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4-{2-methyl-1-[4-(1,2,4-oxadiazol-3-yl)piperidin-1-yl]propan-2-yl}morpholine
[1-(1H-1,3-benzodiazol-2-ylmethyl)pyrrolidin-3-yl]methanamine
2-[3-(2,5-difluorophenyl)phenoxy]acetamide
8-{6-cyclopropyl-3-methyl-[1,2]oxazolo[5,4-b]pyridine-4-carbonyl}-1-oxa-8-azaspiro[4.5]decane
(4-{[1-(6-methoxy-1-methyl-1H-indole-2-carbonyl)pyrrolidin-3-yl]methyl}phenyl)methanol
N-[(3R,4R)-3-hydroxy-1-[2-(pyridin-2-yl)acetyl]piperidin-4-yl]pyridine-4-carboxamide
1-(4-ethyl-1,2,3-thiadiazole-5-carbonyl)-4-(5-methylpyridin-2-yl)piperidin-4-ol
8-[2-(3,4-dimethyl-6-oxo-1,6-dihydropyridazin-1-yl)acetyl]-2-(3-methylbutyl)-2,8-diazaspiro[5.5]undecan-3-one
5-({4-[(4-chlorophenyl)methyl]piperazin-1-yl}methyl)-2-(pyridin-2-yl)pyrimidine
3-[(3R,4R)-3-(hydroxymethyl)-4-{[(2-methoxyethyl)(methyl)amino]methyl}pyrrolidine-1-carbonyl]-6-methyl-1,4-dihydroquinolin-4-one
N-[(3,4-difluorophenyl)methyl]-3-[1-(4-formylbenzoyl)piperidin-3-yl]propanamide
2-[(1S,5R)-3-(pyrazine-2-carbonyl)-3,6-diazabicyclo[3.2.2]nonane-6-carbonyl]pyridin-3-ol
7-cyclopentyl-2-(4-propyl-1,2,3-thiadiazole-5-carbonyl)-2,7-diazaspiro[4.5]decan-6-one
2-(3-{[4-(6-methylpyridazin-3-yl)piperazin-1-yl]methyl}-1H-indol-1-yl)acetamide
1-(4-benzyl-4-hydroxypiperidin-1-yl)-2-[5-(pyrrolidin-1-ylmethyl)-1H-1,2,3,4-tetrazol-1-yl]ethan-1-one
3-{imidazo[1,2-a]pyridin-2-yl}-N-{2H,3H-imidazo[2,1-b][1,3]thiazol-6-ylmethyl}propanamide
N-[(5-methyl-1,2-oxazol-3-yl)methyl]-3-(1-methyl-1H-pyrrol-2-yl)-1H-pyrazole-5-carboxamide
3-(1H-imidazol-2-yl)-N-[(2,3,4-trifluorophenyl)methyl]benzamide
N-{[2-(2,3-difluoro-4-methylphenoxy)pyridin-3-yl]methyl}-2-(4-methyl-1,2,5-oxadiazol-3-yl)acetamide
N-{[2-(2-methyl-1H-imidazol-1-yl)phenyl]methyl}-1,2,3,4-tetrahydronaphthalen-2-amine
1-(2-methanesulfonylethyl)-4-(3-phenyl-1H-pyrazole-4-carbonyl)piperazine
N-[(5-cyclopropyl-1H-pyrazol-3-yl)methyl]-5-(2-methoxyphenoxymethyl)-N-methyl-1H-pyrazole-3-carboxamide
N-[(1-benzyl-1H-imidazol-2-yl)methyl]-5-methyl-4-(1-methyl-1H-pyrazol-5-yl)pyrimidin-2-amine
(1S,5R)-3-methyl-6-[(5-methylthiophen-2-yl)methyl]-3,6-diazabicyclo[3.2.2]nonane
1-[1-(2,3-dihydro-1H-inden-2-yl)piperidin-4-yl]-N-(2-ethoxyethyl)piperidine-3-carboxamide
