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3-{1-[3-(3-methoxyphenyl)-1H-pyrazole-4-carbonyl]piperidin-4-yl}-1,3-oxazolidin-2-one
1-{6-cyclopentyl-1-methyl-1H-pyrazolo[3,4-d]pyrimidin-4-yl}-4-(pyridin-3-yl)piperidin-4-ol
N-[(1-ethyl-1H-imidazol-2-yl)methyl]-2-[3-(trifluoromethyl)phenoxymethyl]-1,3-oxazole-4-carboxamide
2-[4-(2-methylquinolin-4-yl)-2-(morpholin-4-ylmethyl)phenoxy]-N-(1,3-thiazol-2-ylmethyl)acetamide
8-[(2S)-2-hydroxypropanoyl]-3-(2-phenylethyl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
3-{[3-(dimethylamino)propyl](methyl)amino}-N-(2-phenylethyl)piperidine-1-carboxamide
ethyl 1-{2-[(5-methyl-1,3,4-thiadiazol-2-yl)sulfanyl]acetyl}-3-[(2E)-3-phenylprop-2-en-1-yl]piperidine-3-carboxylate
2-(4-fluorophenoxymethyl)-4-[3-(methoxymethyl)pyrrolidine-1-carbonyl]-1,3-oxazole
3-(1-{1-[(1-ethyl-5-methyl-1H-pyrazol-4-yl)methyl]piperidin-4-yl}-1H-pyrazol-5-yl)-1-(3-fluorophenyl)urea
N-{[2-(1H-1,3-benzodiazol-1-yl)pyridin-3-yl]methyl}-5H,6H,7H,8H,9H-[1,2,3,4]tetrazolo[1,5-a]azepine-9-carboxamide
2-[4-(5-ethyl-1,3,4-oxadiazol-2-yl)piperazin-1-yl]-4-(propan-2-yl)-6-(trifluoromethyl)pyrimidine
methyl 4-methyl-3-[(3-oxopiperazine-1-carbonyl)amino]benzoate
3-(3,4-difluorophenyl)-N,N-diethyl-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridine-5-sulfonamide
N-{[1-(2-methoxyethyl)-1H-imidazol-5-yl]methyl}-5-[(4H-1,2,4-triazol-3-ylsulfanyl)methyl]furan-2-carboxamide
4,6-dimethyl-1-{3-[2-(2-methylpropyl)-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-6-yl]-3-oxopropyl}-1,2-dihydropyrimidin-2-one
ethyl 4-[1-(4-fluorophenyl)-2,2-dimethylcyclopropaneamido]piperidine-1-carboxylate
N-[4-(1,3-benzoxazol-2-yl)phenyl]-1-benzylpiperidine-4-carboxamide
N-[(1-ethyl-1H-imidazol-2-yl)methyl]-1-[1-(pyridin-3-ylmethyl)piperidin-4-yl]piperidine-3-carboxamide
ethyl 1-[(2-amino-1,3-thiazol-4-yl)methyl]-4-oxo-5-phenoxy-1,4-dihydropyridine-3-carboxylate
(1S,5R)-3-(oxan-4-yl)-6-[4-(1H-1,2,4-triazol-3-yl)benzoyl]-3,6-diazabicyclo[3.2.2]nonane
2-ethyl-5-fluoro-1-{1-[(5-methylfuran-2-yl)methyl]piperidin-4-yl}-1H-1,3-benzodiazole
methyl 2-[N-methyl-1-(4-{[1-(2-phenylethyl)piperidin-4-yl]oxy}phenyl)formamido]acetate
N-[1-methyl-6-(propan-2-yloxy)-1H-indazol-3-yl]-2H-1,3-benzodioxole-5-carboxamide
2-(1-benzyl-3-oxopiperazin-2-yl)-N-(1,3-dihydroxypropan-2-yl)acetamide
