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N-benzyl[(6-cyanopyridin-3-yl)amino]sulfonamide
6-(methoxymethyl)-N-[(4-methyl-1,3-benzoxazol-2-yl)methyl]pyrimidin-4-amine
1-(2-methylpropyl)-3-(morpholine-4-carbonyl)-N-[3-(propan-2-yloxy)propyl]-4,5,6,7-tetrahydro-1H-indazol-5-amine
2-methyl-N-{1-[3-(2-methylpropyl)-1,2,4-oxadiazol-5-yl]ethyl}-1,3-benzoxazole-6-carboxamide
N-methyl-N-[(2-methyl-1,3-thiazol-4-yl)methyl]-2-[4-(4-methyl-1,4-diazepan-1-yl)-6-oxo-1,6-dihydropyridazin-1-yl]acetamide
N4-[3-(5-cyclopropyl-1H-pyrazol-1-yl)propyl]-N2,N2-dimethyl-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepine-2,4-diamine
1-{1-[(3-methylphenyl)methyl]piperidin-4-yl}-3-(pyrrolidine-1-carbonyl)piperidine
3-(1H-imidazol-1-yl)-6-{1-methyl-1H-pyrrolo[2,3-b]pyridin-4-yl}pyridazine
(2R,3R,6R)-5-[(dimethyl-1,2-oxazol-4-yl)sulfonyl]-3-phenyl-1,5-diazatricyclo[5.2.2.02,6]undecane
8-[(5-cyclopropyl-1,2,4-oxadiazol-3-yl)methyl]-2-(3-methoxypropyl)-2,8-diazaspiro[5.5]undecan-3-one
2-(4-chloro-2-methylphenoxy)-1-[4-(pyridin-4-yl)piperidin-1-yl]ethan-1-one
N-[1-(3,5-difluorophenyl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]-2-(1-methylpiperidin-4-yl)acetamide
4-({[2-(3,5-dimethyl-1H-pyrazol-1-yl)ethyl]carbamoyl}amino)-N-(oxolan-2-ylmethyl)benzamide
1-cyclohexyl-N-(1-{imidazo[1,2-a]pyrimidin-2-yl}propyl)piperidine-4-carboxamide
ethyl 2-{4-[(4-methylphenyl)methyl]-3-oxopiperazin-1-yl}-1,3-oxazole-4-carboxylate
(3S,4S)-1-{2-[(cyclopropylmethyl)sulfanyl]acetyl}-4-(pyridin-2-yl)pyrrolidine-3-carboxylic acid
N-[3-(4-{[3-(4-fluorophenyl)-3-(furan-2-yl)propyl]amino}piperidin-1-yl)phenyl]pyridine-4-carboxamide
3-[1-(2,2-dimethyl-4-oxo-3,4-dihydro-2H-pyran-6-carbonyl)piperidin-3-yl]-N-[(2-fluorophenyl)methyl]propanamide
4-(4-acetyl-1,4-diazepane-1-carbonyl)-1-(pyridin-3-ylmethyl)pyrrolidin-2-one
1-[3-(4-methyl-1H-1,3-benzodiazol-2-yl)piperidin-1-yl]-3-(1-methyl-1H-pyrazol-4-yl)propan-1-one
3-[1-(2-amino-4-methyl-1,3-thiazole-5-carbonyl)piperidin-4-yl]-N-(3-methylphenyl)propanamide
1-(3,3-dimethyl-4-phenylpyrrolidine-1-carbonyl)cyclopropane-1-carboxamide
5-(1,3-benzothiazol-2-yl)-N-(2-hydroxyethyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-2-carboxamide
3-[(2E)-3-phenylprop-2-en-1-yl]-1-(pyrimidin-2-yl)piperidine-3-carboxylic acid
1-{[(3-chloro-2-propoxyphenyl)carbamoyl]amino}cyclopentane-1-carboxamide
