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1-[3-(3-methyl-1H-pyrazol-1-yl)propanoyl]-4-{[2-(trifluoromethyl)phenyl]methyl}-1,4-diazepan-5-one
3-{3-[methyl(2-methylpropyl)amino]propyl}-8-[(2S)-pyrrolidine-2-carbonyl]-1-oxa-3,8-diazaspiro[4.5]decan-2-one
3-[(2S,6S)-6-(hydroxymethyl)-8-oxa-4-azatricyclo[7.4.0.02,6]trideca-1(9),10,12-triene-4-carbonyl]-2-methyl-4,5,6,7-tetrahydro-1H-indol-4-one
1-(2-methylpropyl)-N-{1-[3-(pyridin-2-yl)-1,2,4-oxadiazol-5-yl]ethyl}piperidin-4-amine
N-[2-methyl-3-(3-methyl-1,2,4-oxadiazol-5-yl)phenyl]furan-2-carboxamide
1-[2-(1H-imidazol-1-yl)propanoyl]-3',4'-dihydro-1'H-spiro[piperidine-4,2'-quinoxaline]-3'-one
7-cyclohexyl-2-(pyrazin-2-yl)-2,7-diazaspiro[4.5]decan-6-one
N3-ethyl-N5-[(5-fluoro-2-methylphenyl)methyl]-4-oxo-1-(2-phenylethyl)-1,4-dihydropyridine-3,5-dicarboxamide
4-[(2-chloro-4-fluorophenyl)methyl]-2-(morpholin-4-ylmethyl)-1,4-oxazepane
(3R,4S)-1-{2-[2-(3-methoxyphenyl)ethyl]benzoyl}-3,4-dimethylpiperidin-4-ol
N-{[6-chloro-4-(pyrrolidin-1-yl)quinazolin-2-yl]methyl}-1-[(1S,4R)-7,7-dimethyl-2-oxobicyclo[2.2.1]heptan-1-yl]methanesulfonamide
1-(cyclopropylmethyl)-5-(2,3-difluoro-4-methylphenyl)-1H,4H-pyrazolo[3,4-d]imidazole
[(2-methylphenyl)methyl](prop-2-en-1-yl)(pyridin-3-ylmethyl)amine
4-{[3-(difluoromethoxy)phenyl]methyl}-1-(4-methoxyphenyl)piperazin-2-one
1-{5-[(3R,4R)-3-cyclobutyl-3-hydroxy-4-methylpyrrolidine-1-carbonyl]-2-methylphenyl}imidazolidin-2-one
4-(cyclopropylmethyl)-1-[(2,3,6-trifluorophenyl)methyl]-1,4-diazepan-5-one
ethyl 4-(5-cyclopropyl-1,3,4-oxadiazol-2-yl)piperazine-1-carboxylate
6-[(2E)-3-(2,3-difluorophenyl)prop-2-enoyl]-N-[2-(pyridin-2-yl)ethyl]-6-azaspiro[2.5]octane-1-carboxamide
5-ethyl-N-{[1-(1H-imidazol-1-ylmethyl)cyclopropyl]methyl}pyrimidin-2-amine
5-[3-(1H-pyrazol-1-ylmethyl)benzoyl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carboxylic acid
(2S)-N-(2-hydroxyethyl)-2-methoxy-2-phenyl-N-[(2E)-3-phenylprop-2-en-1-yl]acetamide
2-({1-[(2,3-difluorophenyl)methyl]piperidin-4-yl}oxy)-4-methoxy-N-(2-methoxyethyl)benzamide
1-{1-[(2Z)-2-chloro-3-phenylprop-2-en-1-yl]piperidin-4-yl}-N-(2-hydroxyethyl)-N-methyl-1H-1,2,3-triazole-4-carboxamide
2-fluoro-N-(oxolan-2-ylmethyl)-N-({3-[2-(thiophen-3-yl)ethoxy]phenyl}methyl)benzene-1-sulfonamide
