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[(2S)-1-[3-(2-phenylethyl)-1,2-oxazole-5-carbonyl]pyrrolidin-2-yl]methanol
3-(methoxymethyl)-1-[(5-propylfuran-2-yl)methyl]piperidine
4-[2-({4-benzyl-5-[1-(cyclohexylmethyl)piperidin-4-yl]-4H-1,2,4-triazol-3-yl}sulfanyl)ethyl]morpholine
1-cyclopentyl-N-(3-methylbutyl)-4-oxo-5-[4-(piperidin-1-yl)piperidine-1-carbonyl]-1,4-dihydropyridine-3-carboxamide
(4aS,8aR)-6-[2-(2-ethyl-1H-imidazol-1-yl)acetyl]-1-(3-methoxypropyl)-decahydro-1,6-naphthyridin-2-one
8-[4-methoxy-3-(morpholin-4-yl)benzoyl]-2,8-diazaspiro[4.5]decan-3-one
N-[(3S,5S)-5-(ethylcarbamoyl)-1-(thiophen-2-ylmethyl)pyrrolidin-3-yl]-1-methyl-1H-pyrazole-5-carboxamide
2-(dimethyl-1,2-oxazol-4-yl)-1-[7-(5-methylthiophen-2-yl)-9-(oxan-2-ylmethoxy)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]ethan-1-one
2-[(E)-2-{4-[2-(oxan-2-yl)-1H-imidazol-1-yl]phenyl}ethenyl]pyridine
4-[4-(4-ethoxyphenyl)-1H-imidazol-2-yl]pyridine
4-[(2H-1,3-benzodioxol-5-ylmethyl)amino]-5-methyl-N-(2-methylpropyl)thieno[2,3-d]pyrimidine-6-carboxamide
1-(2-{4-[(4-methyl-1H-pyrazol-1-yl)methyl]piperidin-1-yl}-2-oxoethyl)piperidin-2-one
4-{1-benzyl-5-[(4-hydroxyphenyl)methyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carbonyl}piperazin-2-one
8-(3-fluoro-4-methylbenzoyl)-2-methyl-2,8-diazaspiro[4.5]decane-3-carboxylic acid
methyl 3-[1-(1-ethylpiperidin-3-yl)piperidin-4-yl]propanoate
1-methyl-3-propyl-N-{[3-(pyrrolidin-1-ylmethyl)phenyl]methyl}-1H-pyrazole-5-carboxamide
5-(cycloheptylamino)-1-methyl-N-(thiophen-2-ylmethyl)-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
{[3-(3,4-dimethylphenyl)-1H-pyrazol-4-yl]methyl}[2-(3-fluorophenyl)ethyl]amine
(4aS,8aR)-6-{imidazo[1,2-a]pyridine-3-carbonyl}-1-[2-(methylamino)ethyl]-decahydro-1,6-naphthyridin-2-one
N-ethyl-3-[3-(2-methylphenyl)-1,2,4-oxadiazol-5-yl]-N-(pyridin-2-ylmethyl)propanamide
N-(2-methyl-1,3-benzothiazol-6-yl)-4-(thiophen-2-ylmethyl)-1,4-diazepane-1-carboxamide
N-methyl-2-[methyl(2-phenylethyl)amino]-2,3-dihydro-1H-indene-2-carboxamide
1-{[2-(2,5-difluorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-4-(pyrrolidine-1-carbonyl)piperidine
1-[1-(2-methoxyethyl)pyrrolidine-3-carbonyl]-4-[(2E)-3-phenylprop-2-en-1-yl]piperazine
3-[2-(6-methoxynaphthalen-2-yl)morpholin-4-yl]-N-(propan-2-yl)propanamide
1-(2-aminoethyl)-N-{[2-(3-methylphenyl)-1,3-thiazol-4-yl]methyl}-1H-1,2,3-triazole-4-carboxamide
4-cyano-N-(cyclobutylmethyl)-1-methyl-N-(oxolan-2-ylmethyl)-1H-pyrrole-2-carboxamide
(2R,6R)-11-methoxy-4-(pyrimidin-2-ylmethyl)-8-oxa-4-azatricyclo[7.4.0.02,6]trideca-1(13),9,11-triene-6-carboxylic acid
N-(3-chloro-4-fluorophenyl)-3-(1-{spiro[2.3]hexane-1-carbonyl}piperidin-4-yl)propanamide
N-{2-[(2-methylquinolin-8-yl)oxy]ethyl}thiolan-3-amine
N,N-dimethyl-7-(3-methyl-1H-pyrazole-5-carbonyl)-2-(pyridin-2-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-amine
2-(dimethylamino)-N-[2-(ethanesulfonyl)ethyl]-2-(2-fluorophenyl)acetamide
5-(2-fluorophenyl)-3-[4-(3-methoxypropyl)piperidin-1-yl]-1,2,4-triazine
2-methoxy-1-[7-(1,2,3,4-tetrahydroquinoline-1-sulfonyl)-1,2,3,4-tetrahydroisoquinolin-2-yl]ethan-1-one
3-(4,5-dimethyl-1H-pyrazol-3-yl)-1-{2-[3-(pyridin-2-yl)-1,2,4-oxadiazol-5-yl]pyrrolidin-1-yl}propan-1-one
ethyl 1-{[2-(2-chlorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-1H-pyrazole-4-carboxylate
2-amino-1-{3-[2-methyl-6-(pyrrolidin-1-yl)pyrimidin-4-yl]piperidin-1-yl}ethan-1-one
methyl (1R,3S,3aR,6aS)-1-ethyl-5-methyl-4,6-dioxo-3-(1-phenyl-1H-pyrazol-4-yl)-octahydropyrrolo[3,4-c]pyrrole-1-carboxylate
N-{[1-(4-fluorophenyl)-3,5-dimethyl-1H-pyrazol-4-yl]methyl}-6-methyl-4-oxo-4H-pyran-2-carboxamide
2-[(3-methoxyphenyl)methyl]-8-(morpholine-4-carbonyl)-2,8-diazaspiro[4.5]decan-3-one
N-(2-{2-[(methylsulfanyl)methyl]-1,3-thiazol-4-yl}ethyl)-3,4-dihydro-2H-1-benzopyran-3-carboxamide
3-(2H-1,3-benzodioxol-5-yl)-N-({5-fluoro-7-[2-(methylsulfanyl)pyrimidin-4-yl]-2,3-dihydro-1-benzofuran-2-yl}methyl)propanamide
2-[(8-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]-3-(pyrrolidine-1-carbonyl)pyridine
N-[1-(1H-imidazol-1-yl)-3,3-dimethylbutan-2-yl]-3-(pyridin-4-yl)propanamide
4-(1-methyl-4-{4-[(propan-2-yloxy)methyl]piperidin-1-yl}-1H-pyrazolo[3,4-d]pyrimidin-6-yl)pyridine
4-(1-benzyl-4-phenylpiperidine-4-carbonyl)thiomorpholine
N-methyl-6-oxo-4-[(1s,4s)-4-aminocyclohexyl]-1H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridine-3-carboxamide
N,N-diethyl-2-{1-[(2-fluorophenyl)methyl]-2-methyl-4-oxo-4,5,6,7-tetrahydro-1H-indol-3-yl}acetamide
N-cyclopentyl-N-ethyl-5-(2-methoxyphenoxymethyl)-1H-pyrazole-3-carboxamide
3-{[(2-methoxyethyl)[(3-methylthiophen-2-yl)methyl]amino]methyl}-N-methylpyridin-2-amine