[(4-ethyl-5-{1-[6-(methoxymethyl)pyridine-2-carbonyl]piperidin-4-yl}-4H-1,2,4-triazol-3-yl)methyl]dimethylamine
8-[(5-ethyl-1,3,4-oxadiazol-2-yl)methyl]-3-(2-phenoxyethyl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
7-(cyclobutylmethyl)-2-[(5-methoxy-4-oxo-4H-pyran-2-yl)methyl]-2,7-diazaspiro[4.5]decan-6-one
N-(3-methylphenyl)-3-{1-[3-(methylsulfanyl)propanoyl]piperidin-4-yl}propanamide
ethyl 2-[methyl({[1-(2-phenylethyl)-2-(propane-2-sulfonyl)-1H-imidazol-5-yl]methyl})amino]acetate
1-ethyl-4-[3-(piperidin-1-ylmethyl)piperidin-1-yl]piperidine
[(3R,5R)-1-(2-aminopyrimidin-4-yl)-5-{[(2-methoxyethyl)(methyl)amino]methyl}piperidin-3-yl]methanol
N-(furan-2-ylmethyl)-N,1-dimethyl-5-({[2-(trifluoromethyl)phenyl]methyl}amino)-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
ethyl 2,4-dimethyl-5-[2-(pyridin-2-yl)piperidine-1-carbonyl]-1H-pyrrole-3-carboxylate
2-[4-(1,4-dithiepan-6-yl)-1-[1-(propan-2-yl)piperidin-4-yl]piperazin-2-yl]ethan-1-ol
6-{4-[2-(cyclopent-1-en-1-yl)acetyl]-6-hydroxy-1,4-diazepan-1-yl}pyrazine-2-carboxamide
({1-[(2-fluorophenyl)methyl]-2-methanesulfonyl-1H-imidazol-5-yl}methyl)(furan-2-ylmethyl)(prop-2-yn-1-yl)amine
2-{3-[1-(but-3-en-1-yl)-1H-pyrazol-3-yl]phenyl}pyridine-3-carbonitrile
2-[2-methyl-3-(7-methyl-1H-1,3-benzodiazol-2-yl)-1H-indol-1-yl]acetamide
N-[(3,5-dimethyl-1-propyl-1H-pyrazol-4-yl)methyl]-3-(4-hydroxyphenyl)-1H-pyrazole-5-carboxamide
N-{[2-(morpholin-4-yl)pyridin-3-yl]methyl}-5-(pyrrolidin-2-yl)thiophene-2-carboxamide
4-({2-[5-(oxolan-2-yl)-1,2,4-oxadiazol-3-yl]ethyl}amino)-N-(propan-2-yl)pyridine-2-carboxamide
1-(2-{1-[(5-phenyl-1,2,4-oxadiazol-3-yl)methyl]piperidin-2-yl}ethyl)pyrrolidin-2-one
1-{1-[(6-chloro-2H-chromen-3-yl)methyl]piperidin-3-yl}pyrrolidin-2-one
(2S)-N-{[3-(thiophen-2-ylmethyl)-1,2,4-oxadiazol-5-yl]methyl}piperidine-2-carboxamide
5-methyl-5-phenyl-1-[(1-propyl-1H-pyrazol-4-yl)methyl]piperidin-2-one
N-[2-(3,6-dioxo-1,2,3,6-tetrahydropyridazin-1-yl)ethyl]-2,5,7-trimethylquinoline-4-carboxamide
3-methyl-1-(1-{[4-(pyrrolidin-1-ylmethyl)thiophen-2-yl]methyl}piperidin-4-yl)butan-1-ol
(3R,4S)-1-(2-methylpyrimidine-5-carbonyl)-4-propylpyrrolidin-3-amine
2-{[2-(1,3-benzothiazol-2-yloxy)hex-5-en-1-yl](methyl)amino}-N,N-dimethylacetamide
N-methyl-2-oxo-N-(pyrazin-2-ylmethyl)-1-[(1r,4r)-4-hydroxycyclohexyl]-2,3-dihydro-1H-1,3-benzodiazole-5-carboxamide