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3-{[1-(oxolan-3-ylmethyl)piperidin-4-yl]oxy}pyridine
3-{3-[2-(2,4-difluorophenyl)ethyl]piperidine-1-carbonyl}pyridin-1-ium-1-olate
(3aS,6aR)-3-[2-(4-fluorophenyl)ethyl]-5-[(2-propylpyrimidin-5-yl)methyl]-hexahydro-2H-pyrrolo[3,4-d][1,3]oxazol-2-one
N-[3-(cyclohexylsulfanyl)propyl]-4-methyl-2-(pyridin-3-yl)pyrimidine-5-carboxamide
4-[4-(1-ethoxyethyl)phenyl]-3,5-dimethyl-1H-pyrazole
6-methoxy-1-methyl-N-[(5-methylpyrazin-2-yl)methyl]-1H-indole-2-carboxamide
N-[3-(dimethylamino)-2,2-dimethylpropyl]-3-[(3-hydroxyazetidin-1-yl)sulfonyl]benzamide
3-(5-{[3-(2-methylphenoxy)azetidin-1-yl]methyl}furan-2-yl)-1H-pyrazole
(2-{2-[1-(1H-indole-6-carbonyl)piperidin-4-yl]-1H-imidazol-1-yl}ethyl)dimethylamine
1-(cyclohexylmethyl)-6-oxo-N-{[1-(piperidin-1-yl)cyclopentyl]methyl}piperidine-3-carboxamide
(3aS,6aS)-2-ethyl-5-{[3-(2-hydroxyethoxy)phenyl]methyl}-1-oxo-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
1-oxo-N-(oxolan-2-ylmethyl)-N-[(2E)-3-phenylprop-2-en-1-yl]-1,2-dihydroisoquinoline-4-carboxamide
4-{[4-(furan-2-carbonyl)-1,4-diazepan-1-yl]methyl}-1H-pyrazole-3-carboxylic acid
(1R,2S,9R)-11-[3-(pyrrolidine-1-carbonyl)pyridin-2-yl]-7,11-diazatricyclo[7.3.1.02,7]tridecan-6-one
2-[1-(2,3-dimethylphenyl)piperidin-4-yl]-2,7-diazaspiro[4.5]decan-6-one
(2S,4R)-1-(2,3-dihydro-1H-inden-2-yl)-N-(1,1-dioxo-1λ6-thiolan-3-yl)-4-[(4-methoxyphenyl)sulfanyl]pyrrolidine-2-carboxamide
2-methyl-3-{[4-(1,2,4-oxadiazol-3-yl)piperidin-1-yl]methyl}quinoxaline
2-(adamantan-1-yl)-1-[4-(1-methoxypropan-2-yl)piperidin-1-yl]ethan-1-one
3-[(3R,4S)-1-(2-ethylbenzoyl)-4-(4-methylpiperazin-1-yl)piperidin-3-yl]propan-1-ol
N-[(2-methyl-1H-1,3-benzodiazol-6-yl)methyl]-2-(methylsulfanyl)-1,3-thiazole-4-carboxamide
6-(4-methoxyphenyl)-N,7-dimethyl-8-oxo-N-(propan-2-yl)-7H,8H-imidazo[1,2-a]pyrazine-2-carboxamide
1-(propan-2-yl)-4-{trimethyl-1H-pyrazolo[3,4-d]pyrimidin-4-yl}-1,4-diazepane
1-(3-ethyl-1,2-oxazole-5-carbonyl)-3-[4-(4-methylphenyl)-1H-pyrazol-5-yl]piperidine
(2S,4S)-4-amino-1-[3-(2-methoxyphenyl)benzoyl]-N-methylpyrrolidine-2-carboxamide
5-(4-oxo-4,5,6,7-tetrahydro-1-benzofuran-3-carbonyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-2-carboxylic acid
