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3-[(3R,4S)-1-(1-tert-butyl-1H-pyrrole-3-carbonyl)-4-(morpholin-4-yl)piperidin-3-yl]propanoic acid
3-(5-oxo-1-{[2-(trifluoromethyl)phenyl]methyl}pyrrolidin-3-yl)-1-(thiophen-2-yl)urea
1-cyclopropanecarbonyl-N-[3-(3,5-dimethyl-1H-pyrazol-4-yl)propyl]piperidine-4-carboxamide
N-(5-fluoro-2-methoxyphenyl)-4-(2-methoxyethyl)piperazine-1-carboxamide
(5S,9aS,9bS)-5-(2-butyl-1H-imidazol-4-yl)-2-[(2-methoxyphenyl)methyl]-octahydro-1H-pyrrolo[3,4-h]pyrrolizin-1-one
4-(3,4-dimethoxyphenyl)-3-[(trimethyl-1H-pyrazol-1-yl)methyl]-4,5-dihydro-1H-1,2,4-triazol-5-one
N-(2,1,3-benzoxadiazol-5-ylmethyl)-5-[(4-hydroxypiperidin-1-yl)methyl]-N-methyl-1,2-oxazole-3-carboxamide
N-[(3R,4S)-1-acetyl-4-cyclopropylpyrrolidin-3-yl]-2-(morpholin-4-yl)benzamide
1-({3-methylimidazo[1,5-a]pyridin-1-yl}methyl)-4-(thiophen-2-ylmethyl)-1,4-diazepane
1-{1-[3-(2-methylphenyl)phenyl]piperidin-4-yl}-1,4-diazepane
2-[(3,5-difluorophenyl)methyl]-8-[(2S)-2-hydroxypropanoyl]-2,8-diazaspiro[4.5]decan-3-one
6-(4-ethylphenyl)-N-methyl-N-(oxolan-3-yl)imidazo[2,1-b][1,3]thiazole-3-carboxamide
1-(3-methylbutyl)-3-[3-(pyridin-4-yl)propyl]-8-(thian-4-yl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
2-{4-methyl-6-[4-(1H-1,2,3-triazole-5-carbonyl)piperazin-1-yl]pyrimidin-2-yl}phenol
1-[2-(cyclohex-1-en-1-yl)acetyl]-N-[4-(3-methylphenyl)phenyl]piperidine-4-carboxamide
1-ethyl-8-{[2-(morpholin-4-yl)pyrimidin-5-yl]methyl}-1,3,8-triazaspiro[4.5]decane-2,4-dione
(4aS,8aS)-2-{[3-fluoro-5-(trifluoromethyl)phenyl]methyl}-decahydro-2,7-naphthyridin-4a-ol
3-{5-[1-(2-ethoxyethyl)-3-methyl-1H-pyrazol-5-yl]-1,2,4-oxadiazol-3-yl}-6-methylpyridazine
7-(2-aminopyridine-4-carbonyl)-2-(pyridin-2-yl)-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
ethyl 3-benzyl-1-[(2,4-difluorophenyl)carbamoyl]piperidine-3-carboxylate
6-[2-(2H-1,3-benzodioxol-5-yl)acetyl]-N-[(4-phenyloxan-4-yl)methyl]-6-azaspiro[2.5]octane-1-carboxamide
(2S,4R)-N-{2-azatricyclo[9.4.0.03,8]pentadeca-1(11),3,5,7,12,14-hexaen-5-yl}-4-[(4-fluorophenyl)sulfanyl]-1-(pyridin-4-ylmethyl)pyrrolidine-2-carboxamide
3-[1-(2-methoxyethyl)-1H-imidazol-2-yl]-1-{7-methylthieno[3,2-d]pyrimidin-4-yl}piperidine
N-[(5-cyclobutyl-1,2,4-oxadiazol-3-yl)methyl]-N-methyl-5-oxo-1-(pyridin-2-ylmethyl)pyrrolidine-3-carboxamide
(2S,4R)-N-[2-(3-fluorophenyl)ethyl]-4-[(4-fluorophenyl)sulfanyl]-1-[(3-hydroxyphenyl)methyl]pyrrolidine-2-carboxamide
