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N-(butan-2-yl)-6-methyl-2-oxo-N-(3-phenylprop-2-yn-1-yl)-1,2-dihydropyridine-3-carboxamide
3-(5-{[2-(3-methoxyphenyl)azetidin-1-yl]methyl}furan-2-yl)-1H-pyrazole
1-(1,3-dimethyl-2-oxo-2,3-dihydro-1H-1,3-benzodiazol-5-yl)-3-(3-ethoxypropyl)urea
N-[4-(1-methyl-1H-pyrazol-4-yl)phenyl]-3-oxobutanamide
N4-(1-cycloheptylpiperidin-3-yl)-N1,N1-dimethylpiperidine-1,4-dicarboxamide
2-{spiro[indene-1,4'-piperidine]-1'-ylmethyl}pyridine-3-carboxylic acid
2-methyl-N-[2-(5-methylfuran-2-yl)-2-(morpholin-4-yl)ethyl]-1,3-benzoxazole-6-carboxamide
1-{6-[4-(cyclohexylmethyl)-3-(2-hydroxyethyl)piperazin-1-yl]pyridin-3-yl}ethan-1-one
7-[2-(morpholin-4-yl)pyridine-3-carbonyl]-5H,6H,7H,8H-imidazo[1,2-a]pyrazine-3-carboxamide
3-(azocan-1-yl)-1-(1,4-oxazepan-4-yl)propan-1-one
(4aR,8aR)-7-[(6-chloro-2H-1,3-benzodioxol-5-yl)methyl]-4a-hydroxy-N,N-dimethyl-decahydro-2,7-naphthyridine-2-carboxamide
1-[2-(1-methyl-1H-imidazol-2-yl)benzoyl]-4-[(2-methylphenyl)methyl]piperazine
2-[5-(4-propylpyrimidin-5-yl)-3-(pyridin-4-yl)-1H-1,2,4-triazol-1-yl]acetic acid
1-[1'-(4,6-dimethylpyridine-3-carbonyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-5-yl]-2-methoxyethan-1-one
N-{2-[(1-methyl-1H-imidazol-2-yl)sulfanyl]ethyl}-1,9-dioxaspiro[5.5]undecan-4-amine
4-hydroxy-1-[3-(6-methyl-2-oxo-1,2-dihydropyridin-1-yl)propanoyl]piperidine-4-carboxylic acid
N-[1-(2-{4-[(1S,4S)-2-azabicyclo[2.2.1]heptan-2-ylmethyl]-3-methyl-1H-pyrazol-1-yl}ethyl)piperidin-4-yl]acetamide
3-[4-(2-chlorophenyl)-3-oxopiperazin-1-yl]propanoic acid
1-(3-chlorophenyl)-4-{1-[(3-methoxyphenyl)methyl]piperidin-3-yl}piperazine
N-[(1-ethylpyrrolidin-2-yl)methyl]-3-{1-[(4-methyl-1H-imidazol-2-yl)methyl]piperidin-4-yl}propanamide
N-{[2-(dimethylamino)-5,8-dimethoxyquinolin-3-yl]methyl}-2-ethyl-N-[(4-methoxyphenyl)methyl]butanamide
3-{[1-(4-chlorophenyl)-3-cyclopropyl-1H-1,2,4-triazol-5-yl](pyrrolidin-1-yl)methyl}pyridine
ethyl 1-(4-acetylbenzoyl)-3-[(4-fluorophenyl)methyl]piperidine-3-carboxylate
methyl[(4-methyl-1H-imidazol-5-yl)methyl][2-(morpholin-4-yl)propyl]amine
2-(pyridin-2-yl)-5-{[3-(pyridin-3-yl)azetidin-1-yl]methyl}pyrimidine
4-{2-[1-(2,3-dihydro-1H-indene-5-carbonyl)piperidin-2-yl]ethyl}morpholine
4-[(1-cyclopropanecarbonylpiperidin-4-yl)oxy]-N-(2-hydroxyethyl)-N-(propan-2-yl)benzamide
4-(4-{[4-methoxy-3-(methoxymethyl)phenyl]methyl}piperazin-1-yl)-6-methylpyrimidin-2-amine
1-(1,3-dimethyl-1H-pyrazole-5-carbonyl)-4-[(4-fluorophenyl)methyl]-3-(propan-2-yl)-1,4-diazepan-5-one
N-[(3-ethyl-4,5-dihydro-1,2-oxazol-5-yl)methyl]-5-methyl-1-benzofuran-2-carboxamide
2-[(1S,5R)-3-[(4-methoxyphenyl)methyl]-3,6-diazabicyclo[3.2.2]nonan-6-yl]-1-(morpholin-4-yl)ethan-1-one
5-propyl-N-(3-{[1,2,4]triazolo[4,3-a]pyridin-3-yl}propyl)pyrazolo[1,5-a]pyrimidin-7-amine
N-[(3S,7S,8aS)-3-(4-aminobutyl)-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-3-tert-butyl-1-methyl-1H-pyrazole-5-carboxamide
(4-{[4-(1-methyl-1H-imidazol-2-yl)piperidin-1-yl]sulfonyl}phenyl)urea
4-[4-ethyl-5-(1H-1,2,4-triazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]-1-(5-methoxyfuran-2-carbonyl)piperidine
1-(cyclopropylmethyl)-N-methyl-5-(1-methyl-3-propyl-1H-pyrazole-5-carbonyl)-N-(1,3-thiazol-4-ylmethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
N-{[1-(furan-2-ylmethyl)piperidin-4-yl]methyl}pyrrolidine-1-sulfonamide
2-{2-[(3S)-3-(dimethylamino)azepan-1-yl]-2-oxoethyl}-5,6-dimethyl-2,3-dihydropyridazin-3-one
5-{[(isoquinolin-5-ylmethyl)(methyl)amino]methyl}-N-(oxolan-2-ylmethyl)pyrimidin-2-amine
5-(10-methoxy-3,4,5,6-tetrahydro-2H-1,5-benzoxazocine-5-carbonyl)-1-(pyridin-2-ylmethyl)piperidin-2-one
2-propyl-N-{[2-(pyrazin-2-yl)-1,3-thiazol-4-yl]methyl}-1,3-thiazole-4-carboxamide
1-[4-(morpholin-4-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl]-5-phenylpentan-1-one
4-(3-tert-butyl-1H-pyrazol-1-yl)-1-(furan-2-carbonyl)piperidine-4-carboxylic acid
2-(carbamoylamino)-N-({1-[(3,5-dimethylphenyl)methyl]pyrrolidin-3-yl}methyl)acetamide
N-butyl-3-fluoro-N-(furan-2-ylmethyl)pyridine-4-carboxamide
methyl N-(2-{4-[4-methyl-5-(pyrrolidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}-2-oxoethyl)carbamate
(5S,9aS,9bS)-2-methyl-5-(1-phenyl-1H-pyrazol-4-yl)-octahydro-1H-pyrrolo[3,4-h]pyrrolizin-1-one
ethyl 3-({3-[4-(2H-1,3-benzodioxol-5-ylmethyl)piperazin-1-yl]piperidine-1-carbonyl}amino)propanoate
1-[4-(piperidin-1-ylmethyl)phenoxy]-3-(1,2,3,4-tetrahydroisoquinolin-2-yl)propan-2-ol
4-phenyl-1-{[3-(thiophen-2-yl)-1,2,4-oxadiazol-5-yl]methyl}azepane