(3R,9aR)-3-(hydroxymethyl)-8-[(6-methylpyridin-2-yl)methyl]-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
2,3,5-trimethyl-N-{2-[(1-methyl-1H-imidazol-2-yl)sulfanyl]ethyl}pyrazolo[1,5-a]pyrimidin-7-amine
N-(2-methyl-1-{5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}propyl)-2,3-dihydro-1-benzofuran-7-carboxamide
3-(pentan-2-yl)-8-{pyrazolo[1,5-a]pyrimidine-3-carbonyl}-1-oxa-3,8-diazaspiro[4.5]decan-2-one
7-(3,5-dichloro-2-methoxybenzoyl)-3-methyl-1-oxa-3,7-diazaspiro[4.4]nonan-2-one
4-[1-(3-methoxyphenyl)-1H-pyrazol-4-yl]-2-[3-(1H-pyrazol-1-yl)azetidin-1-yl]pyrimidine
(3R,4R)-3-cyclopropyl-4-methyl-1-(2-phenoxyethyl)pyrrolidin-3-ol
2-[2-(pyridin-3-yl)ethyl]-9-[2-(pyrrolidin-1-yl)acetyl]-2,9-diazaspiro[5.5]undecan-3-one
5-cyclobutyl-N-(2-{4-methyl-5H,6H,7H-cyclopenta[d]pyrimidin-2-yl}ethyl)-1,3,4-oxadiazol-2-amine
4-[3-(3-methylphenoxymethyl)piperidine-1-carbonyl]benzonitrile
2-(5-acetylthiophen-3-yl)-N-[3-(4-methoxyphenyl)propyl]acetamide
5-ethyl-2-{4-phenyl-1-[3-(1H-1,2,3,4-tetrazol-5-yl)propyl]-1H-imidazol-5-yl}pyridine
4-{2-[(cyclopropylmethyl)sulfanyl]acetyl}-1,9-dimethyl-1,4,9-triazaspiro[5.6]dodecan-10-one
N5-cyclopentyl-N6-[2-methyl-2-(morpholin-4-yl)propyl]-[1,2,5]oxadiazolo[3,4-b]pyrazine-5,6-diamine
(2R,6R)-11-methoxy-4-[2-(pyrrolidin-1-yl)acetyl]-8-oxa-4-azatricyclo[7.4.0.02,6]trideca-1(13),9,11-triene-6-carboxylic acid
1-(prop-2-en-1-yl)-4-{4-[2-(pyridin-4-yl)ethyl]piperazine-1-carbonyl}pyrrolidin-2-one
1-[(3-methoxyphenyl)methyl]-6-oxo-N-{[2-(1H-pyrazol-1-ylmethyl)phenyl]methyl}piperidine-3-carboxamide
N-[2-(dimethylamino)ethyl]-N-ethyl-2-(4-fluorophenyl)imidazo[1,2-a]pyridine-6-carboxamide
3-(3,4-dimethoxyphenyl)-N,N-bis(prop-2-en-1-yl)-5-(1H-1,2,3,4-tetrazol-1-yl)benzamide
3-{4-[(4-fluorophenyl)methyl]-3-(propan-2-yl)-1,4-diazepan-1-yl}propanamide
3-{2-[4-(4-chlorophenyl)piperazin-1-yl]ethyl}-4-(dimethyl-1,2-oxazol-4-yl)-4,5-dihydro-1H-1,2,4-triazol-5-one
1-{[3-(methoxymethyl)-1,2,4-oxadiazol-5-yl]methyl}-3,3-diphenylpiperidine
2-amino-2-methyl-1-[3-(4-phenoxybenzoyl)piperidin-1-yl]propan-1-one
(4aS,7aR)-1-{8-methylimidazo[1,2-a]pyridine-2-carbonyl}-4-propyl-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
N-{1-[5-(trifluoromethyl)pyridin-2-yl]piperidin-3-yl}cyclohex-1-ene-1-carboxamide
4-methyl-N-[(5-oxopyrrolidin-2-yl)methyl]-N,2-bis(propan-2-yl)pyrimidine-5-carboxamide