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N-{1-[2-(dimethylamino)-2,3-dihydro-1H-indene-2-carbonyl]piperidin-4-yl}acetamide
3-ethyl-N-[2-(2-ethylphenoxy)ethyl]-N,4-dimethyl-1H-pyrazole-5-carboxamide
2-{1-[(2-ethoxyphenyl)methyl]-3-oxopiperazin-2-yl}-N-[(4-methyl-1H-imidazol-2-yl)methyl]acetamide
5-[1-(2,3-dihydro-1H-inden-4-yl)-3-(thiophen-2-ylmethyl)-1H-1,2,4-triazol-5-yl]piperidin-2-one
4-[3-cyclopropyl-5-(1,2,3-thiadiazol-4-yl)-1H-1,2,4-triazol-1-yl]-2-methylpyridine
2-(2-phenyl-1H-imidazol-1-yl)-1-[2-(1H-pyrazol-1-ylmethyl)-1,4-oxazepan-4-yl]ethan-1-one
1-[4-(3-methylphenoxy)piperidin-1-yl]-2-(morpholin-4-yl)-2-(pyridin-3-yl)ethan-1-one
ethyl 3-[(2-{4-[(dimethylamino)methyl]phenyl}piperidine-1-carbonyl)amino]propanoate
1-methyl-1'-(5-propyl-1,3,4-oxadiazol-2-yl)-1,2-dihydrospiro[indole-3,4'-piperidine]-2-one
4-({2,4-dimethyl-5H,6H-furo[2,3-d]pyrimidin-6-yl}methyl)-3-methylpyridine
3-(4-methyl-1,3-thiazol-5-yl)-N-({1-[(2-methyl-1H-imidazol-1-yl)methyl]cyclopropyl}methyl)propanamide
1-{5-[5-(furan-2-yl)-1,2,4-oxadiazol-3-yl]-6-methyl-1,2,3,4-tetrahydro-2,7-naphthyridin-2-yl}-2-(methylsulfanyl)ethan-1-one
ethyl 1-[(2,3-dimethoxyphenyl)methyl]-4-[(3-methoxyphenyl)methyl]piperidine-4-carboxylate
N-methyl-N-{[3-(methylsulfanyl)phenyl]methyl}-2-{2-oxo-1-oxa-3,8-diazaspiro[4.5]decan-3-yl}acetamide
propan-2-yl (4aR,7aS)-4-[(4-ethylphenyl)methyl]-6,6-dioxo-octahydro-6λ6-thieno[3,4-b]piperazine-1-carboxylate
8-{[4-(1H-pyrazol-1-ylmethyl)phenyl]methyl}-1-oxa-8-azaspiro[4.5]decan-3-ol
N-[(3R,4S)-1-(2-ethoxyethyl)-4-phenylpyrrolidin-3-yl]-4,4,4-trifluorobutanamide
3-[ethyl(pyridin-4-ylmethyl)amino]-N-[3-(trifluoromethyl)phenyl]piperidine-1-carboxamide
1,3-dimethyl-N-{[1-(propan-2-yl)-1H-pyrazol-4-yl]methyl}-1H-pyrazolo[3,4-d][1,3]thiazol-5-amine
(2R,6R)-4-[2-(2,5-dimethylphenyl)acetyl]-8-oxa-4-azatricyclo[7.4.0.02,6]trideca-1(13),9,11-triene-6-carboxylic acid
N-[(4-ethyl-4H-1,2,4-triazol-3-yl)methyl]-N-methyl-5-[3-(phenoxymethyl)-1,2,4-oxadiazol-5-yl]pyridin-2-amine
1-({2-[3-(propan-2-yl)-[1,2,4]triazolo[3,4-b][1,3,4]thiadiazol-6-yl]thiophen-3-yl}sulfonyl)pyrrolidine
7-methyl-4-(1-methylpiperidin-4-yl)-2-(thiophen-3-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepine
2-ethyl-N-{[4-methyl-6-(trifluoromethyl)pyrimidin-2-yl]methyl}pyrimidine-5-carboxamide
N-[2-(1,3-benzothiazol-2-yl)ethyl]-1-[(1s,4s)-4-aminocyclohexyl]-1H-1,2,3-triazole-4-carboxamide
