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(4S,4aS,8aS)-1-[(1-methyl-1H-imidazol-4-yl)sulfonyl]-4-phenyl-decahydroquinolin-4-ol
2,6-dimethyl-4-{3-[(methylsulfanyl)methyl]piperidine-1-carbonyl}quinoline
2-hydroxy-3-(2-methylphenoxy)-N-[(1-phenyl-1H-1,2,3,4-tetrazol-5-yl)methyl]propanamide
9-[2-(2-methoxyethoxy)acetyl]-2-[(5-methylpyrazin-2-yl)methyl]-2,9-diazaspiro[5.5]undecan-3-one
1-[(1S,5R)-3-benzoyl-3,6-diazabicyclo[3.2.2]nonan-6-yl]-3-phenoxypropan-1-one
3-(3-{5-[2-(3,5-dimethyl-1H-pyrazol-1-yl)ethyl]-4-phenyl-1H-imidazol-1-yl}propyl)pyridine
2-{[2-(propylsulfanyl)pyrimidin-5-yl]methyl}-2,8-diazaspiro[4.5]decane
8-(4-chlorobenzoyl)-3-phenyl-1,8-diazaspiro[4.5]decan-2-one
N-[1-(2,3-dimethylphenyl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]but-2-ynamide
[(3,4-difluorophenyl)methyl]({1-[1-(3-fluorophenyl)-5-methyl-1H-pyrazol-4-yl]ethyl})amine
N-[1-(2,3-dimethylphenyl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]-4-(1H-1,2,3,4-tetrazol-1-yl)butanamide
N-(2,6-dimethylphenyl)-2-{2-[methyl(pyridin-2-ylmethyl)amino]acetamido}benzamide
5-[4-(piperidine-1-sulfonyl)-1,4-diazepane-1-carbonyl]pyridin-2-amine
3-{[(1S,5R)-6-(3-methylbut-2-en-1-yl)-7-oxo-3,6-diazabicyclo[3.2.2]nonan-3-yl]methyl}benzonitrile
N-[1-(naphthalen-2-ylmethyl)azepan-3-yl]-6-oxo-1,4,5,6-tetrahydropyridazine-3-carboxamide
1-[5-(2-phenylethyl)-1,3,4-thiadiazol-2-yl]-3-[1-(1H-1,2,3,4-tetrazol-5-yl)ethyl]urea
2-cyclopropyl-8-[(2,3-dichlorophenyl)methyl]-2,8-diazaspiro[5.5]undecan-3-one
2-hydroxy-5-({3-methyl-2-oxo-1-oxa-3,7-diazaspiro[4.5]decan-7-yl}methyl)benzoic acid
1-methyl-3-(naphthalen-2-ylmethyl)-8-(pyridin-4-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
5,6-dimethyl-2-(4-{[4-(pyridin-3-yl)piperazin-1-yl]methyl}phenyl)-3,4-dihydropyrimidin-4-one
N,N-dimethyl-7-(2-phenoxyethanesulfonyl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-amine
methyl 2-({2-[(4-chlorophenyl)methyl]-3-oxo-2,8-diazaspiro[4.5]decane-8-carbonyl}amino)acetate
2-(2-cyclopropyl-1H-1,3-benzodiazol-1-yl)-N-[2-(pyrrolidine-1-sulfonyl)ethyl]acetamide
2-{1-[(6-methylpyridin-2-yl)methyl]-4-{[3-(methylsulfanyl)phenyl]methyl}piperazin-2-yl}ethan-1-ol
(1,4-dioxan-2-ylmethyl)[(2-methoxynaphthalen-1-yl)methyl]methylamine
2-(2-chloro-4-{[(1S,5R)-6-(cyclobutylmethyl)-3,6-diazabicyclo[3.2.2]nonan-3-yl]methyl}phenoxy)acetamide
