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N-[(3-cyclohexyl-1,2,4-oxadiazol-5-yl)methyl]-5-methyl-1-propyl-1H-pyrazole-4-carboxamide
(3S,4R)-1-(3-ethyl-4-methyl-1H-pyrazole-5-carbonyl)-4-(pyridin-3-yl)pyrrolidine-3-carboxylic acid
N-{[2-(2,6-dimethylphenoxy)pyridin-3-yl]methyl}-2-(1H-1,2,4-triazol-1-yl)propanamide
3-(2-methylpyridin-4-yl)-5-[2-(piperidin-2-yl)ethyl]phenol
2-(adamantan-1-yl)-5-(3-methylpiperidine-1-carbonyl)pyrimidin-4-ol
1-ethyl-N-[1-(1H-indol-5-yl)ethyl]-3-methyl-1H-pyrazole-4-carboxamide
N-[2-(4-methyl-5-{[2-(morpholin-4-yl)ethyl]sulfanyl}-4H-1,2,4-triazol-3-yl)ethyl]-4-phenylbenzamide
4-{[1-(2-methoxyacetyl)piperidin-4-yl]oxy}-N-[(5-methyl-1,2-oxazol-3-yl)methyl]benzamide
2-(1H-indol-3-yl)-N-{[8-(pyridin-4-ylmethyl)-1-oxa-8-azaspiro[4.5]decan-2-yl]methyl}acetamide
2-(2-phenyl-1H-imidazol-1-yl)-N-[(4-sulfamoylphenyl)methyl]acetamide
5-[2,2-bis(prop-2-en-1-yl)pyrrolidine-1-carbonyl]-1-[2-(pyridin-2-yl)ethyl]piperidin-2-one
3-methyl-5-[3-(4-phenylphenyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-5-carbonyl]-1H-pyrazole
2-({[(3R,4R)-1-(2,3-difluoro-4-methoxybenzoyl)-4-(hydroxymethyl)pyrrolidin-3-yl]methyl}(methyl)amino)ethan-1-ol
N-[2-(cyclohex-1-en-1-yl)ethyl]-2-methyl-N-{[6-(morpholin-4-yl)-2H-[1,3]dioxolo[4,5-g]quinolin-7-yl]methyl}propanamide
N-[3-methyl-1-(4-methylphenyl)-1H-pyrazol-5-yl]-2-[4-(1,3-thiazol-2-yl)-1H-pyrazol-1-yl]acetamide
4-[(2-fluoro-3-methylphenyl)methyl]-1,3λ6,4-oxathiazinane-3,3-dione
N-ethyl-1-[6-methyl-2-(pyridin-3-yl)pyrimidin-4-yl]pyrrolidine-3-carboxamide
N-(1-phenylbutyl)-3-(4H-1,2,4-triazol-4-yl)benzamide
(3S,4S)-1-[2-(2-amino-4,6-dimethylpyrimidin-5-yl)acetyl]-4-(pyridin-2-yl)pyrrolidine-3-carboxylic acid
1-{3-[(3R,4S)-4-hydroxy-3,4-dimethylpiperidin-1-yl]-3-oxopropyl}azepan-2-one
3-{[ethyl(propan-2-yl)carbamoyl]methyl}-N-(2-methoxyethyl)-4-methyl-3,4-dihydro-2H-1,4-benzoxazine-6-carboxamide
N,N-dimethyl-5-({3-[4-(4-methylphenyl)-1H-pyrazol-5-yl]piperidin-1-yl}methyl)-1,3-thiazol-2-amine
5-acetyl-N-{[4-(propan-2-yl)-1,2,3-thiadiazol-5-yl]methyl}-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carboxamide
3-[benzyl({[6-(dimethylamino)pyridin-3-yl]methyl})amino]-1λ6-thiolane-1,1-dione
N-[2-(5-methoxy-1H-1,3-benzodiazol-2-yl)ethyl]-N-methyl-2-(methylamino)acetamide
1-[(3-hydroxyphenyl)methyl]-N-[3-(1H-pyrazol-1-yl)phenyl]pyrrolidine-2-carboxamide
N-[2-(1H-imidazol-1-yl)-1-phenylethyl]-1,3-dimethyl-1H-pyrazolo[3,4-d][1,3]thiazol-5-amine
3-(2-phenylethyl)-5-(1H-pyrrol-2-yl)-1H-1,2,4-triazole
{[3-(3-fluorophenyl)oxolan-3-yl]methyl}[2-methyl-1-(morpholin-4-yl)propan-2-yl]amine
1-({5-[2-(2-methylpropyl)-5H,6H,7H-pyrrolo[3,4-d]pyrimidine-6-carbonyl]furan-2-yl}methyl)-1H-imidazole
4-(1-{1-[(4-methoxy-2,5-dimethylphenyl)methyl]piperidin-4-yl}-1H-1,2,3-triazole-4-carbonyl)morpholine
8-fluoro-2-{[3-(1-methyl-1H-imidazol-2-yl)piperidin-1-yl]methyl}-1,4-dihydroquinolin-4-one
1-(3-chlorophenyl)-4-[6-(hydroxymethyl)pyridine-2-carbonyl]piperazin-2-one
5-[4-(4-fluorophenyl)-1,4-diazepane-1-carbonyl]-2-methylpyrimidin-4-ol
7-{pyrazolo[1,5-a]pyridine-7-carbonyl}-2,7-diazaspiro[4.4]nonane-1,3-dione
N-[1-(methoxymethyl)cyclopentyl]-1,5-dimethyl-1H-pyrrole-2-carboxamide
N-({1-[(2-methoxyphenyl)methyl]piperidin-4-yl}methyl)-N-(2-methylpropyl)pyrazine-2-carboxamide
2-(3-benzyl-1-methyl-2-oxo-2,3-dihydro-1H-indol-3-yl)-N-(pyrimidin-4-ylmethyl)acetamide
N-{[3-(benzyloxy)phenyl]methyl}-1-ethyl-5-oxopyrrolidine-3-carboxamide
methyl(pyrazin-2-ylmethyl){[3-(thiophen-2-yl)-1,2,4-oxadiazol-5-yl]methyl}amine
{2-[2-(3-methoxyphenyl)piperidin-1-yl]-2-oxoethyl}urea
propyl N-({5-methanesulfonyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)carbamate
3-(4-methyl-1,3-thiazol-5-yl)-N-{5H,6H,7H-pyrrolo[2,1-c][1,2,4]triazol-3-ylmethyl}propanamide
3-[(3S,7S,8aS)-3-[(benzyloxy)methyl]-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-1-[2-(trifluoromethyl)phenyl]urea
2-(phenylamino)-N-{[4-(propan-2-yl)-1,2,3-thiadiazol-5-yl]methyl}pyrimidine-5-carboxamide
2-[3-(3,4-difluorophenyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-5-carbonyl]-4-methyl-1H-pyrrole
1-[(4-chlorophenyl)methyl]-5-(4-methoxypiperidine-1-carbonyl)piperidin-2-one
(3R,5R)-5-{4-[(4-fluorophenyl)methyl]piperazine-1-carbonyl}pyrrolidin-3-ol
2-(3-methylbutyl)-8-(2-methylpyrimidin-4-yl)-2,8-diazaspiro[5.5]undecan-3-one
2-methylpropyl (2R,3S,6R)-3-(3-methoxyphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecane-5-carboxylate