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N-[3-(3,5-dimethyl-1H-pyrazol-1-yl)propyl]-N,1,6-trimethyl-1H-pyrazolo[3,4-d]pyrimidin-4-amine
N4,N4-dimethyl-N6-[3-(4-methyl-1,3-thiazol-2-yl)propyl]pyrimidine-4,6-diamine
methyl(1,2-oxazol-5-ylmethyl){[1-(2-phenylethyl)-2-(propane-2-sulfonyl)-1H-imidazol-5-yl]methyl}amine
1-ethyl-4-({2-oxo-3-phenyl-1,8-diazaspiro[4.5]decan-8-yl}methyl)-1H-pyrrole-2-carbonitrile
4-[(4-hydroxy-5-methoxypyridin-2-yl)methyl]-7-(4-methylphenyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
(1s,4s)-N-[(4-fluorophenyl)(pyridin-4-yl)methyl]-4-hydroxycyclohexane-1-carboxamide
3-[4-(3,4-difluorophenyl)-1H-pyrazol-5-yl]-1-[(2-ethoxyphenyl)methyl]piperidine
2-{[methyl(4,5,6,7-tetrahydro-1H-indazol-3-ylmethyl)amino]methyl}pyridine-3-carboxylic acid
2,6-dioxo-N-[3-(trimethyl-1H-pyrazol-1-yl)propyl]-1,2,3,6-tetrahydropyrimidine-4-carboxamide
N-{[2-(2-methyl-5-phenylfuran-3-yl)-6-oxo-1,6-dihydropyrimidin-4-yl]methyl}acetamide
N-(1-cycloheptylpiperidin-3-yl)-1-ethyl-3-methyl-1H-pyrazole-5-carboxamide
2-amino-4-[5-(hydroxymethyl)furan-2-yl]-6-(3-methylphenyl)-5,6,7,8-tetrahydro-1,6-naphthyridine-3-carbonitrile
N-(2H-1,3-benzodioxol-5-ylmethyl)-1-methyl-6-oxo-N-(pentan-3-yl)-1,6-dihydropyridine-3-carboxamide
3-fluoro-7-methyl-N-[2,2,2-trifluoro-1-(pyridin-2-yl)ethyl]imidazo[1,2-a]pyridine-2-carboxamide
4,4-difluoro-N-[3-(1H-1,2,4-triazol-1-yl)phenyl]piperidine-1-carboxamide
{[2-(4-cyclohexylpiperazine-1-carbonyl)imidazo[1,2-a]pyridin-3-yl]methyl}(dicyclopropylmethyl)methylamine
N-[4-(furan-2-yl)phenyl]-4-[(1S,2S)-2-hydroxycyclohexyl]piperazine-1-carboxamide
N-methyl-3-(1-methylpiperidin-2-yl)-N-[(2E)-3-phenylprop-2-en-1-yl]propanamide
N-methyl-2-[1-(naphthalen-2-ylmethyl)-3-oxopiperazin-2-yl]-N-(1,2-oxazol-5-ylmethyl)acetamide
6-[({[2-(1H-1,2,4-triazol-1-yl)pyridin-3-yl]methyl}amino)methyl]-1,4-oxazepan-6-ol
1-(cyclohexylmethyl)-N,N-dimethyl-5-{[(2-methylphenyl)methyl]amino}-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
N-({1-[2-(4-methoxyphenyl)ethyl]piperidin-3-yl}methyl)-N,5-dimethylpyrazine-2-carboxamide
(1S,5R)-6-(3-methylbut-2-en-1-yl)-3-[3-(trifluoromethyl)benzoyl]-3,6-diazabicyclo[3.2.2]nonan-7-one
N-[2-(dimethylamino)ethyl]-4-(6-methoxypyridin-2-yl)-1H-pyrrolo[2,3-b]pyridin-6-amine
N-(2,1,3-benzothiadiazol-5-ylmethyl)-1-methyl-6-(propan-2-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-amine
N-[(4-methanesulfonylmorpholin-2-yl)methyl]-1,3-dimethyl-1H-pyrazolo[3,4-d][1,3]thiazol-5-amine
4-[6-(3-chlorophenyl)imidazo[2,1-b][1,3]thiazole-3-carbonyl]-1,2-dimethylpiperazine
N-(3-{4-[(2R,6S)-2,6-dimethylmorpholin-4-yl]piperidin-1-yl}phenyl)-3-(trifluoromethyl)benzamide
6-[(1R,5R)-6-benzyl-3,6-diazabicyclo[3.2.2]nonan-3-yl]-N-ethyl-N-methylpyridine-3-carboxamide
6-(4-chlorophenyl)-N-methyl-N-(pyrazin-2-ylmethyl)imidazo[2,1-b][1,3]thiazole-3-carboxamide
6-({methyl[(2-phenyl-1,3-thiazol-4-yl)methyl]amino}methyl)-1,4-oxazepan-6-ol
2-(5-amino-1H-1,2,3,4-tetrazol-1-yl)-N-[(8-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]acetamide
2-(5-{[(2R,6S)-6-phenyl-2-(prop-2-en-1-yl)-1,2,3,6-tetrahydropyridin-1-yl]methyl}-1,2,4-oxadiazol-3-yl)pyrazine
2-[1-(cyclohexylmethyl)-3-oxopiperazin-2-yl]-N-{[1-(2-hydroxyethyl)piperidin-4-yl]methyl}acetamide
2-{4-[2-(trifluoromethyl)pyrimidin-4-yl]morpholin-2-yl}ethan-1-amine
N-[1-(4-ethoxy-3-fluorophenyl)ethyl]-3-(pyridin-2-yl)-1H-pyrazole-5-carboxamide
2-cyclopropyl-4-phenyl-9-(pyrimidin-2-ylmethyl)-2,9-diazaspiro[5.5]undecan-3-one
1-(1-phenylcyclohexanecarbonyl)-3-(4H-1,2,4-triazol-3-yl)piperidine
4-{[2-(4-methoxynaphthalen-1-yl)-1H-imidazol-1-yl]methyl}-3,5-dimethyl-1,2-oxazole
[(3S,5R)-1-(3,4-difluorobenzoyl)-5-(morpholin-4-ylmethyl)piperidin-3-yl]methanol
5-[4-(1,2,3,4-tetrahydronaphthalen-2-yl)piperazine-1-carbonyl]quinoxaline
1-[3-(hydroxymethyl)-3-(2-methoxyethyl)piperidin-1-yl]-2-[3-(trifluoromethyl)phenyl]ethan-1-one
6-methoxy-1-[5-(2-methoxyacetyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-yl]hexan-1-one
2-{1-tert-butyl-3-[(2-methoxyphenyl)methyl]-1H-1,2,4-triazol-5-yl}-6-methyl-4H-pyran-4-one
N-methyl-2-oxo-6-phenyl-N-[1-(1,3-thiazol-2-yl)ethyl]-1,2-dihydropyridine-3-carboxamide
3-(4-fluorophenoxymethyl)-1-(5-methyl-1,3-oxazole-4-carbonyl)piperidine
1-{5-methanesulfonyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-yl}-2-(methylamino)ethan-1-one
3-(3-{2-[2-(trifluoromethyl)phenyl]ethyl}piperidine-1-carbonyl)-1H-pyrazol-5-amine
N-(3-carbamoyl-4-fluorophenyl)-4-cyclobutanecarbonyl-1,4-diazepane-1-carboxamide
4-[1-(pentan-2-yl)-1H,4H-pyrazolo[3,4-d]imidazol-5-yl]-2,1,3-benzoxadiazole