9-[2-(4-chlorophenyl)-2-hydroxyacetyl]-2-methyl-2,9-diazaspiro[5.5]undecan-3-one
(2S,4R)-1-benzyl-4-{[(4-methoxy-2,5-dimethylphenyl)methyl]amino}-N-methylpyrrolidine-2-carboxamide
4-[5-(5-methoxyfuran-2-carbonyl)-1-(3-methylbutyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carbonyl]morpholine
methyl 3-[(cyclohexylformamido)methyl]-5-(2,3-dihydro-1,4-benzodioxine-6-sulfonamido)benzoate
N-[(3S,4R)-1-(3-cyano-2-methoxypyridin-4-yl)-4-(5-methylfuran-2-yl)pyrrolidin-3-yl]acetamide
N-(4-cyano-2-ethylphenyl)-4-(furan-2-carbonyl)-1,4-diazepane-1-carboxamide
[3-(3,5-dimethyl-1H-pyrazol-4-yl)propyl](methyl)[2-methyl-2-(morpholin-4-yl)propyl]amine
2-(3-phenylpiperidin-1-yl)-1-[3-(pyridin-2-yl)azetidin-1-yl]ethan-1-one
N-[1-(1-methyl-1H-pyrazol-5-yl)propyl]-1-(9H-purin-6-yl)piperidin-4-amine
N-[(4-fluorophenyl)methyl]-4-[4-(piperazin-1-ylmethyl)-1H-1,2,3-triazol-1-yl]piperidine-1-carboxamide
7-[(3-methoxyphenyl)methyl]-2-(pyrazine-2-carbonyl)-2,7-diazaspiro[4.5]decane
5-{[(2-methylphenyl)methyl](oxolan-2-ylmethyl)carbamoyl}-1H-imidazole-4-carboxylic acid
9-[(2S)-2-hydroxypropanoyl]-2-[2-(1H-imidazol-4-yl)ethyl]-2,9-diazaspiro[5.5]undecan-3-one
N-[4-(2-methoxyphenyl)-1H-pyrrolo[2,3-b]pyridin-6-yl]piperidin-4-amine
{3-[(3-chloropyridin-4-yl)methyl]-9-(3-methylbutyl)-3,9-diazaspiro[5.5]undecan-1-yl}methanol
5-{[(5-cyclopropyl-1,3,4-oxadiazol-2-yl)amino]methyl}-1,3-dimethyl-2,3-dihydro-1H-1,3-benzodiazol-2-one
N-(2,4-difluorophenyl)-3-{[2-(2-hydroxyethyl)-3-oxopiperazin-1-yl]methyl}benzamide
N-{1H,4H,5H,6H,7H,8H-cyclohepta[c]pyrazol-3-ylmethyl}-N-methyl-3-(1-methyl-1H-pyrrol-2-yl)-1H-pyrazole-5-carboxamide
methyl 1-[(3R,5S)-1-[(4-methoxy-2,3-dimethylphenyl)methyl]-5-(4-phenylpiperazine-1-carbonyl)pyrrolidin-3-yl]-1H-1,2,3-triazole-4-carboxylate
5-[2-(methylsulfanyl)phenoxymethyl]-N-[(1R,2S)-2-phenylcyclopropyl]-1,2-oxazole-3-carboxamide
N-{1-[1-(2,3-dihydroxypropyl)piperidin-4-yl]-1H-pyrazol-5-yl}-2,2-dimethylpropanamide
N-[1-(dimethylamino)propan-2-yl]-2-[3-methyl-5-oxo-4-(2-phenylethyl)-4,5-dihydro-1H-1,2,4-triazol-1-yl]acetamide
N-[(4-methyl-1,2,3-thiadiazol-5-yl)methyl]-2-(pyrrolidin-1-yl)benzamide
(3S,5R)-1-(2-amino-6-methylpyrimidin-4-yl)-5-[(pyridin-4-ylmethyl)carbamoyl]piperidine-3-carboxylic acid