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6-{1-[(5-chloro-3-ethyl-1-methyl-1H-pyrazol-4-yl)methyl]piperidin-3-yl}-2-methylpyrimidin-4-ol
3-(2-methoxyethyl)-1-{[2-(methylamino)-1,3-thiazol-4-yl]methyl}piperidine-3-carboxylic acid
2-methyl-4-[(2R,3R,6R)-3-phenyl-1,5-diazatricyclo[5.2.2.02,6]undecane-5-carbonyl]phenol
N-(2-ethyl-2H-1,2,3-triazol-4-yl)-2-[5-(4-methoxyphenyl)-1H-indazol-1-yl]acetamide
2-[4-({[1-(3,5-dimethylphenyl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]amino}methyl)phenoxy]ethan-1-ol
2-(3-fluoro-4-methoxyphenyl)-2-(4-hydroxy-4-phenylpiperidin-1-yl)acetic acid
1-(5,6,7,8-tetrahydronaphthalen-1-yl)-3-[3-(1H-1,2,4-triazol-1-yl)propyl]urea
N-[(5-fluoro-3-methyl-1H-indol-2-yl)methyl]-1-(pyrimidin-2-yl)piperidin-3-amine
1-(3-chloro-5-methylpyridin-2-yl)-4-{[3,5-dimethyl-1-(propan-2-yl)-1H-pyrazol-4-yl]methyl}piperazine
N-[(3-ethyl-1,2-oxazol-5-yl)methyl]-N-methyl-2-(2-methyl-5-oxopyrrolidin-1-yl)acetamide
1-{3-fluoro-7-methylimidazo[1,2-a]pyridine-2-carbonyl}-4-(4-methylphenoxy)piperidine
3-methyl-1-(1-{6-[2-(methylsulfanyl)phenyl]pyridine-3-carbonyl}piperidin-3-yl)butan-1-one
4-(4-{[({1-[2-(2-methoxyphenyl)ethyl]piperidin-3-yl}methyl)(methyl)amino]methyl}phenyl)but-3-yn-1-ol
N-[1-(pyrazin-2-yl)propan-2-yl]-2-(2,5,7-trimethyl-1H-indol-3-yl)acetamide
3-cyclohexyl-N-methyl-N-[(5-phenyl-1,2-oxazol-3-yl)methyl]-1H-pyrazole-4-carboxamide
2-{4-[(1,3-dimethyl-1H-pyrazol-4-yl)methyl]-1-[(4-ethoxyphenyl)methyl]piperazin-2-yl}ethan-1-ol
2-{1-[(1R,2R,4R)-bicyclo[2.2.1]hept-5-ene-2-carbonyl]piperidin-4-yl}-1-methyl-1H-1,3-benzodiazole
(3S,4R)-1-[5-(methoxymethyl)furan-2-carbonyl]-4-(pyridin-3-yl)pyrrolidine-3-carboxylic acid
ethyl 4-(2-phenoxyethyl)-1-phenylmethanesulfonylpiperidine-4-carboxylate
4-methyl-6-{4-[(1-phenyl-1H-1,2,3-triazol-4-yl)methyl]piperazin-1-yl}pyrimidin-2-amine
2-(2-ethoxyphenyl)-1-[4-(6-hydroxy-2-methylpyrimidin-4-yl)piperidin-1-yl]ethan-1-one
N-methyl-N-{[3-(1H-pyrazol-1-yl)phenyl]methyl}-4-(pyrrolidine-1-carbonyl)pyridin-2-amine
5-propyl-N-[2-(1H-pyrazol-1-yl)ethyl]pyrazolo[1,5-a]pyrimidin-7-amine
4-{3-[5-(1H-imidazol-1-ylmethyl)-4-methyl-4H-1,2,4-triazol-3-yl]piperidine-1-carbonyl}-2-methoxypyridine