N-[2-(7-{[4-(propan-2-yl)phenyl]methyl}-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl)ethyl]cyclobutanecarboxamide
1-[2-methoxy-4-({[(5-methylthiophen-2-yl)methyl]amino}methyl)phenoxy]-3-[methyl(propan-2-yl)amino]propan-2-ol
4-(1-benzyl-5-{[4-(pyrrolidin-1-yl)phenyl]methyl}-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carbonyl)piperazin-2-one
5-[4-(3-phenylpropyl)-1,4-diazepane-1-carbonyl]-1,2-dihydropyridin-2-one
2-(2-methoxyethyl)-5-{[4-(2-methoxyphenyl)-3,3-dimethylpiperazin-1-yl]methyl}pyrimidine
N-{[1-(2-methoxyethyl)piperidin-3-yl]methyl}-2-methyl-5-phenylpyrazolo[1,5-a]pyrimidin-7-amine
4-[(1-methyl-1H-imidazol-2-yl)methyl]-N-[3-(2-methyl-2H-1,2,3,4-tetrazol-5-yl)phenyl]piperazine-1-carboxamide
ethyl 1-[(4-methoxyphenyl)methyl]-5-[(1-methyl-1H-1,3-benzodiazol-2-yl)methyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylate
methyl({[1-(2-methylpropyl)-2-phenylmethanesulfonyl-1H-imidazol-5-yl]methyl})(thiophen-3-ylmethyl)amine
8-[2-(4-hydroxyphenyl)acetyl]-2-(2-methoxyethyl)-2,8-diazaspiro[5.5]undecan-3-one
4-{8-chloro-1H,2H,3H,4H,5H-pyrido[4,3-b]indole-2-carbonyl}-2-(4H-1,2,4-triazol-4-yl)pyridine
1-methyl-4-[(3-phenylphenyl)methyl]-2,3,4,5-tetrahydro-1H-1,4-benzodiazepine-2,5-dione
1-(4-{dimethyl-1H-pyrazolo[3,4-d][1,3]thiazol-5-yl}piperazin-1-yl)-3-methylbutan-1-one
1-(4-{[2-(4-chlorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}piperazin-1-yl)ethan-1-one
1-[(2R,3R)-3-amino-2-hydroxy-2,3-dihydrospiro[indene-1,4'-piperidine]-1'-yl]-3-(1H-1,2,3,4-tetrazol-1-yl)propan-1-one
methyl[(1-phenyl-1H-1,2,3-triazol-4-yl)methyl]{[4-(propan-2-yl)-4H-1,2,4-triazol-3-yl]methyl}amine
N,N-dimethyl-2-({5-[4-(2-phenylethyl)piperidine-1-carbonyl]pyridin-2-yl}amino)acetamide
3-[4-(2-amino-6-methylpyrimidin-4-yl)-6-hydroxy-1,4-diazepan-1-yl]propanoic acid
1-ethoxy-3-({5-methylpyrazolo[1,5-a]pyrimidin-7-yl}amino)propan-2-ol
2-amino-2-methyl-1-[3-(1-methyl-1H-imidazol-2-yl)piperidin-1-yl]propan-1-one
N3-cyclohexyl-N5-(1-methoxypropan-2-yl)-1-(2-methylpropyl)-4-oxo-1,4-dihydropyridine-3,5-dicarboxamide
N-[(1-cyclopentylpiperidin-3-yl)methyl]-3-(methylsulfanyl)-N-[2-(piperidin-1-yl)ethyl]propanamide
3-{2-[2-(4-fluorophenyl)pyrrolidin-1-yl]-2-oxoethyl}-3-phenyl-1-(pyridin-4-ylmethyl)pyrrolidine-2,5-dione
N-{2-[({5-[(dimethylamino)methyl]furan-2-yl}methyl)sulfanyl]ethyl}-5,6-dimethylpyridine-3-carboxamide
4-methoxy-N-methyl-3-{3-[1-(pyrrolidin-1-yl)ethyl]phenyl}benzamide