ethyl 1-(1-methyl-2-oxo-1,2-dihydroquinolin-4-yl)-5-{[(1,2,3,4-tetrahydronaphthalen-1-yl)amino]methyl}-1H-pyrazole-4-carboxylate
2-[6-hydroxy-4-(5-methyl-1,2,4-oxadiazol-3-yl)-1,4-diazepan-1-yl]-N-(pyridin-2-ylmethyl)acetamide
2-{1-[(2-ethoxyphenyl)methyl]-4-(pyridin-4-ylmethyl)piperazin-2-yl}ethan-1-ol
5-(2-fluorophenyl)-3-[2-(2-methoxyphenyl)pyrrolidin-1-yl]-1,2,4-triazine
{3-[(4-fluorophenyl)methyl]-1-(6-methylpyridine-2-carbonyl)piperidin-3-yl}methanol
7-methyl-6-oxo-N-[4-(1,3-thiazol-4-yl)phenyl]-2,7-diazaspiro[4.5]decane-2-carboxamide
4-(1-methyl-2-oxopyrrolidin-3-yl)-8-thia-4,6-diazatricyclo[7.5.0.02,7]tetradeca-1(9),2(7),5-trien-3-one
N-{3-[2-(4-methanesulfonylphenyl)-1H-imidazol-1-yl]phenyl}acetamide
N-({6-ethyl-2-methoxy-5-oxo-5H,6H,7H-pyrrolo[3,4-b]pyridin-3-yl}methyl)-2-(2H-1,2,3,4-tetrazol-2-yl)acetamide
4-methyl-N-[3-(1H-1,2,4-triazol-1-ylmethyl)phenyl]-1,2,3,6-tetrahydropyridine-1-carboxamide
N-cyclopentyl-4,6-dimethyl-N-({1-[2-(2-methylphenyl)ethyl]piperidin-4-yl}methyl)-2-oxo-1,2-dihydropyridine-3-carboxamide
(2R,3R,6R)-3-(2,3-difluorophenyl)-5-(1-ethyl-1H-pyrazole-3-carbonyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
N-({6-ethyl-2-methoxy-5-oxo-5H,6H,7H-pyrrolo[3,4-b]pyridin-3-yl}methyl)-2,3-dihydro-1-benzofuran-7-carboxamide
N-(3-chloro-4-methoxyphenyl)-3-[1-(3-phenoxypropanoyl)piperidin-3-yl]propanamide
2-{3-[1-(pyridin-2-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}pyridine-4-carboxamide
3-[4-methyl-5-(piperidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]-1-[(4-methylphenyl)methyl]piperidine
2-(2-methyl-1H-imidazol-1-yl)-1-{4-[4-(2-methylphenyl)-1H-pyrazol-5-yl]piperidin-1-yl}propan-1-one
1-(furan-2-carbonyl)-4-{[2-(4-methoxy-2,5-dimethylphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-1,4-diazepane
2-ethyl-N-[2-(2-oxo-1,3-oxazinan-3-yl)ethyl]pyrimidine-5-carboxamide
2-amino-6-{4-[(3-chloro-2-fluorophenyl)methyl]piperazin-1-yl}-3,4-dihydropyrimidin-4-one
1-[3-(6-hydroxy-2-methylpyrimidin-4-yl)piperidin-1-yl]-2-(1,2,3,4-tetrahydroisoquinolin-2-yl)ethan-1-one
N-phenyl-5-(1H-1,2,4-triazole-5-carbonyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carboxamide
2-(3-methoxy-2-oxo-1,2-dihydropyridin-1-yl)-N-methyl-N-{[1-(2-methylphenyl)-1H-pyrazol-4-yl]methyl}acetamide
2,2-dimethyl-N-(1-{1-[3-(5-methylfuran-2-yl)butyl]piperidin-4-yl}-1H-pyrazol-5-yl)propanamide
N-[3-(4-fluorophenyl)phenyl]-1-(2-methylfuran-3-carbonyl)piperidine-3-carboxamide