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(2S)-1-{[6-chloro-2-(1,2,3,4-tetrahydroisoquinoline-2-carbonyl)imidazo[1,2-a]pyridin-3-yl]methyl}pyrrolidine-2-carboxamide
4-(5-methylpyridin-2-yl)-1-{[2-(pyridin-2-yl)pyrimidin-5-yl]methyl}piperidin-4-ol
methyl 5-(cycloheptylamino)-3-(2-methoxyacetamido)-1-(3-phenylpropyl)-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
5-{4-[1-(morpholin-4-yl)ethyl]phenyl}-2,3-dihydro-1H-inden-1-one
3-(2-chlorophenyl)-4-{3-cyclopropyl-[1,2,4]triazolo[3,4-b][1,3,4]thiadiazol-6-yl}-5-methyl-1,2-oxazole
1-(2-hydroxy-3-{4-methoxy-2-[({[3-(propan-2-yl)-1,2-oxazol-5-yl]methyl}amino)methyl]phenoxy}propyl)piperidin-4-ol
4-[(4-methyl-1H-pyrazol-1-yl)methyl]-1-[7-(propan-2-yl)-[1,2,4]triazolo[1,5-a]pyrimidine-5-carbonyl]piperidine
(3R,4S)-1-(naphthalene-1-carbonyl)-4-propylpyrrolidin-3-amine
N-(2-fluoro-4-methylphenyl)-2-[4-(1-phenylethyl)-1H-1,2,3-triazol-1-yl]acetamide
N-[(2-chlorophenyl)methyl]-1-methyl-2-oxo-N-(prop-2-en-1-yl)-1,2,5,6,7,8-hexahydroquinoline-3-carboxamide
3-chloro-N-(3-ethoxypropyl)-4-[(1-methanesulfonylpiperidin-4-yl)oxy]benzamide
N-benzyl-5-[(2,3-dihydro-1H-inden-2-yl)amino]-N,1-dimethyl-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
1-[(5-{4-[(3,5-dimethyl-1H-pyrazol-1-yl)methyl]phenyl}-1,2,4-oxadiazol-3-yl)methyl]-4-methylpiperazine
methyl 2-({2-[6-(pyrrolidin-1-yl)pyrimidin-4-yl]ethyl}carbamoyl)piperidine-1-carboxylate
6-methyl-8-[(1R,6S)-9-methyl-3,9-diazabicyclo[4.2.1]nonane-3-carbonyl]-4-oxa-2,5-diazatricyclo[7.3.0.03,7]dodeca-1(9),2,5,7-tetraene
(3R,5S)-N-{1-[(3-methylphenyl)methyl]cyclopropyl}-5-(morpholine-4-carbonyl)piperidine-3-carboxamide
4-[3-(furan-2-yl)-1H-pyrazol-1-yl]-1-(pyridazine-3-carbonyl)piperidine-4-carboxylic acid
(1S,5R)-3-[(4-methoxyphenyl)methyl]-6-(5-methylthiophene-3-carbonyl)-3,6-diazabicyclo[3.2.2]nonane
2-{1-[(2-chloro-4-fluorophenyl)methyl]-3-oxopiperazin-2-yl}-N-[2-(2-oxo-1,3-oxazolidin-3-yl)ethyl]acetamide
1-(2-{1-[2-(3,4-dimethoxyphenyl)acetyl]piperidin-2-yl}ethyl)-N-(propan-2-yl)-1H-1,2,3-triazole-4-carboxamide
N-{[4-benzyl-5-(methylsulfanyl)-4H-1,2,4-triazol-3-yl]methyl}-2-(thiophen-3-yl)acetamide
(3S,4R)-4-(2H-1,3-benzodioxol-5-yl)-1-[(4-acetamidophenyl)methyl]pyrrolidine-3-carboxylic acid
[(4-fluorophenyl)methyl][2-methyl-2-(morpholin-4-ylmethyl)propyl](pyridin-4-ylmethyl)amine
[(1,3-dimethyl-1H-pyrazol-5-yl)methyl][(3-methylthiophen-2-yl)methyl](pyridin-2-ylmethyl)amine
