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1-methyl-N-{[3-(pyrrolidin-1-ylmethyl)phenyl]methyl}piperidin-4-amine
1-{1-[2-(1-methyl-3-oxopiperazin-2-yl)acetyl]piperidin-4-yl}-2,3-dihydro-1H-1,3-benzodiazol-2-one
N-(2-{5-[(2-methoxyethyl)sulfanyl]-4-methyl-4H-1,2,4-triazol-3-yl}ethyl)-1-(4-methoxyphenyl)cyclopentane-1-carboxamide
N-[(2S,4R,6S)-2-benzyl-6-(4-methyl-1H-imidazol-5-yl)oxan-4-yl]acetamide
4-(4-ethyl-1H-pyrazol-5-yl)-1-[3-(3-methylphenyl)-1H-pyrazole-4-carbonyl]piperidine
(2S,4S)-4-amino-N,N-diethyl-1-[1-methyl-3-(thiophen-2-yl)-1H-pyrazole-5-carbonyl]pyrrolidine-2-carboxamide
6-methoxy-3-{2-[9-methoxy-7-(thiophen-2-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]-2-oxoethyl}-2,3-dihydro-1H-indol-2-one
1-(2H-1,3-benzodioxol-5-yl)-N-[1-(1-methyl-1H-pyrazol-5-yl)propyl]piperidin-4-amine
N-{2-methyl-1-[7-(4-oxo-4H-chromene-2-carbonyl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl]propyl}furan-3-carboxamide
N-[2-(2-chlorophenyl)-1-{1-[(2-fluorophenyl)methyl]piperidin-4-yl}ethyl]-N-methylfuran-2-carboxamide
6-ethyl-N4-{[1-(furan-2-ylmethyl)piperidin-3-yl]methyl}-5-methylpyrimidine-2,4-diamine
methyl({[4-methyl-5-(piperidin-4-ylmethyl)-4H-1,2,4-triazol-3-yl]methyl})[(5-phenyl-1H-pyrazol-3-yl)methyl]amine
2-(1-methyl-4-{[4-(propan-2-yl)-1,3-thiazol-2-yl]methyl}piperazin-2-yl)ethan-1-ol
N-(3-{[(2-fluorophenyl)methyl]sulfanyl}propyl)-4,5,6-trimethyl-2-oxo-1,2-dihydropyridine-3-carboxamide
ethyl({1-[2-(3-fluorophenyl)ethyl]piperidin-3-yl}methyl)(1H-pyrazol-3-ylmethyl)amine
4-(1-{[5-(methoxymethyl)-1H-pyrazol-3-yl]methyl}-1H-1,2,3-triazol-4-yl)quinoline
2-{1-[1-(furan-2-yl)ethyl]-1H-1,2,3-triazol-4-yl}quinolin-4-ol
3-({[(2-aminopyrimidin-5-yl)methyl](methyl)amino}methyl)-N-(1,2,4-thiadiazol-5-yl)benzamide
4-{[(2R,3R)-3-(dimethylamino)-2-hydroxy-2,3-dihydrospiro[indene-1,4'-piperidine]-1'-yl]carbonyl}-6-methyl-1,2-dihydropyridin-2-one
1-[3-(thiomorpholine-4-sulfonyl)benzoyl]-1,4-diazepane
1-[(4-chlorophenyl)methyl]-3-(pyrrolidin-1-yl)piperidine
2-[(4-cyclobutanecarbonyl-1,4-diazepan-1-yl)methyl]-8-fluoroquinolin-4-ol
2-{4-[3-(1H-1,3-benzodiazol-5-yl)-1,2,4-oxadiazol-5-yl]piperidin-1-yl}acetamide
3-(2,4-difluorophenyl)-1-[(3S,4S)-3,4-dihydroxy-4-methylpiperidin-1-yl]propan-1-one
2-(2-methoxyethyl)-N-(4-methoxyphenyl)-3-oxo-2,9-diazaspiro[5.5]undecane-9-carboxamide