2-{4-[2-(pyrrolidin-1-ylmethyl)-1,4-oxazepane-4-carbonyl]-1H-1,2,3-triazol-1-yl}ethan-1-amine
2-(4-benzyl-2-oxopyrrolidin-1-yl)-N-methyl-N-(2-phenylethyl)acetamide
2-(5-amino-1,3,4-thiadiazol-2-yl)-1-{4-[3-(propan-2-yl)-1H-pyrazol-5-yl]piperidin-1-yl}ethan-1-one
4-methoxy-2-({3-[4-(piperidine-1-carbonyl)-1H-1,2,3-triazol-1-yl]piperidin-1-yl}methyl)phenol
6-(aminomethyl)-N-[1-(1H-pyrazol-1-yl)propan-2-yl]pyrimidin-4-amine
2,3-dimethyl-5-(4-{4-methyl-5-[(4-methylpiperazin-1-yl)methyl]-4H-1,2,4-triazol-3-yl}piperidin-1-yl)pyrazine
1-[(2S,4R)-4-(1H-1,2,3,4-tetrazol-1-yl)-1-{[4-(trifluoromethyl)phenyl]methyl}pyrrolidine-2-carbonyl]azepane
[3-ethyl-1-(7-methoxy-4-methylquinazolin-2-yl)piperidin-3-yl]methanol
N-(5-oxo-1-{[2-(trifluoromethyl)phenyl]methyl}pyrrolidin-3-yl)-2-(2-oxopyrrolidin-1-yl)acetamide
(3aS,6aR)-5-(6-aminopyrimidin-4-yl)-3-[3-(morpholin-4-yl)propyl]-hexahydro-2H-pyrrolo[3,4-d][1,3]oxazol-2-one
methyl 5-(4-acetamidobenzenesulfonyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-2-carboxylate
6-(3-methoxy-5-methylthiophene-2-carbonyl)-2-(2-methylpropyl)-5H,6H,7H-pyrrolo[3,4-d]pyrimidine
(2R,3S,6R)-3-(2,3-difluorophenyl)-N-ethyl-1,5-diazatricyclo[5.2.2.02,6]undecane-5-carboxamide
6-{3-[4-(4-fluorophenyl)piperazin-1-yl]piperidin-1-yl}pyridine-3-carbonitrile
1-[(5-cyclopentylthiophen-2-yl)methyl]azepan-4-ol
N-{[3-(pyridin-2-yl)-1,2-oxazol-5-yl]methyl}-2-(pyridin-3-yl)-2-(pyrrolidin-1-yl)acetamide
5-(5-{[3-(2-methylpropyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]methyl}furan-2-yl)-1H-pyrazole
5-(3-methoxyphenoxymethyl)-N-methyl-N-(propan-2-yl)-1,2-oxazole-3-carboxamide
methyl 1-[(3S,5S)-5-{[2-(4-fluorophenyl)ethyl]carbamoyl}-1-(3-methylbut-2-en-1-yl)pyrrolidin-3-yl]-1H-1,2,3-triazole-4-carboxylate
(2S)-2-{2-cyclopropyl-3-oxo-2,9-diazaspiro[5.5]undecane-9-carbonyl}pyrrolidine-1-carboxamide
N-[2-(4-methylmorpholin-2-yl)ethyl]-3-(3-methylphenyl)-1H-pyrazole-4-carboxamide
6-[(3-hydroxypropyl)amino]-N-{[5-(propan-2-yl)-1,2,4-oxadiazol-3-yl]methyl}pyridine-3-carboxamide
3-(2,4-dimethoxybenzoyl)-1-(1,2-oxazol-3-ylmethyl)piperidine
2-cyclopropyl-6-oxo-N-[1-(pyridin-2-ylmethyl)piperidin-4-yl]-1,6-dihydropyrimidine-5-carboxamide
N-[(4-sulfamoylphenyl)methyl]pyrazolo[1,5-a]pyridine-7-carboxamide