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2-(3-methoxypropyl)-8-(1H-pyrrole-3-carbonyl)-2,8-diazaspiro[4.5]decan-3-one
N-{[1-(2-fluorophenyl)-1H-pyrazol-4-yl]methyl}-N-[(1-methyl-1H-imidazol-2-yl)methyl]cyclopropanamine
6-(2-methyl-1,4-oxazepane-4-carbonyl)-1,2,3,4-tetrahydroquinoxaline-2,3-dione
1-(3-chlorophenyl)-5-methyl-4-[3-(4-methyl-1,3-thiazol-5-yl)propanoyl]piperazin-2-one
4-(1-{[3-(4-phenylphenyl)-1H-pyrazol-4-yl]methyl}piperidin-4-yl)morpholine
3-(3-methoxyphenyl)-1-(pyridin-2-ylmethyl)-6-(1,3-thiazole-4-carbonyl)-1,2,5,6,7,8-hexahydro-1,6-naphthyridin-2-one
2-[(3S)-3-hydroxypyrrolidin-1-yl]-1-methyl-N-[2-(1-methyl-1H-1,2,4-triazol-5-yl)ethyl]-1H-1,3-benzodiazole-5-carboxamide
dimethyl({4-methyl-5-[1-(4-methylphthalazin-1-yl)piperidin-3-yl]-4H-1,2,4-triazol-3-yl}methyl)amine
[(2-cyclohexylpyrimidin-5-yl)methyl](methyl)[2-(2-methyl-1H-imidazol-1-yl)ethyl]amine
4-[(2,3-difluoro-6-methoxyphenyl)methyl]-1-methyl-2-phenylpiperazine
2-[2-(1-carbamoylethoxy)phenyl]-N,N-bis(propan-2-yl)benzamide
2-[4-(dimethylamino)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidine-7-carbonyl]-5-(1H-1,2,3,4-tetrazol-1-yl)phenol
3-({[(3,4-dimethoxyphenyl)methyl]amino}methyl)-7-fluoro-1-(pyridin-2-ylmethyl)-1,2-dihydroquinolin-2-one
3-(6-aminopyrimidin-4-yl)-5-[2-(piperidin-2-yl)ethyl]phenol
{[2-(2,4-difluorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}(2,3-dihydro-1,4-benzodioxin-2-ylmethyl)methylamine
4-{3-[(2-methoxyethyl)(methyl)amino]propanoyl}-1-(4-methylphenyl)piperazin-2-one
methyl (2S,4R)-4-[3-(3,5-dimethyl-1H-pyrazol-1-yl)benzamido]-1-[(2-ethoxyphenyl)methyl]pyrrolidine-2-carboxylate
methyl 9-[(1-methyl-5-oxopyrrolidin-3-yl)methoxy]-3-{[4-(2-methylpropyl)phenyl]methyl}-7-oxo-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
2-amino-2-methyl-1-{4-[4-methyl-5-(1H-pyrazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}propan-1-one
2-{[1-(2-methylpyridin-4-yl)-3-(propan-2-yl)-1H-1,2,4-triazol-5-yl]methyl}-2H-1,2,3-benzotriazole
1'-(5-fluoro-1H-indole-3-carbonyl)-2,3-dihydrospiro[indene-1,4'-piperidine]-2-ol
4-{[2-(3-methyl-1,2-oxazol-5-yl)pyrrolidin-1-yl]methyl}-1H-pyrazole-3-carboxylic acid
2-methyl-2-(2-{[2-(1-methylpyrrolidin-2-yl)ethyl]amino}-4-(morpholin-4-yl)pyrimidin-5-yl)propanoic acid
[(3R,4R)-4-{[(2-methoxyethyl)(methyl)amino]methyl}-1-[3-(trifluoromethyl)pyridin-2-yl]pyrrolidin-3-yl]methanol
1-{2-[(1R,5R)-6-(cyclopropylmethyl)-3,6-diazabicyclo[3.2.2]nonan-3-yl]-4-methylpyrimidin-5-yl}ethan-1-one
2-[(2R,6S)-2,6-dimethylmorpholin-4-yl]-N-[2-(4-hydroxyphenyl)-2-oxoethyl]-N-methylacetamide
N-benzyl{[3-(1H-imidazol-5-yl)phenyl]amino}sulfonamide
N-[1-(3-fluorophenyl)-6,6-dimethyl-4,5,6,7-tetrahydro-1H-indazol-4-yl]-2-(2-methyl-1,3-thiazol-4-yl)acetamide
N-(4-{[7-(3-phenylpropyl)-2,7-diazaspiro[4.5]decan-2-yl]methyl}phenyl)acetamide
methyl 2-{3-[(3-ethylphenyl)carbamoyl]propanamido}-2-methylpropanoate
N-[(7-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]-4-oxo-4H-chromene-2-carboxamide
2-ethoxy-3-[3-(2-methylpiperidin-1-yl)azetidine-1-carbonyl]pyridine
N-[4-(methylsulfanyl)phenyl]-4-(4-phenyl-1H-1,2,3-triazol-1-yl)piperidine-1-carboxamide
N-[(1-methylpyrrolidin-3-yl)methyl]-3-phenoxypropanamide
methyl[4-(morpholin-4-yl)butyl]{[3-(2,3,4-trimethoxyphenyl)-1,2,4-oxadiazol-5-yl]methyl}amine
N-[1-(2-chlorophenyl)cyclopropyl]-2-(morpholin-4-yl)-2-(pyridin-3-yl)acetamide
4-{3-[1-(2-methoxyethyl)-1H-imidazol-2-yl]piperidin-1-yl}-3-methylpyridine
4-[(9aS)-octahydro-1H-pyrrolo[1,2-a][1,4]diazepine-2-carbonyl]-3-(3-methoxyphenyl)-1H-pyrazole
2-(naphthalen-1-yl)-N-[(1r,4r)-4-methoxycyclohexyl]acetamide
N-ethyl-5-(2-fluorophenoxymethyl)-N-[(3S,4R)-4-hydroxyoxolan-3-yl]-1H-pyrazole-3-carboxamide
N-[2-(3,4-dimethoxyphenyl)ethyl]-1-[5-(methoxymethyl)furan-2-carbonyl]-N-methylpiperidin-3-amine
2-(4-{[3-(3,5-dimethyl-1H-pyrazol-4-yl)propyl]amino}piperidin-1-yl)pyridine-4-carbonitrile
3-{4-[5-(propan-2-yl)pyrazolo[1,5-a]pyrimidin-7-yl]piperazin-1-yl}propanamide
1-benzyl-8-[(3-methoxyphenyl)methyl]-3-(pyridin-2-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
1-{2-[(5-ethylpyrimidin-2-yl)oxy]hex-5-en-1-yl}piperidine-4-carboxylic acid
1-(4-{[2-(9H-fluoren-2-yl)-1H-imidazol-1-yl]methyl}piperidin-1-yl)ethan-1-one
N-(1-benzothiophen-5-ylmethyl)-3-(4-methyl-4H-1,2,4-triazol-3-yl)propanamide
6-{[(2-amino-1,3-thiazol-4-yl)methyl]amino}-N-[3-(pyridin-2-yl)propyl]pyridine-3-carboxamide
3-cyclohexyl-N-[3-(1-methyl-1H-pyrazol-4-yl)propyl]-1H-pyrazole-4-carboxamide
[4-(1H-1,2,3-benzotriazole-5-carbonyl)-1,4-oxazepan-6-yl]methanol