N-[2-(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)ethyl]-5,6-dimethyl-2-oxo-1,2-dihydropyridine-3-carboxamide
4-[(3-{1-benzyl-3-methyl-1H,4H-pyrazolo[3,4-d]imidazol-5-yl}phenyl)methyl]morpholine
N-[(7S,8aS)-2-methyl-octahydropyrrolo[1,2-a]piperazin-7-yl]-3-[(5-methyl-1,3,4-thiadiazol-2-yl)sulfanyl]propanamide
4-(1H-imidazol-1-yl)-1-(2-methyl-1,3-thiazole-4-carbonyl)piperidine-4-carboxylic acid
2-{[(6-chloropyridin-3-yl)methyl][(2-methylphenyl)methyl]amino}ethan-1-ol
8-(1-ethyl-5-methyl-1H-pyrazole-4-carbonyl)-3-hexyl-1-oxa-3,8-diazaspiro[4.5]decan-2-one
N-[2-(3,5-dimethyl-1H-pyrazol-4-yl)ethyl]-2-[3-methyl-5-oxo-4-(2-phenylethyl)-4,5-dihydro-1H-1,2,4-triazol-1-yl]acetamide
(2S,4S)-4-(2,5-dimethylbenzamido)-N-ethyl-1-(1H-imidazol-4-ylmethyl)pyrrolidine-2-carboxamide
2-{1-[(6-ethoxyquinolin-2-yl)methyl]-3-oxopiperazin-2-yl}-N-methylacetamide
[(4aS,8aR)-6-[2-(4-fluorophenyl)benzoyl]-decahydro-1,6-naphthyridin-4a-yl]methanol
N-[(1-ethyl-1H-imidazol-2-yl)methyl]-N-methyl-2-(2,4,7-trimethyl-1H-indol-3-yl)acetamide
N-[(1-methylpiperidin-3-yl)methyl]-2-[(pyridin-2-ylmethyl)amino]benzamide
(1R,5S)-N-[3-methoxy-5-(1H-1,2,3,4-tetrazol-1-yl)phenyl]-3,6-diazabicyclo[3.2.2]nonane-6-carboxamide
dimethyl[2-(1-{[2-(pyridin-2-yl)pyrimidin-5-yl]methyl}piperidin-2-yl)ethyl]amine
5-benzyl-4-(1-methyl-1H-pyrazole-5-carbonyl)-1-(4-methylphenyl)piperazin-2-one
1-[2-(methylamino)pyridine-3-carbonyl]-4-phenoxypiperidine-4-carboxylic acid
7-methoxy-N-{[5-(2-methylpropyl)-1,2-oxazol-3-yl]methyl}-1,2,3,4-tetrahydronaphthalen-2-amine
N-cyclohexyl-3-(4-methyl-4H-1,2,4-triazol-3-yl)-N-(pyridin-2-ylmethyl)propanamide
2-[4-({5-[(3-fluorophenyl)methyl]-6-oxo-2H,5H,6H-[1,3]dioxolo[4,5-g]quinolin-7-yl}methyl)piperazin-1-yl]-N-(propan-2-yl)acetamide
4-(5-cyano-1H-1,3-benzodiazol-2-yl)benzoic acid
(3S,4S)-4-(naphthalen-2-yl)-1-(1H-pyrrole-2-carbonyl)piperidin-3-ol
1-({2-[(propan-2-yl)amino]pyrimidin-5-yl}methyl)-4-(1H-pyrazol-1-yl)piperidine-4-carboxylic acid
5-({3-[2-(4-methoxy-3-methylphenyl)pyridin-4-yl]pyrrolidin-1-yl}methyl)pyrimidin-2-amine
1-{2-[3-(oxolan-3-yl)-1,2,4-oxadiazol-5-yl]ethyl}piperidine-4-carboxamide
N-{[2-(dimethylamino)-1,3-thiazol-4-yl]methyl}-4-(piperidin-1-ylmethyl)benzamide