14-hexaene
1-{1-[(3-fluorophenyl)methyl]-6-oxopiperidine-3-carbonyl}-4-(piperidin-1-yl)piperidine-4-carboxamide
8-cyclopropanecarbonyl-2-(1-methyl-1H-pyrrole-2-carbonyl)-2,8-diazaspiro[4.5]decane-3-carboxylic acid
4-[4-(dimethylamino)-2-(pyridin-4-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl]-4-oxobutanamide
8-fluoro-N-{[2-(1H-pyrazol-1-ylmethyl)phenyl]methyl}quinoline-2-carboxamide
3-(2,4-dichlorophenyl)-2,5-dimethylpyrazine
2-[4-(pyridin-2-ylmethoxy)piperidin-1-yl]-4-(pyridin-3-yl)pyrimidine
11-[4-(cyclopropylamino)-5-methylthieno[2,3-d]pyrimidine-6-carbonyl]-7,11-diazatricyclo[7.3.1.02,7]trideca-2,4-dien-6-one
5,5-dimethyl-3-{[4-(propan-2-yl)-4H-1,2,4-triazol-3-yl]methyl}-1,3-oxazolidine-2,4-dione
5-ethyl-5-[1-(3-ethyl-5-methyl-1,2-oxazole-4-carbonyl)piperidin-4-yl]imidazolidine-2,4-dione
5-chloro-3-methyl-N-[2-(3-{[methyl(1,3-thiazol-4-ylmethyl)amino]methyl}phenoxy)propyl]-1H-indole-2-carboxamide
4-[(4-{4-ethyl-5-[(2-methyl-1H-imidazol-1-yl)methyl]-4H-1,2,4-triazol-3-yl}piperidin-1-yl)methyl]pyridine
2-[5-(2-ethylpyridin-4-yl)-1-(3-fluorophenyl)-1H-1,2,4-triazol-3-yl]acetamide
N-cyclohexyl-3-{3'-oxo-3',4'-dihydro-1'H-spiro[piperidine-4,2'-quinoxaline]-1-yl}propanamide
1-{2-[5-(1-methyl-1H-indol-2-yl)-4-phenyl-1H-imidazol-1-yl]ethyl}piperidin-3-ol
1-(2,6-dimethoxypyrimidin-4-yl)-2-methyl-1,4-diazepan-5-one
{1-[2-(2-chloro-4-methylphenoxy)ethyl]-3-(prop-2-en-1-yl)piperidin-3-yl}methanol
2-[2-(cyclohexyloxy)ethyl]-7,7-dimethyl-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-4-one
methyl 5-[1-(2-methylpropyl)-5-oxopyrrolidine-3-carbonyl]-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-2-carboxylate
5-{[3-(4-chlorophenyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]methyl}-N-ethylpyrimidin-2-amine
N-[(3R,4S)-4-cyclopropyl-1-(3-fluoropyridin-4-yl)pyrrolidin-3-yl]methanesulfonamide
N-[2-(3-{[methyl(pyrazin-2-ylmethyl)amino]methyl}phenoxy)propyl]furan-2-carboxamide
1-[(2-butyl-5-chloro-1H-imidazol-4-yl)methyl]-3-(1-methyl-1H-imidazole-2-carbonyl)piperidine
N-[1-(1H-imidazol-1-yl)-3,3-dimethylbutan-2-yl]-1-methyl-2-oxo-1,2-dihydroquinoline-3-carboxamide
2-{3-[3-(2-cyclopropyl-1,3-benzoxazol-5-yl)phenyl]-1H-pyrazol-1-yl}ethan-1-ol
5-methoxy-2-[4-(4-methyl-1H-1,3-benzodiazol-2-yl)piperidine-1-carbonyl]-4H-pyran-4-one
N-{[2-(1H-1,3-benzodiazol-1-yl)pyridin-3-yl]methyl}-1-ethyl-3-methylpiperidine-3-carboxamide
1,3-dimethyl-N-{1-[3-(2-methylpropyl)-1,2,4-oxadiazol-5-yl]ethyl}-2,6-dioxo-1,2,3,6-tetrahydropyrimidine-4-carboxamide
N,1-dimethyl-N-{[2-(2-methylpropoxy)phenyl]methyl}-3-(trifluoromethyl)-1H-pyrazole-5-carboxamide
(4aR,7aS)-1-methyl-4-{[3-(1H-pyrazol-1-yl)phenyl]methyl}-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
4-cyclohexanecarbonyl-9-methoxy-7-(quinolin-3-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepine
3-methanesulfonamido-N-methyl-N-(quinolin-5-ylmethyl)propanamide
3-[(3R,4S)-1-(benzenesulfonyl)-4-(morpholin-4-yl)piperidin-3-yl]propanoic acid
1-(2-hydroxyethyl)-N-[2,2,2-trifluoro-1-(pyridin-3-yl)ethyl]-1H-1,3-benzodiazole-5-carboxamide
N-[(2,4-dimethoxyphenyl)methyl]-3-[1-(thiophene-3-carbonyl)piperidin-3-yl]propanamide
N-{[5-(4-methoxyphenyl)-1,2-oxazol-3-yl]methyl}-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
1-({1-[1-(propan-2-yl)-1H-pyrazole-4-carbonyl]piperidin-3-yl}methyl)-1H-1,2,3-triazole-4-carboxylic acid
1-(4-benzylpiperazine-1-carbonyl)-6-(2-methoxypyridine-3-carbonyl)-6-azaspiro[2.5]octane
5-cyclopropanecarbonyl-1'-[(1-ethyl-1H-pyrazol-4-yl)methyl]-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
N-({5-cyclohexyl-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}methyl)-9H-purin-6-amine
N-cyclopentyl-N-{[4-methoxy-3-(thiophen-2-ylmethoxy)phenyl]methyl}-1-methyl-4-oxo-1,4-dihydroquinoline-3-carboxamide
4-{[6-(4-fluorophenyl)pyridin-3-yl]methyl}morpholine
1-[1-(1,3-thiazol-2-ylmethyl)piperidin-3-yl]pyrrolidin-2-one
(3S,4R)-4-(hydroxymethyl)-1-[3-(trifluoromethyl)-1H-pyrazole-5-carbonyl]piperidin-3-ol
5-{[1-(2-methoxyacetyl)pyrrolidin-3-yl]methyl}-1,2-dihydropyridin-2-one
N-[(1-{[5-(methoxymethyl)furan-2-yl]methyl}piperidin-3-yl)methyl]-4-phenylbenzamide
(2S,4S,5R)-5-(2-fluorophenyl)-4-{[2-(4-hydroxyphenyl)ethyl]carbamoyl}-1-methylpyrrolidine-2-carboxylic acid
N-benzyl-1-methyl-5-(pyridin-2-ylmethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
1-{2-[3-(2,3-dimethylphenyl)-1,2,4-oxadiazol-5-yl]ethyl}-1H-1,2,3,4-tetrazole