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3-chloro-N-[1-(4-propyl-4H-1,2,4-triazol-3-yl)ethyl]pyridine-4-carboxamide
1-(1-benzothiophene-5-carbonyl)-3-(pyrrolidin-1-ylmethyl)piperidin-3-ol
N-[4-(4-{[(3S)-2-oxoazepan-3-yl]amino}piperidin-1-yl)phenyl]-2-phenoxyacetamide
4-[1-(4-fluorophenyl)cyclopropanecarbonyl]-3-methyl-1-[(3-methylphenyl)methyl]piperazin-2-one
2-{1-[(2-fluoro-4-methoxyphenyl)methyl]-3-oxopiperazin-2-yl}acetamide
5-{[3-(3,4-difluorophenyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]methyl}-2-(methoxymethyl)pyrimidine
2-butyl-8-{[1,2,3,4]tetrazolo[1,5-a]pyridine-6-carbonyl}-2,8-diazaspiro[5.5]undecan-3-one
2-amino-1-(azocan-1-yl)-2-(3,5-dimethyl-1H-pyrazol-4-yl)ethan-1-one
N-(4-{4-[(1,2,3,4-tetrahydronaphthalen-1-yl)amino]piperidin-1-yl}phenyl)-2H-1,3-benzodioxole-5-carboxamide
4-[2-(3-methoxyphenyl)azetidine-1-carbonyl]-2-propyl-1,3-thiazole
[(2-fluorophenyl)methyl](1H-imidazol-2-ylmethyl)(2-methoxyethyl)amine
(1S,5R)-3-[2-(2-methyl-1,3-thiazol-4-yl)acetyl]-6-(1,3-thiazol-4-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
4-{4-[(2,3-difluoro-4-methoxyphenyl)methyl]-2-oxopiperazin-1-yl}benzonitrile
(3S,4R)-1-methyl-3-{[4-(3-methylpyridin-2-yl)piperazin-1-yl]methyl}piperidin-4-ol
2-{1-[(2-chloro-6-fluorophenyl)methyl]pyrrolidin-2-yl}-1,3-thiazole
2-methyl-4-{pyrazolo[1,5-a]pyridin-7-yl}-1H-imidazole
N-[(1-cyclohexylpyrrolidin-3-yl)methyl]-5,7-dimethylpyrido[2,3-d]pyrimidin-4-amine
N-cyclooctyl-4-[(3S,4S)-3,4-dihydroxypiperidin-1-yl]-4-oxobutanamide
N-[2-(dimethylamino)-5,6,7,8-tetrahydroquinazolin-5-yl]cyclopropanecarboxamide
N-butyl-3-[2-(furan-2-ylmethyl)-5-oxopyrrolidin-2-yl]propanamide
N-[1-(1-{1H,4H,5H,6H-cyclopenta[c]pyrazole-3-carbonyl}piperidin-4-yl)-1H-pyrazol-5-yl]-2-methylbenzamide
N-[2-(pyridin-3-yl)ethyl]-2-[2,6,6-trimethyl-1-(2-methylpropyl)-4-oxo-4,5,6,7-tetrahydro-1H-indol-3-yl]acetamide
4-cyclobutaneamido-N-[3-(3,5-dimethyl-1H-pyrazol-4-yl)propyl]benzamide
N-[(3-ethyl-1,2-oxazol-5-yl)methyl]-N,5-dimethyl-3-phenyl-1,2-oxazole-4-carboxamide
3-[5-(2-cyclohexylethyl)-1,3,4-oxadiazol-2-yl]-N-[2-(pyridin-3-yl)ethyl]propanamide
N-{5H,6H,7H,8H-imidazo[1,2-a]pyridin-3-yl}-1H,4H,5H,6H-cyclopenta[c]pyrazole-3-carboxamide
5-chloro-6-(3-{[4-(hydroxymethyl)phenyl]methyl}pyrrolidin-1-yl)-2-methylpyrimidin-4-ol
N-(3-{1-azabicyclo[3.2.1]octan-5-yloxy}phenyl)-5-methyl-1,2-oxazole-3-carboxamide
2-(4-methoxy-3-methylphenyl)-N-[2-(4-methylmorpholin-2-yl)ethyl]acetamide
4-{[1-(dimethylsulfamoyl)piperidin-4-yl]oxy}-N-(3-hydroxy-2,2-dimethylpropyl)benzamide
2-(4-cyclohexyl-1,4-diazepan-1-yl)-2-(3-hydroxyphenyl)acetic acid
8-[3-(5-methyl-1,3,4-oxadiazol-2-yl)phenyl]quinoline
(4aS,8aR)-6-(2-methylpyrimidin-4-yl)-1-[2-(thiophen-2-yl)ethyl]-decahydro-1,6-naphthyridin-2-one
{4-[(4-chlorophenyl)methyl]-1-[3-(dimethylamino)pyrazin-2-yl]piperidin-4-yl}methanol
(3R,4R)-1-(7-chloroquinolin-4-yl)-4-(hydroxymethyl)piperidin-3-ol
1-[1-(2-phenylethyl)piperidin-4-yl]-N-(pyrimidin-4-ylmethyl)piperidine-3-carboxamide
3-(1H-imidazol-4-yl)-2-[(2-propyl-1,3-thiazol-4-yl)formamido]propanoic acid
1-[2-(methylsulfanyl)ethyl]-5-{2-[(prop-2-en-1-yl)amino]ethyl}pyrrolidin-2-one
4-{[2-(dimethyl-1,3-thiazol-5-yl)-1H-imidazol-1-yl]methyl}benzene-1-sulfonamide
4-[(2-cyclohexylpyrimidin-5-yl)methyl]-N,N-dimethylpiperazine-1-sulfonamide
4-(1,3-dimethyl-1H-pyrazol-4-yl)-N-(2-{imidazo[1,2-a]pyridin-2-yl}ethyl)pyrimidin-2-amine
N-{4,5-dimethyl-3-[3-(1H-pyrazol-5-yl)piperidine-1-carbonyl]thiophen-2-yl}-2-methylpropanamide
5-(pyrrolidine-1-carbonyl)-2-(2,3,4,5-tetrahydro-1-benzoxepin-4-ylmethyl)pyridine
3-[3-({[2-(1H-1,2,4-triazol-5-ylsulfanyl)ethyl]amino}methyl)-1H-indol-1-yl]propanamide
3-(4-methoxyphenoxymethyl)-1-(1-methyl-1H-pyrrole-2-carbonyl)piperidine
{1-[5-methyl-1-(naphthalen-1-yl)-1H-pyrazol-4-yl]ethyl}({[2-methyl-4-(1H-pyrazol-1-yl)phenyl]methyl})amine
2-[1-({6-cyclopentyl-1-methyl-1H-pyrazolo[3,4-d]pyrimidin-4-yl}amino)ethyl]phenol
4-benzyl-3-{1-[(3-hydroxyphenyl)methyl]piperidin-4-yl}-4,5-dihydro-1H-1,2,4-triazol-5-one
N-(2-methoxyethyl)-N,5-dimethyl-4-(piperidin-1-yl)thieno[2,3-d]pyrimidine-6-carboxamide
8-fluoro-2-({2-methyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-5-yl}methyl)quinolin-4-ol