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N-cyclohexyl-1-oxo-N-(pyridin-2-ylmethyl)-1,2-dihydroisoquinoline-4-carboxamide
N,N,4-trimethyl-3-[({[1,2,4]triazolo[4,3-a]pyridin-8-yl}carbamoyl)methyl]-3,4-dihydro-2H-1,4-benzoxazine-6-carboxamide
(3R,5S)-N-(2-phenylethyl)-1-(pyridin-4-ylmethyl)-5-[3-(trifluoromethyl)phenoxymethyl]piperidine-3-carboxamide
1-(2-chloro-5-fluorophenyl)-3-[(5-cyclopentyl-1,2,4-oxadiazol-3-yl)methyl]-3-methylurea
(1R,5R)-6-({7-chloro-4-oxo-4H-pyrido[1,2-a]pyrimidin-2-yl}methyl)-N,N-dimethyl-3,6-diazabicyclo[3.2.2]nonane-3-carboxamide
butyl 4-oxo-2-(pyridin-4-yl)-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidine-7-carboxylate
2-(5-methyl-1H-pyrazol-1-yl)-1-[4-(1,2,3,4-tetrahydronaphthalen-2-yl)piperazin-1-yl]ethan-1-one
({6-chloro-2-[(2R,6S)-2,6-dimethylmorpholine-4-carbonyl]imidazo[1,2-a]pyridin-3-yl}methyl)[2-(2-fluorophenyl)ethyl]amine
N-{2-[9-oxo-8-(2-phenylethyl)-2,8-diazaspiro[5.5]undecan-2-yl]ethyl}acetamide
6-(2,4-dimethoxypyrimidin-5-yl)quinoline
2-[1-(4-methoxyphenyl)cyclopentanecarbonyl]-7-methyl-2,7-diazaspiro[4.5]decan-6-one
1-[2-hydroxy-2-(pyridin-2-yl)ethyl]-5,5-diphenylpiperidin-2-one
2-{dimethyl-[1,2]oxazolo[5,4-d]pyrimidin-4-yl}benzamide
N,N-dimethyl-5-{2-[1-(propan-2-yl)piperidin-4-yl]acetyl}-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
N-cyclopropyl-1-(2-{1-[3-(3-methoxyphenyl)propanoyl]piperidin-2-yl}ethyl)-1H-1,2,3-triazole-4-carboxamide
3-chloro-5-(2-{4-[(dimethylamino)methyl]phenyl}piperidine-1-carbonyl)-1,2-dihydropyridin-2-one
5-[4-methoxy-3-(methoxymethyl)phenyl]-1-methyl-3-(propan-2-yl)-1H,4H-pyrazolo[3,4-d]imidazole
N-(1,1-dioxo-2,3-dihydro-1λ6-thiophen-3-yl)-4-methyl-2-(4-methylpiperazin-1-yl)pyrimidine-5-carboxamide
5-{4-[(2-methoxyphenyl)methyl]piperazine-1-carbonyl}-N-(3-methylbutyl)-1-(2-methylpropyl)-4-oxo-1,4-dihydropyridine-3-carboxamide
2-ethyl-N-{3-[(pyridin-3-yl)amino]propyl}pyrimidine-5-carboxamide
1-(4-fluorophenyl)-4-{5-methyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carbonyl}-1,4-diazepane
2-(dimethyl-1,2-oxazol-4-yl)-N-[1-methyl-4-(morpholin-4-yl)-1H-indazol-3-yl]acetamide
4-(2,5-dimethylfuran-3-carbonyl)-6-[(3-methoxyphenyl)methoxy]-1-(2-methylpropyl)-1,4-diazepan-2-one
1-{2-azatricyclo[9.4.0.03,8]pentadeca-1(11),3,5,7,12,14-hexaen-5-yl}-3-ethyl-3-[(3S,4R)-4-hydroxyoxolan-3-yl]urea
