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2-(1-methyl-1H-pyrrol-2-yl)-2-oxo-N-[2-(1H-1,2,4-triazol-5-ylsulfanyl)ethyl]acetamide
1-({3-[2-(1,3-thiazol-2-yl)piperidine-1-carbonyl]-1,2-oxazol-5-yl}methyl)piperidin-4-ol
2-(1-methylpyrrolidin-3-yl)-9-(thiophen-2-ylmethyl)-2,9-diazaspiro[5.5]undecan-3-one
1-[(3-chlorophenyl)methyl]-4-[4-(1H-pyrazol-3-yl)benzoyl]piperazine
3-phenyl-8-{thieno[3,2-d]pyrimidin-4-yl}-1,8-diazaspiro[4.5]decan-2-one
4-(oxolane-2-carbonyl)-7-(pyridin-3-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
2-(3-{[4-(2-methylpyridin-4-yl)-1,4-diazepan-1-yl]methyl}phenoxy)acetamide
N-[2-(4-benzylpiperazin-1-yl)ethyl]-5,7-dimethylpyrido[2,3-d]pyrimidin-4-amine
3-[3-(2-fluorophenyl)-1,2,4-oxadiazol-5-yl]-1-[(2S)-2-(pyrrolidin-1-ylmethyl)pyrrolidin-1-yl]propan-1-one
2-amino-4-(2-methyl-1H-imidazol-4-yl)-6-phenyl-5,6,7,8-tetrahydroquinoline-3-carbonitrile
2-(3-fluorophenyl)-N-({7-[(2,3,4-trimethoxyphenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}methyl)acetamide
N-({3-[2-(4-fluorophenyl)ethoxy]phenyl}methyl)-4-(2-oxopyrrolidin-1-yl)-N-(pyridin-4-ylmethyl)benzamide
3-(2-{1-methyl-2-oxo-1,2-dihydrospiro[indole-3,4'-piperidine]-1'-yl}-2-oxoethyl)-1,3-diazinane-2,4-dione
4-cyclopentyl-N-methyl-N-[(4-methyl-4H-1,2,4-triazol-3-yl)methyl]pyrimidin-2-amine
2-{1-[(2-fluoro-4-methoxyphenyl)methyl]-3-oxopiperazin-2-yl}-N-methyl-N-(2-phenylethyl)acetamide
2-{1-[(3,5-dimethoxyphenyl)methyl]-3-oxopiperazin-2-yl}acetamide
1-ethyl-N-(3-hydroxypropyl)-N-[(5-methylthiophen-2-yl)methyl]-3-(propan-2-yl)-1H-pyrazole-5-carboxamide
ethyl 4-(2-methoxyethyl)-1-{5-[(methylsulfanyl)methyl]furan-2-carbonyl}piperidine-4-carboxylate
1-(3-chlorophenyl)-4-[(3-{2-[1-(pyridine-2-carbonyl)piperidin-2-yl]ethoxy}phenyl)methyl]piperazine
9-[(3-fluoro-4-methylphenyl)methyl]-2-[2-(pyridin-2-yl)ethyl]-2,9-diazaspiro[5.5]undecan-3-one
1-(4-{[2-(3-methoxyphenyl)ethyl]amino}-5-methylthieno[2,3-d]pyrimidine-6-carbonyl)-N,N-dimethylpyrrolidin-3-amine
(5S)-5-{[(pyridin-3-ylmethyl)(4,5,6,7-tetrahydro-1,3-benzothiazol-2-ylmethyl)amino]methyl}pyrrolidin-2-one
4-(2-{5H,6H-imidazo[2,1-b][1,3]thiazol-3-yl}acetyl)-3-methyl-1-(2-methylpropyl)piperazin-2-one