2-methyl-4-(1-{[1-(phenoxymethyl)cyclopropyl]methyl}-1H-imidazol-2-yl)-1,3-oxazole
2-{4-[(4-aminoazepan-1-yl)methyl]phenoxy}-1-(pyrrolidin-1-yl)ethan-1-one
(1R,2R,6S,7S)-4-[5-fluoro-4-(morpholin-4-yl)pyrimidin-2-yl]-10-oxa-4-azatricyclo[5.2.1.02,6]decane
3-[3-(dimethyl-1,2-oxazol-4-yl)propyl]-1-[2-methyl-5-(5-methyl-1,3,4-oxadiazol-2-yl)phenyl]urea
N-(1-methoxypropan-2-yl)-1-{5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-yl}piperidine-4-carboxamide
1-cyclobutyl-3-(3-methoxybenzoyl)piperidine
1-[(3-cyclopropyl-1H-pyrazol-5-yl)methyl]-4-(5-methyl-1,2,4-oxadiazol-3-yl)-1,4-diazepan-6-ol
N-(2-ethoxyethyl)-3-(4-methyl-5-oxo-1,4-diazepane-1-carbonyl)benzene-1-sulfonamide
4-{[4-(2,6-difluorophenyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl]methyl}-2-(propan-2-yl)pyrimidine
5-(2-fluorophenoxymethyl)-N-(2-oxopyrrolidin-3-yl)-1H-pyrazole-3-carboxamide
1-(carbamoylmethyl)-N-ethyl-N-(pyridin-4-ylmethyl)piperidine-3-carboxamide
2-butyl-5-[4-(4-methylphenoxy)piperidine-1-carbonyl]-1,3-benzoxazole
5-[(1,5-dimethyl-1H-pyrazol-4-yl)methyl]-2-(3-fluorophenyl)-8-methoxy-2,3,4,5-tetrahydro-1,5-benzothiazepine
N-[1-(1-{[1-(pyridin-3-yl)-1H-pyrrol-2-yl]methyl}piperidin-4-yl)-1H-pyrazol-5-yl]benzamide
N-cyclopentyl-3-{methyl[(1-methyl-1H-pyrazol-4-yl)methyl]sulfamoyl}benzamide
methyl 2-{[4-(4-methoxyphenyl)-2-methyl-3-oxopiperazine-1-carbonyl]amino}acetate
5,7-dimethyl-N-[(4-propyl-4H-1,2,4-triazol-3-yl)methyl]pyrazolo[1,5-a]pyrimidine-2-carboxamide
ethyl 1-[(3-chloro-4-hydroxyphenyl)methyl]-4-{[3-(trifluoromethyl)phenyl]methyl}piperidine-4-carboxylate
4-[4-cyclopropyl-5-(1H-imidazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]-1-[(trimethyl-1H-imidazol-2-yl)methyl]piperidine
2,6-dimethyl-5-{2-[(1S,5R)-3-(oxan-4-yl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]-2-oxoethyl}-3,4-dihydropyrimidin-4-one
5-[(4aS,8aR)-decahydroisoquinoline-2-carbonyl]-1-[(5-methylfuran-2-yl)methyl]-4-oxo-N-(prop-2-en-1-yl)-1,4-dihydropyridine-3-carboxamide
1-[2-(azepan-1-yl)-2-oxoethyl]-3-(3-methoxypropyl)piperidine-3-carboxylic acid
N-[2-(dimethylamino)-5,6,7,8-tetrahydroquinazolin-5-yl]-2-(2-oxoazepan-1-yl)acetamide
2-[(1R,3S,3aS,6aR)-5-ethyl-1-(hydroxymethyl)-3-(7-methoxy-2H-1,3-benzodioxol-5-yl)-octahydropyrrolo[3,4-c]pyrrol-1-yl]ethan-1-ol
1-cyclopropyl-6-oxo-N-[(5-phenyl-1,2,4-oxadiazol-3-yl)methyl]piperidine-3-carboxamide