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3,3-dimethyl-1-[(3S,4R)-1-(6-oxo-1,6-dihydropyridine-3-carbonyl)-4-(propan-2-yl)pyrrolidin-3-yl]urea
3-(1-methylpiperidin-2-yl)-1-{4-[2-(1H-pyrrol-1-yl)ethyl]piperazin-1-yl}propan-1-one
N-[(1R,2R,4S)-bicyclo[2.2.1]heptan-2-yl]-2-(pyridin-4-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-amine
2-methyl-5-propyl-N-{[2-(1H-1,2,4-triazol-1-yl)pyridin-3-yl]methyl}pyrimidin-4-amine
(2S)-2-amino-3-hydroxy-1-{4-hydroxy-4-[3-(trifluoromethyl)phenyl]piperidin-1-yl}propan-1-one
3-{[2-(hydroxymethyl)-2,5-dihydro-1H-pyrrol-1-yl]methyl}-5,6,7-trimethoxy-1,2-dihydroquinolin-2-one
2-[3-(2-methoxyphenoxy)propyl]-4,6-dimethylpyrimidine
6-phenyl-2-{2-[(pyrimidin-2-yl)amino]ethyl}-2,3-dihydropyridazin-3-one
(4aS,7aR)-1-(3,5-dimethylbenzoyl)-4-(2-methylpropanoyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
ethyl 1-[(3-acetylphenyl)methyl]-4-[(3-methoxyphenyl)methyl]piperidine-4-carboxylate
1-(oxan-4-yl)-3-{2-[2-(pyridin-2-yl)ethoxy]phenyl}urea
2-[(3aS,6aR)-3-cyclopentyl-2-oxo-hexahydro-2H-pyrrolo[3,4-d][1,3]oxazol-5-yl]-5H,6H,7H-cyclopenta[b]pyridine-3-carboxamide
1-cyclopentanecarbonyl-N-[2-(furan-2-yl)-2-hydroxyethyl]piperidine-4-carboxamide
N-{[2-(1,2,3,4-tetrahydroisoquinolin-2-yl)pyridin-3-yl]methyl}oxan-4-amine
7-(2-hydroxyethyl)-2-[2-(4-methyl-1,4-diazepan-1-yl)acetyl]-2,7-diazaspiro[4.5]decan-6-one
N-{[2-(azocan-1-yl)pyridin-3-yl]methyl}-2-(3-chloro-4-hydroxyphenyl)acetamide
(1S,5R)-6-(cyclopropylmethyl)-N-(3,4-dimethoxyphenyl)-7-oxo-3,6-diazabicyclo[3.2.2]nonane-3-carboxamide
5-methyl-1'-{4-methyl-6H,7H,8H-cyclopenta[g]quinolin-2-yl}-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
4-[(2,3-dihydro-1,4-benzodioxin-6-ylmethyl)amino]-1-(2,3-dihydro-1H-inden-2-yl)pyrrolidin-2-one
[(3R,4S)-4-[(4-methyl-1,4-diazepan-1-yl)methyl]-1-{[2-(propan-2-yl)pyrimidin-5-yl]methyl}pyrrolidin-3-yl]methanol
2-(1-{[4-methoxy-3-(1H-pyrazol-1-ylmethyl)phenyl]methyl}piperidin-2-yl)pyridine
{[1-benzyl-2-(2-methylpropanesulfonyl)-1H-imidazol-5-yl]methyl}(methyl)(propan-2-yl)amine
1-[(3R,4R)-3-hydroxy-4-(hydroxymethyl)piperidin-1-yl]-2-(1,2,3,4-tetrahydroisoquinolin-2-yl)ethan-1-one
N-(1-{1-[3-(5-methylfuran-2-yl)butyl]piperidin-4-yl}-1H-pyrazol-5-yl)acetamide
