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(3S,9aR)-8-{[4-methoxy-3-(methoxymethyl)phenyl]methyl}-2,3-dimethyl-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
N-(2-{4-methyl-5H,6H,7H-cyclopenta[d]pyrimidin-2-yl}ethyl)-1H-pyrrolo[2,3-b]pyridin-6-amine
N'-cycloheptyl-N-ethyl-N-(2-methylprop-2-en-1-yl)butanediamide
4-(3-methoxyphenyl)-3-[1-(propan-2-yloxy)ethyl]-4,5-dihydro-1H-1,2,4-triazol-5-one
4-{[2-(4-methoxyphenyl)-8-methylquinolin-3-yl]methyl}-1-methylpiperazin-2-one
8-[(6-ethoxypyridin-3-yl)methyl]-2,8-diazaspiro[4.5]decan-3-one
N-[(7R,8aS)-2-methyl-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-2-oxobutanamide
N-[(3R,7S,8aS)-3-(2-methylpropyl)-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-3-chlorothiophene-2-carboxamide
N-[(6-chloro-1H-1,3-benzodiazol-2-yl)methyl]oxolane-3-carboxamide
2-(3-hydroxyphenyl)-2-(4-phenyl-1,2,3,6-tetrahydropyridin-1-yl)acetic acid
(3S,4R)-4-(2-methoxyphenyl)-1-[1-(propan-2-yl)-1H-pyrazole-4-carbonyl]pyrrolidine-3-carboxylic acid
(3aR,6aR)-2-[2-(2H-1,3-benzodioxol-5-yl)acetyl]-5-(2-methoxyethyl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
N-(1-{imidazo[2,1-b][1,3]thiazol-6-yl}ethyl)-2-oxo-1,2,5,6,7,8-hexahydroquinoline-3-carboxamide
1-[7-(1-benzothiophen-3-yl)-9-(oxolan-3-yloxy)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]-2-ethylbutan-1-one
1-(2-fluoro-4-methylbenzoyl)-4-[4-(3-methylphenyl)-1H-pyrazol-5-yl]piperidine
2-cyclopropyl-N-[4-(dimethylamino)phenyl]-3-oxo-2,9-diazaspiro[5.5]undecane-9-carboxamide
2-propyl-N-[1-(pyrazin-2-yl)propan-2-yl]-1,3-thiazole-4-carboxamide
5-[2-(aminomethyl)-7-fluoro-2,3-dihydro-1-benzofuran-5-yl]-1,3,6-trimethyl-1,2,3,4-tetrahydropyrimidine-2,4-dione
2-{[(3R,4R)-4-amino-3-hydroxypiperidin-1-yl]methyl}-6-fluoro-1,4-dihydroquinolin-4-one
(3S,4S)-1-[(2-cyclohexylpyrimidin-5-yl)methyl]-4-(pyridin-2-yl)pyrrolidine-3-carboxylic acid
5-(2-{1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl}-2-oxoethyl)-3-methyl-1,2,3,4-tetrahydropyrimidine-2,4-dione
5-[5-(1-cyclopropanecarbonylpiperidin-4-yl)-1,2,4-oxadiazol-3-yl]-1H-1,3-benzodiazole
4-{[4-(4-methanesulfonylpiperazine-1-carbonyl)furan-2-yl]methyl}morpholine
5-(1-benzofuran-2-yl)-N-[2-(dimethyl-1,3-thiazol-2-yl)ethyl]-1,2,4-triazin-3-amine
3-{2-[6-(methylsulfanyl)-1,2,3,4-tetrahydroisoquinolin-2-yl]ethyl}-2,3-dihydro-1,3-benzoxazol-2-one
3-butyl-4-ethyl-1-(2-oxo-2-{4-oxo-3H,4H,5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-7-yl}ethyl)-4,5-dihydro-1H-1,2,4-triazol-5-one
N-[(2S)-3-(1H-imidazol-4-yl)-1-oxo-1-{4-[2-(1H-1,2,4-triazol-1-yl)ethyl]piperazin-1-yl}propan-2-yl]acetamide
2-[4-(1H-indazole-3-carbonyl)-1-(2-phenylethyl)piperazin-2-yl]ethan-1-ol
[(6-chloro-2H-1,3-benzodioxol-5-yl)methyl][1-(5-methyl-1-phenyl-1H-pyrazol-4-yl)ethyl]amine
N-{2-[(2-methylquinolin-8-yl)oxy]ethyl}-3-(4H-1,2,4-triazol-4-yl)benzamide
4-{1-[1-(2-methoxyethyl)piperidin-4-yl]piperidine-3-carbonyl}morpholine
2-{1-cyclopentyl-4-[(5-methoxy-3-methyl-1H-indol-2-yl)methyl]piperazin-2-yl}ethan-1-ol
3-(3-hydroxy-3-methylbutyl)-N-[(6-methoxy-1H-1,3-benzodiazol-2-yl)methyl]benzamide
1-{3-[(4-fluorophenyl)amino]piperidin-1-yl}-3-(1H-1,2,3,4-tetrazol-1-yl)propan-1-one
8-[2-(2-methyl-1H-imidazol-1-yl)acetyl]-2-(pyridin-3-ylmethyl)-2,8-diazaspiro[5.5]undecan-3-one
2-{1-[(4-fluorophenyl)methyl]-3-oxopiperazin-2-yl}-N-{[4-(2-oxopyrrolidin-1-yl)phenyl]methyl}acetamide
2,5-dimethyl-3-[4-(5-phenyl-1,2-oxazole-3-carbonyl)piperazin-1-yl]pyrazine
N-(4-cyclohexylphenyl)-4-[2-(1H-1,2,4-triazol-1-yl)ethyl]piperazine-1-carboxamide
2-(2-chlorophenyl)-N,3-dimethyl-N-(1,3-thiazol-2-ylmethyl)-3H-imidazo[4,5-b]pyridine-6-carboxamide
4-{1-[2-(4-methyl-1,4-diazepan-1-yl)acetyl]piperidin-3-yl}benzoic acid
8-{[4-(difluoromethoxy)phenyl]methyl}-2-(2-methylpropyl)-2,8-diazaspiro[4.5]decan-3-one
N-[2-(3,4-dimethoxyphenyl)ethyl]-N,2-dimethyl-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
methyl[3-(1-methyl-1H-imidazol-2-yl)propyl]({3-phenylpyrazolo[1,5-a]pyrimidin-6-yl}methyl)amine
(2R,3R,6R)-3-(3,5-difluorophenyl)-5-[(4-methyl-1H-imidazol-5-yl)methyl]-1,5-diazatricyclo[5.2.2.02,6]undecane
7-(1,3-benzothiazol-2-yl)-4-[(2,4-dimethoxyphenyl)methyl]-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
{[1-butyl-2-(4-methylpentanesulfonyl)-1H-imidazol-5-yl]methyl}[(1-ethylpyrrolidin-3-yl)methyl]methylamine
4-{4-[2-(methoxymethyl)piperidine-1-carbonyl]phenyl}-2-methylbutan-2-ol
N-cyclopropyl-3-{2-ethyl-4-phenyl-2,9-diazaspiro[5.5]undecan-9-yl}propanamide
ethyl[(1-methyl-1H-imidazol-2-yl)methyl][3-(5-methylfuran-2-yl)butyl]amine
6-fluoro-4-{1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-5-carbonyl}-1,2-dihydroquinolin-2-one