ethyl 4-{1-[(2-phenyl-1,3-thiazol-5-yl)methyl]piperidin-3-yl}piperazine-1-carboxylate
5-{[4-(adamantan-1-yl)piperazin-1-yl]methyl}-N,N-dimethylpyridin-2-amine
3-benzyl-1-(3-ethyl-5-methyl-1,2-oxazole-4-carbonyl)piperidine-3-carboxylic acid
({2-[(dimethylamino)methyl]phenyl}methyl)[(2-ethylpyrimidin-5-yl)methyl]methylamine
2-{4-[(6-fluoroquinolin-2-yl)methyl]-1-(3-methylbutyl)piperazin-2-yl}ethan-1-ol
8-cyclopentanecarbonyl-2-[(5-methylpyrazin-2-yl)methyl]-2,8-diazaspiro[5.5]undecan-3-one
(3R,4R)-4-(2-methoxyethyl)-3-methyl-1-[2-(1H-1,2,4-triazol-3-yl)benzoyl]piperidin-4-ol
N-(2,1,3-benzoxadiazol-5-ylmethyl)-3-(3-fluorophenyl)-N-methyl-1H-pyrazole-4-carboxamide
(3S,4S)-1-[(2-chloro-4-fluorophenyl)methyl]-4-(dimethylamino)pyrrolidin-3-ol
N-{[2-(1H-imidazol-1-yl)pyridin-3-yl]methyl}-3-(5-methylfuran-2-yl)-1H-pyrazole-5-carboxamide
3-[(dimethyl-1,2-oxazol-4-yl)methyl]-3-methyl-1-(6-methyl-2H-1,3-benzodioxol-5-yl)urea
2-{2-[(2,4-dimethyl-3-oxopiperazin-1-yl)methyl]-4-(pyrazin-2-yl)phenoxy}acetic acid
2-(dimethylamino)-N-{[2-(2-fluorophenoxy)pyridin-3-yl]methyl}propanamide
N-butyl-1-(furan-2-ylmethyl)-4-oxo-5-(3-phenylpiperidine-1-carbonyl)-1,4-dihydropyridine-3-carboxamide
8-[(5-fluoro-2-methoxyphenyl)methyl]-2-(2-methoxyethyl)-2,8-diazaspiro[5.5]undecan-3-one
(3R,5S)-N-cyclopentyl-5-[(2,3-dihydro-1H-inden-5-yloxy)methyl]piperidine-3-carboxamide
2-(dimethylamino)-8-[2-methyl-6-(piperidin-3-yl)pyrimidin-4-yl]-1,3,8-triazaspiro[4.5]dec-1-en-4-one
3-{1,4-dioxa-8-azaspiro[4.5]decan-8-ylmethyl}-1-[(2-fluorophenyl)methyl]-3-hydroxypiperidin-2-one
2-(5-{[4-(adamantan-2-yl)piperazin-1-yl]methyl}-1,2,4-oxadiazol-3-yl)pyrazine
3-[(2R,3R,6R)-5-{[2-(methoxymethyl)pyrimidin-5-yl]methyl}-1,5-diazatricyclo[5.2.2.02,6]undecan-3-yl]phenol
4-(4-{[7-(2-methoxyethyl)-2,7-diazaspiro[4.5]decan-2-yl]methyl}phenyl)but-3-yn-1-ol
2-(4-chlorophenyl)-4-(5-cyclopropyl-1,3-oxazole-4-carbonyl)morpholine
(8R,9aS)-8-hydroxy-2-{[2-(1H-pyrazol-1-yl)phenyl]methyl}-octahydro-1H-pyrido[1,2-a]piperazine-1,4-dione
3-(1,2-oxazinan-2-yl)-N-{1-[2-(1H-pyrazol-1-yl)phenyl]ethyl}propanamide
4-[1-(2,3,4,5-tetrahydro-1-benzoxepin-4-ylmethyl)azetidin-3-yl]morpholine
5-{[3-(naphthalene-2-carbonyl)piperidin-1-yl]methyl}-N-(propan-2-yl)pyrimidin-2-amine