(1R,3S)-3-ethoxy-7-[3-(1H-1,2,3,4-tetrazol-1-yl)-1H-pyrazole-4-carbonyl]-7-azaspiro[3.5]nonan-1-ol
4-[5-(thiophen-3-ylmethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-3-yl]benzonitrile
3-[1-cyclohexyl-3-(2-methoxyethyl)-1H-1,2,4-triazol-5-yl]-4,5,6,7-tetrahydro-1H-indazole
N-(3,4-dimethylphenyl)-1-[2-(1H-imidazol-2-yl)benzoyl]piperidin-3-amine
N-(2-{2-[2-(benzyloxy)phenyl]-1H-imidazol-1-yl}ethyl)acetamide
7-(2-methylphenyl)-4-[3-(pyridin-3-yl)propyl]-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
N-({3-methyl-7-[2-(thiophen-3-yl)acetyl]-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl}methyl)-1H-1,3-benzodiazole-5-carboxamide
N-{1H,4H,5H,6H,7H,8H-cyclohepta[c]pyrazol-3-ylmethyl}-1-[(3-fluorophenyl)methyl]-N-methyl-6-oxopiperidine-3-carboxamide
1-cyclopentyl-N-[(2,4-difluorophenyl)methyl]-4-oxo-5-(piperidine-1-carbonyl)-1,4-dihydropyridine-3-carboxamide
N-[(1-benzyl-1H-imidazol-2-yl)methyl]-1-ethyl-5-methyl-1H-pyrazole-4-carboxamide
4-[5-(3-propyl-1,2,4-oxadiazol-5-yl)-1H-pyrazol-3-yl]phenol
1-{4-[3-(3-methoxypropyl)piperidine-1-carbonyl]phenyl}ethan-1-one
[(5-chloro-1,3-dimethyl-1H-pyrazol-4-yl)methyl](ethyl){[5-(2-methylpropyl)-1,2,4-oxadiazol-3-yl]methyl}amine
N-[2-(2-chlorophenyl)-1-{1-[(4-acetamidophenyl)methyl]piperidin-4-yl}ethyl]-N-methylfuran-2-carboxamide
N-methyl-2-oxo-N-[(2-phenyl-1,3-thiazol-5-yl)methyl]-1,2-dihydroquinoline-4-carboxamide
1-cyclohexyl-3-[(4-methoxyphenyl)methyl]-5-(pyrrolidin-3-yl)-1H-1,2,4-triazole
N-{[7-chloro-2-(3-methylphenyl)quinolin-3-yl]methyl}-2-methyl-N-[3-(2-oxopyrrolidin-1-yl)propyl]-1,3-thiazole-4-carboxamide
(5S,9aS,9bS)-2-cyclopentyl-5-[4-(2-hydroxyethoxy)phenyl]-octahydro-1H-pyrrolo[3,4-h]pyrrolizin-1-one
4-[3-(furan-2-yl)-1,2,4-oxadiazol-5-yl]-N-methyl-N-[2-(4-methyl-1,3-thiazol-5-yl)ethyl]butanamide
N-(1,1-dioxo-1λ6-thian-4-yl)-3-(4-methoxyphenyl)-3-phenylpropanamide
N-cyclopropyl-2-[3-oxo-1-(thiophen-2-ylmethyl)piperazin-2-yl]-N-[(trimethyl-1H-pyrazol-4-yl)methyl]acetamide
6,7-dimethyl-2-{2-[2-(trifluoromethyl)morpholin-4-yl]ethyl}-1H-1,3-benzodiazole
[2-(3,5-dimethyl-1H-pyrazol-4-yl)ethyl]({[7-fluoro-2-(thiophen-3-yl)quinolin-3-yl]methyl})amine
3-[(3S,5S,9R)-2,8-dioxo-1,7-diazatricyclo[7.3.0.03,7]dodecan-5-yl]-1-[3-(trifluoromethyl)phenyl]urea
3-[3-(2-methoxyethyl)-1,2,4-oxadiazol-5-yl]-1-(oxan-4-yl)piperidine
4-{[2-(6-methylpyridazin-3-yl)phenyl]methyl}morpholine