{2-[3-(4-methyl-1H-1,3-benzodiazol-2-yl)piperidin-1-yl]-1,3-thiazol-4-yl}methanol
(3S,4R)-4-(pyridin-3-yl)-1-[2-(1H-1,2,3,4-tetrazol-5-yl)benzoyl]pyrrolidine-3-carboxylic acid
1-(3-chlorophenyl)-4-(2-ethylpyrimidine-5-carbonyl)-5-methylpiperazin-2-one
1-{[1-(2-methoxyethyl)-1H-imidazol-5-yl]methyl}-4-phenyl-5-[1-(prop-2-en-1-yl)-1H-pyrazol-4-yl]-1H-imidazole
{[1-({1-[(2-fluoro-5-methylphenyl)methyl]piperidin-4-yl}methyl)-1H-1,2,3-triazol-4-yl]methyl}urea
5-[(4aS,7aR)-6,6-dioxo-4-propyl-octahydro-6λ6-thieno[3,4-b]piperazine-1-carbonyl]pyridine-2-carbonitrile
(2E)-1-[7-(cyclohexylmethyl)-2,7-diazaspiro[4.5]decan-2-yl]-3-(pyridin-4-yl)prop-2-en-1-one
3-[(4-butyl-3-oxopiperazin-1-yl)methyl]-6-methyl-1,2-dihydroquinolin-2-one
3-(5-methyl-1H-pyrazol-1-yl)-1-[(1S,5R)-3-(oxan-4-yl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]propan-1-one
[(3R,4S)-4-{[(2R,6S)-2,6-dimethylmorpholin-4-yl]methyl}-1-[(4-fluoro-3-methylphenyl)methyl]pyrrolidin-3-yl]methanol
2-{1-[(2-chloro-4-fluorophenyl)methyl]-3-oxopiperazin-2-yl}-N-(oxan-4-yl)acetamide
4-ethyl-3-{[1-(2-propyl-1,3-thiazole-4-carbonyl)piperidin-4-yl]methyl}-4,5-dihydro-1H-1,2,4-triazol-5-one
1-(1-benzothiophen-3-ylmethyl)-4-(hydroxymethyl)azepan-4-ol
2,3-dimethyl-5-phenyl-N-[3-(1H-1,2,3-triazol-1-yl)propyl]pyrazolo[1,5-a]pyrimidin-7-amine
1-[(4-phenylphenyl)methyl]-4-(pyridin-4-ylmethyl)-1,4-diazepan-5-one
1-[4-(3-methyl-2-oxoimidazolidin-1-yl)phenyl]-3-{1-[5-(propan-2-yl)-1,3,4-oxadiazol-2-yl]ethyl}urea
6-[(2-fluorophenyl)methoxy]-1-[(4-methoxyphenyl)methyl]-4-{pyrazolo[1,5-a]pyrimidine-2-carbonyl}-1,4-diazepan-2-one
N-[(1-methyl-1,2,3,4-tetrahydroquinolin-6-yl)methyl]-2-oxo-6-({1,3,3-trimethyl-6-azabicyclo[3.2.1]octan-6-yl}methyl)-1,2-dihydropyridine-3-carboxamide
N-cyclohexyl-4-(cyclopropylmethyl)-5-oxo-3-(propan-2-yl)-1,4-diazepane-1-carboxamide
N-{[2-(1H-imidazol-1-yl)pyridin-3-yl]methyl}-7-(propan-2-yl)-[1,2,4]triazolo[1,5-a]pyrimidine-5-carboxamide
N-[(3R,4S)-4-cyclopropyl-1-(oxan-4-yl)pyrrolidin-3-yl]-1-(1H-imidazol-1-ylmethyl)cyclopropane-1-carboxamide
4-[(2-hydroxyethyl)sulfamoyl]-N-methyl-N-[(1-methyl-1H-pyrazol-4-yl)methyl]benzamide
6,7-dimethoxy-2-[1-(pyridin-2-ylmethyl)piperidin-3-yl]-1,2,3,4-tetrahydroisoquinoline
7-(2-cyclohexylethyl)-2-[2-(pyridin-3-yl)acetyl]-2,7-diazaspiro[4.5]decan-6-one
2-({6-oxo-1-[2-(pyridin-2-yl)ethyl]piperidin-3-yl}formamido)acetamide
N-[1-(pyridin-3-ylmethyl)azepan-4-yl]-2-(1,2,3,4-tetrahydroisoquinolin-2-yl)acetamide