1-[(3S,4S)-4-hydroxy-1,1-dioxo-1λ6-thiolan-3-yl]-3-(6-methoxy-2-oxo-2,3-dihydro-1H-1,3-benzodiazol-5-yl)urea
N-[(2R,3R)-1'-(furan-3-carbonyl)-2-methoxy-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]pyridine-2-carboxamide
1-(2-methoxyethyl)-8-[(1-methyl-1H-1,3-benzodiazol-2-yl)methyl]-3-(pyridin-3-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
(8aS)-2-{[3-(2-methylphenyl)-1,2,4-oxadiazol-5-yl]methyl}-octahydropyrrolo[1,2-a]piperazine-1,4-dione
3-[1-(1-benzothiophen-2-ylmethyl)piperidin-4-yl]-1-(4-phenylpiperazin-1-yl)propan-1-one
[1-(5-methyl-1-phenyl-1H-pyrazol-4-yl)ethyl]({[3-(trifluoromethyl)phenyl]methyl})amine
N-{5,7-dimethylpyrido[2,3-d]pyrimidin-4-yl}-1-methanesulfonylpiperidin-4-amine
methyl 3-benzamido-1-(oxolan-2-ylmethyl)-5-[(2-phenylethyl)amino]-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
3-{5-[1-(4-chlorophenyl)cyclobutyl]-1,3,4-oxadiazol-2-yl}-1-[4-(2-methoxyethoxy)piperidin-1-yl]propan-1-one
(3S,4S)-1-[4-(ethylamino)pyrimidin-2-yl]-4-(4-methylpiperazin-1-yl)pyrrolidin-3-ol
4-{[1-methyl-6-(pyridin-4-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-yl]amino}-1,2,3,4-tetrahydroquinolin-2-one
(4aS,8aR)-1-(2-aminoethyl)-6-(1-phenylpiperidin-4-yl)-decahydro-1,6-naphthyridin-2-one
3-methyl-7-(3-propyl-1H-pyrazole-4-carbonyl)-1-oxa-3,7-diazaspiro[4.4]nonan-2-one
9-[(5-chloro-1,3-dimethyl-1H-pyrazol-4-yl)sulfonyl]-3-methyl-3,9-diazaspiro[5.6]dodecane
N-(5-methyl-2,1,3-benzothiadiazol-4-yl)-3-(4H-1,2,4-triazol-3-yl)piperidine-1-carboxamide
4-benzyl-3-ethyl-1-(1H-imidazol-4-ylmethyl)-1,4-diazepan-5-one
N-[4-chloro-3-(3-methyl-1,2,4-oxadiazol-5-yl)phenyl]acetamide
3-[(dimethylamino)methyl]-1-[(1-methyl-1H-imidazol-2-yl)methyl]piperidin-3-ol
N2-{1-methyl-6-propyl-1H-pyrazolo[3,4-d]pyrimidin-4-yl}-N1-(3-methylpyridin-2-yl)ethane-1,2-diamine
3-(3-hydroxy-3-methylbutyl)-N-[1-(5-methyl-1,3,4-oxadiazol-2-yl)ethyl]benzamide
1-[2-(3-fluorophenyl)ethyl]-N-[(4-methylphenyl)methyl]-6-oxopiperidine-3-carboxamide
1-methyl-N-(oxolan-2-ylmethyl)-N-(thiophen-3-ylmethyl)-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
1-{4-hydroxy-4-[3-(trifluoromethyl)phenyl]piperidin-1-yl}-6-methoxyhexan-1-one
4-{4-[3-(4-fluorophenyl)benzoyl]piperazin-1-yl}-2-(pyridin-4-ylmethyl)-2,3-dihydro-1H-isoindole-1,3-dione
2-(morpholin-3-yl)-1-[2-(pyrrolidin-1-ylmethyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-5-yl]ethan-1-one