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4,6-dimethyl-1-{2-[(3-methylpyrazin-2-yl)amino]ethyl}-1,2-dihydropyrimidin-2-one
1-(4-chlorophenyl)-N-{[1-(3-methylbut-2-en-1-yl)piperidin-3-yl]methyl}cyclopropane-1-carboxamide
3-chloro-4-[(1-cyclopropanecarbonylpiperidin-4-yl)oxy]-N-[2-(dimethylamino)ethyl]benzamide
N-{1-[2-(4-methoxyphenyl)ethyl]-5-oxopyrrolidin-3-yl}-2-methylfuran-3-carboxamide
3-[3-(1-benzyl-1H-imidazol-2-yl)piperidine-1-carbonyl]pyridine
2-(1-{[3-(diphenylmethyl)-1,2,4-oxadiazol-5-yl]methyl}piperidin-3-yl)-1H-1,3-benzodiazole
N-(cyclopropylmethyl)-2-{1-[(2E)-3-(2-methoxyphenyl)prop-2-en-1-yl]-3-oxopiperazin-2-yl}acetamide
N-[2-(4,6-dimethyl-2-oxo-1,2-dihydropyrimidin-1-yl)ethyl]-5-methyl-4,5,6,7-tetrahydro-1-benzothiophene-2-carboxamide
[(3R,4R)-4-{[(2R,6S)-2,6-dimethylmorpholin-4-yl]methyl}-1-{5-[(methylsulfanyl)methyl]furan-2-carbonyl}pyrrolidin-3-yl]methanol
3-({[(5-chlorothiophen-2-yl)methyl]amino}methyl)-1-(2,2-dimethylpropyl)-3-hydroxypiperidin-2-one
ethyl 1-[(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)methyl]-4-[(3-methoxyphenyl)methyl]piperidine-4-carboxylate
(3aS,6aS)-2-(ethanesulfonyl)-5-[5-(ethylcarbamoyl)pyridin-2-yl]-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
N1,N1-dimethyl-N4,N4-bis(1,3-oxazol-4-ylmethyl)piperidine-1,4-dicarboxamide
(3S,4R)-1-[2-(cyclopentylcarbamoyl)ethyl]-4-phenylpyrrolidine-3-carboxylic acid
(3S,4R)-1-{[4-(3-hydroxyprop-1-yn-1-yl)thiophen-2-yl]methyl}-4-phenylpyrrolidine-3-carboxylic acid
3-(5-fluoro-1H-1,3-benzodiazol-2-yl)-1-[4-(3-methylpyridin-2-yl)piperazin-1-yl]propan-1-one
N-[2-(methylsulfamoyl)ethyl]-1-benzothiophene-5-carboxamide
4-[4-ethyl-5-(pyrrolidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]-1-(2-phenylethyl)piperidine
1-[(2-fluorophenyl)methyl]-6-oxo-N-[2-(pyridin-2-yl)ethyl]piperidine-3-carboxamide
N'-(3-ethylphenyl)-N-(3-hydroxy-2,2-dimethylpropyl)butanediamide
1-benzyl-N-[2-(3-methoxyphenyl)phenyl]piperidine-4-carboxamide
1-(furan-2-ylmethyl)-N-[(7-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]piperidin-4-amine
N-(1-{7-[(3-methoxyphenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}-3-methylbutyl)pyridine-3-carboxamide
1-[4-(4-ethyl-1H-pyrazol-5-yl)piperidin-1-yl]-2-(3-methoxyphenyl)ethan-1-one
3-[2-(3,4-dimethoxyphenyl)ethyl]-5-methyl-5-(piperidin-4-yl)imidazolidine-2,4-dione
5,7-dimethyl-N-(oxan-3-ylmethyl)pyrido[2,3-d]pyrimidin-4-amine
3-{3-[4-(2-methylphenyl)piperazin-1-yl]piperidine-1-carbonyl}-1H-indazole
6-{[(4aS,7aR)-4-(2-methoxyethyl)-6,6-dioxo-octahydro-6λ6-thieno[3,4-b]piperazin-1-yl]methyl}-1,2,3,4-tetrahydropyrimidine-2,4-dione
5-acetyl-N-[(2-chlorophenyl)methyl]-N-(2-methoxyethyl)thiophene-3-carboxamide
4,4-difluoro-1-{[2-(pyrrolidin-1-yl)-1,3-thiazol-5-yl]methyl}piperidine
1-methyl-N-(2-phenoxyethyl)-3-(trimethyl-1H-pyrazol-4-yl)-1H-pyrazole-5-carboxamide
2-(7-fluoro-2-methyl-1H-indol-3-yl)-N-{2-[(1-methyl-1H-1,2,3,4-tetrazol-5-yl)sulfanyl]ethyl}acetamide
2-[2-(4-ethoxyphenoxymethyl)pyrimidin-4-yl]pyridine-4-carboxylic acid
N4-[2-(diethylamino)ethyl]-5-ethyl-6-methylpyrimidine-2,4-diamine
3-[(2R,3R,6R)-5-(4-ethylbenzoyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-3-yl]phenol
N-[2-(2-methyl-1H-indol-3-yl)ethyl]-2-[5-(pyrrolidin-1-ylmethyl)-1H-1,2,3,4-tetrazol-1-yl]acetamide
1-{[1-(2,5-dimethylphenyl)-3-phenyl-1H-pyrazol-4-yl]methyl}-3-(4-methyl-4H-1,2,4-triazol-3-yl)piperidine
5-methoxy-2-({4-[4-methyl-5-(1H-pyrazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}methyl)-4H-pyran-4-one
N-cyclopentyl-2-{1-[(3,5-dimethoxyphenyl)methyl]-3-oxopiperazin-2-yl}acetamide
2-(dimethylamino)-2-(4-methylphenyl)-1-[4-(pyridin-4-yl)piperazin-1-yl]ethan-1-one
1-[2-amino-7-methyl-4-(pyridin-4-yl)-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-6-yl]-2-(2-methylphenyl)ethan-1-one
3-(1H-imidazol-1-ylmethyl)-1-{[3-(1H-pyrazol-1-yl)phenyl]methyl}piperidine
2,6-diamino-4-(5-chloro-2,3-dimethoxyphenyl)-5,6,7,8-tetrahydroquinoline-3-carbonitrile
2-[3-cyclopropyl-1-(2-methylpyridin-4-yl)-1H-1,2,4-triazol-5-yl]-3,5-difluoropyridine
3-{1-[(1-cycloheptanecarbonylpiperidin-4-yl)methyl]-1H-1,2,3-triazol-4-yl}propan-1-ol
4-{2-[4-(hydroxymethyl)phenyl]acetyl}-1-methyl-1,4,9-triazaspiro[5.6]dodecan-10-one
N-{1-[5-methyl-1-(2-methylphenyl)-1H-pyrazol-4-yl]ethyl}thiophene-3-sulfonamide
1-{2-[(6-methyl-2-propylpyrimidin-4-yl)amino]ethyl}-1,2,3,6-tetrahydropyridazine-3,6-dione
2-(4-methanesulfonylmorpholin-2-yl)-7,7-dimethyl-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-4-one
({7-fluoro-2-[2-(phenylsulfanyl)ethoxy]quinolin-3-yl}methyl)[(5-methylpyrazin-2-yl)methyl]amine