{[5-(oxolan-2-yl)thiophen-2-yl]methyl}[(3-phenyl-1,2,4-oxadiazol-5-yl)methyl](prop-2-en-1-yl)amine
3-hydroxy-2-methyl-N-{[1-(3,3,3-trifluoropropyl)piperidin-4-yl]methyl}benzamide
5-fluoro-4-(pyrrolidin-1-yl)-2-{4-[2-(1H-1,2,4-triazol-1-yl)ethyl]piperazin-1-yl}pyrimidine
N-methyl-6-(morpholin-4-yl)-N-[2-(oxan-2-yl)ethyl]pyrimidin-4-amine
N-{1-[1-(2-methoxyphenyl)-3-(propan-2-yl)-1H-1,2,4-triazol-5-yl]-2-methylpropyl}acetamide
2-[3-(3-chlorophenyl)-1-methyl-1H-pyrazol-4-yl]-4-methyl-1H-1,3-benzodiazole
2-(2-{4-[(5-ethylpyridin-2-yl)methyl]piperazin-1-yl}-1H-1,3-benzodiazol-1-yl)ethan-1-ol
4-{[5-(4-methyl-1,3-thiazole-5-carbonyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl]methyl}thiomorpholine
8-fluoro-2-({[1-(4-methanesulfonylphenyl)ethyl]amino}methyl)quinolin-4-ol
5-[(4-{5-[3-(trifluoromethyl)phenyl]pyrimidin-4-yl}piperidin-1-yl)methyl]-2,1,3-benzothiadiazole
1-{[4-(3-hydroxy-3-methylbutyl)phenyl]methyl}-4-(pyridin-3-yl)piperidin-4-ol
2-({2-[5-(1-ethyl-1H-1,2,4-triazol-5-yl)-4-phenyl-1H-imidazol-1-yl]ethyl}amino)-6-methyl-3,4-dihydropyrimidin-4-one
1-{[1-(3-methoxypropyl)pyrrolidin-3-yl]methyl}-3-(2-methyl-1-benzofuran-7-yl)urea
4-(5-propylpyrimidin-4-yl)-N-(pyridin-3-ylmethyl)-1H-pyrrolo[2,3-b]pyridin-6-amine
N-({2-[(methylsulfanyl)methyl]-1,3-thiazol-4-yl}methyl)-2-oxo-1-oxaspiro[4.4]nonane-4-carboxamide
6-(2-aminoethyl)-2-methyl-N-{1-[3-(2-methylphenyl)-1,2,4-oxadiazol-5-yl]ethyl}pyrimidin-4-amine
N-cyclopropyl-3-[1-(naphthalene-1-carbonyl)piperidin-4-yl]propanamide
2-(2-{1-[(dimethyl-1,2-oxazol-4-yl)methyl]piperidin-2-yl}ethyl)pyridine
3-{1-[(1-ethyl-1H-pyrazol-4-yl)methyl]piperidin-4-yl}-N-[(1-ethylpyrrolidin-2-yl)methyl]propanamide
4-(3,5-dimethoxyphenyl)-2,6-dimethylpyridine
2-(2-aminoethyl)-N-[(2-ethoxy-3-methoxyphenyl)methyl]quinazolin-4-amine
3-(2,5-dioxoimidazolidin-4-yl)-N-{2-[(2-methylquinolin-8-yl)oxy]ethyl}propanamide
3-(2H-1,3-benzodioxol-5-yl)-1-[(1S,5R)-3-cyclobutanecarbonyl-3,6-diazabicyclo[3.2.2]nonan-6-yl]propan-1-one
N-(3-butoxyphenyl)azetidine-1-carboxamide
4-{imidazo[1,2-a]pyridine-6-amido}-N-phenylpiperidine-1-carboxamide
2-(4-{[(3R,5S)-5-(hydroxymethyl)-1-methylpyrrolidin-3-yl]amino}-6-methylpyrimidin-2-yl)phenol
2-({[2-hydroxy-2-(pyridin-2-yl)ethyl]amino}methyl)-6,8-dimethylquinolin-4-ol