N-[(3R,4S)-4-cyclopropyl-1-(pyrimidin-2-ylmethyl)pyrrolidin-3-yl]-2-methanesulfonamidoacetamide
3-butyl-4-[(5-cyclopentyl-1,2,4-oxadiazol-3-yl)methyl]-1-methylpiperazin-2-one
2-methyl-4-{1-[5-(propan-2-yl)pyrimidin-4-yl]piperidin-3-yl}-6-(pyrrolidin-1-yl)pyrimidine
2-{4-[3-(3,5-dimethyl-1H-pyrazol-1-yl)pyrrolidin-1-yl]piperidin-1-yl}pyrimidine
[(1-{1-[1-(4-fluorophenyl)propan-2-yl]piperidin-4-yl}-1H-1,2,3-triazol-4-yl)methyl]urea
1-(benzyloxy)-8-[3-(thiophen-2-yl)propanoyl]-1,8-diazaspiro[4.5]decan-2-one
3-[(1S,5R)-3-(pyridin-2-ylmethyl)-3,6-diazabicyclo[3.2.2]nonane-6-carbonyl]-4,5,6,7-tetrahydro-1,2-benzoxazole
2-methyl-1-[1-(pyridine-3-carbonyl)piperidin-4-yl]-5-(trifluoromethyl)-1H-1,3-benzodiazole
2-{1-[3-(hydroxymethyl)-4-methoxyphenyl]-3,5-dimethyl-1H-pyrazol-4-yl}phenol
1-(3-fluorophenyl)-3-(1-{1-[2-(2-methylphenyl)acetyl]piperidin-4-yl}-1H-pyrazol-5-yl)urea
N-methyl-2-(methylsulfanyl)-N-{[3-(pyridin-4-yl)-1,2,4-oxadiazol-5-yl]methyl}pyridine-3-carboxamide
3-(piperazine-1-sulfonyl)-N-[3-(1H-1,2,3-triazol-1-yl)propyl]benzamide
methyl 4-[4-(2-{[(3-chlorophenyl)methyl]carbamoyl}ethyl)piperidin-1-yl]-4-oxobutanoate
(3S,4S)-1-{[5-fluoro-2-(trifluoromethyl)phenyl]methyl}-4-methylpiperidine-3,4-diol
4-{4-[4-ethyl-5-(pyrrolidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}-2-methylpyrimidine
7-methyl-3-[5-(morpholine-4-carbonyl)pyridin-2-yl]-1H-indole
1-[2-(dimethyl-1,3-thiazol-2-yl)ethyl]-3-(5-ethyl-1-methyl-1H-1,2,4-triazol-3-yl)urea
4-[1-(1-{[5-(4-chlorophenyl)furan-2-yl]methyl}piperidin-4-yl)-1H-1,2,3-triazole-4-carbonyl]morpholine
2-(butylsulfanyl)-6-[3-(1-methyl-1H-imidazole-2-carbonyl)piperidin-1-yl]pyrimidin-4-amine
4-[4-(3,5-dimethyl-1-phenyl-1H-pyrazol-4-yl)pyrimidin-2-yl]-1,4-oxazepane
4-(2-ethylpyrimidine-5-carbonyl)-6-(pyrrolidin-1-ylmethyl)-1,4-oxazepan-6-ol
4-[3-(1-ethyl-1H-imidazol-2-yl)piperidine-1-carbonyl]-N,N-dimethylaniline
[1-(2-methoxy-4-methylbenzenesulfonyl)-3-(prop-2-en-1-yl)piperidin-3-yl]methanol
1-[(2-fluoro-5-methoxyphenyl)methyl]-3-hydroxy-3-[({[1-(hydroxymethyl)cyclobutyl]methyl}amino)methyl]piperidin-2-one
N-cyclopentyl-1-[(4-methoxyphenyl)methyl]-5-(oxolane-3-carbonyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
N-{[2-(3,4-difluorophenoxy)pyridin-3-yl]methyl}-2-(methylamino)-1,3-thiazole-4-carboxamide