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(1R,5R)-6-[3-(2,4-difluorophenyl)propanoyl]-N,N-dimethyl-3,6-diazabicyclo[3.2.2]nonane-3-carboxamide
3-(2-fluorophenyl)-3-{[1-(propan-2-yl)piperidin-4-yl]formamido}propanoic acid
3-(2-{4-[(1-methyl-1H-imidazol-2-yl)methyl]piperazin-1-yl}-2-oxoethyl)-3,4-dihydroquinazolin-4-one
1-butyl-3-(2-methyl-5-sulfamoylphenyl)-1-(pyridin-2-ylmethyl)urea
N,N-dimethyl-2-({2-[methyl(phenyl)amino]acetamido}methyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-5-carboxamide
1-[(3R,4R)-3-cyclopropyl-3-hydroxy-4-methylpyrrolidin-1-yl]-3-(pyrazin-2-yl)propan-1-one
1-{5,7-dimethylpyrido[2,3-d]pyrimidin-4-yl}-4-(5-methylpyridin-2-yl)piperidin-4-ol
3-(3-chloro-1H-1,2,4-triazol-5-yl)-N-{[2-(4-methylpiperazin-1-yl)pyridin-3-yl]methyl}propanamide
9-{3,6-dimethyl-[1,2]oxazolo[5,4-b]pyridine-4-carbonyl}-5-methoxy-1-oxa-9-azaspiro[5.5]undecane
2-(2-tert-butylpyrimidin-5-yl)-N-ethyl-N,7,8-trimethylquinoline-4-carboxamide
2-{3-methyl-5-[3-(2-oxopyrrolidin-1-yl)phenyl]-1H-1,2,4-triazol-1-yl}benzoic acid
3-{2-[(4-methoxyphenyl)methyl]-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-6-yl}-5-propyl-1,2,4-oxadiazole
1-(1-methyl-1H-pyrazole-5-carbonyl)-N-[3-(1H-pyrazol-1-yl)phenyl]pyrrolidine-2-carboxamide
1-(2-{imidazo[2,1-b][1,3]thiazol-6-yl}ethyl)-3-[5-(trifluoromethyl)-1,3,4-thiadiazol-2-yl]urea
(4S)-3-[(2-ethyl-1,3-thiazol-4-yl)methyl]-4-(propan-2-yl)-1,3-oxazolidin-2-one
(3R,5S)-N-[(2-methoxyphenyl)methyl]-5-{[(6-methylpyridin-3-yl)oxy]methyl}piperidine-3-carboxamide
1-[3-(2H-1,3-benzodioxol-5-ylmethyl)-3-methylpiperidin-1-yl]-2-(morpholin-4-yl)ethane-1,2-dione
3-(3-fluorophenyl)-4-(5-methoxy-4-oxo-1,4-dihydropyridine-2-carbonyl)piperazin-2-one
6-[4-(3-chlorophenyl)piperazin-1-yl]-2-methylpyrimidin-4-amine
N-benzyl-N-methyl-1-(prop-2-en-1-yl)-3-(thiomorpholine-4-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
1-methyl-4-[(1-{[2-(trifluoromethoxy)phenyl]methyl}piperidin-3-yl)methyl]piperazine
N-[(5-tert-butyl-1,3-benzoxazol-2-yl)methyl]pyridine-3-carboxamide
1-{[2-(difluoromethoxy)phenyl]methyl}-4-(3-methoxypropyl)piperidine
N-[(1-cyclopentylpiperidin-4-yl)methyl]-N-(oxolan-2-ylmethyl)-2-(2-oxopyrrolidin-1-yl)acetamide
[(3R,4R)-1-[(4-methoxy-3-methylphenyl)methyl]-4-(pyrrolidin-1-ylmethyl)pyrrolidin-3-yl]methanol
2-(oxolan-3-yl)-1-(2-phenoxyethyl)-1H-imidazole
4-(2-methyl-4-propanamidophenyl)benzamide
(2S)-N-(6-methoxy-2-oxo-2,3-dihydro-1H-1,3-benzodiazol-5-yl)-2-(methoxymethyl)pyrrolidine-1-carboxamide
6-(2-aminoethyl)-N-methyl-N-{[3-(1H-pyrazol-1-yl)phenyl]methyl}pyrimidin-4-amine
3-[1-(3-methylbutan-2-yl)-1H-pyrazol-5-yl]-1-[2-(pyridin-4-yl)ethyl]urea
N-[1-(1-methyl-1H-1,2,4-triazol-5-yl)propyl]-6-(2-methylphenyl)imidazo[2,1-b][1,3]thiazole-3-carboxamide
9-[3-(4,5-dimethyl-1H-pyrazol-3-yl)propanoyl]-2-(prop-2-en-1-yl)-2,9-diazaspiro[5.5]undecan-3-one
(3R,4R)-1-(1-benzyl-1H-pyrazole-4-carbonyl)-4-(hydroxymethyl)piperidin-3-ol
7-(2,3-dimethyl-1H-indole-5-carbonyl)-N,N-dimethyl-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-amine
(2S,4R)-4-amino-N-[(4-methyl-5,6,7,8-tetrahydroquinazolin-2-yl)methyl]pyrrolidine-2-carboxamide
N,N-dimethyl-3-[3-(trifluoromethyl)benzoyl]piperidine-1-sulfonamide
3-[3-methyl-1-(1-methyl-1H-1,2,4-triazol-5-yl)butyl]-1-[3-(1H-1,2,4-triazol-1-yl)phenyl]urea
1-[3-(4-phenylbenzoyl)piperidin-1-yl]-3-(1H-1,2,3,4-tetrazol-1-yl)propan-1-one
4-oxo-N-(propan-2-yl)-N-[(trimethyl-1H-pyrazol-4-yl)methyl]-4H-pyrido[1,2-a]pyrimidine-3-carboxamide
5-(propan-2-yl)-N-{1-[3-(pyridin-2-yl)-1,2,4-oxadiazol-5-yl]ethyl}-1,2-oxazole-3-carboxamide
benzyl(methyl)({3-[2-(4-methyl-1,2,5-oxadiazol-3-yl)pyrrolidine-1-carbonyl]-1,2-oxazol-5-yl}methyl)amine
5-(3-methyl-1,2,4-oxadiazol-5-yl)-N-[1-(pyridin-2-ylmethyl)piperidin-3-yl]pyridin-2-amine
1-(4-{1-[2-(6-methoxy-2H-1,3-benzodioxol-5-yl)-1H-imidazol-1-yl]ethyl}phenyl)-1H-1,2,4-triazole
N-[1-(3-methylbutanoyl)piperidin-4-yl]-5-phenyl-1H-pyrrole-2-carboxamide
methyl 2-(cyclopropylsulfamoyl)-6-[(4-phenylphenyl)methyl]-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
4-[(1E)-3-[3-(2-hydroxyethyl)-4-(propan-2-yl)piperazin-1-yl]prop-1-en-1-yl]-2-methoxyphenol
N-[(1S)-1,2,3,4-tetrahydronaphthalen-1-yl]-6-(4H-1,2,4-triazol-4-yl)pyridine-3-carboxamide
1-(4-chlorophenyl)-N-{[7-methoxy-2-(morpholin-4-yl)quinolin-3-yl]methyl}-N-[3-(2-oxopyrrolidin-1-yl)propyl]cyclobutane-1-carboxamide
4-(2,6-dimethylpyridin-3-yl)-N-[2-(3-methylpiperidin-1-yl)ethyl]pyrimidin-2-amine
N-[(1-hydroxycyclohexyl)methyl]-5-[1-(piperidin-1-yl)ethyl]furan-2-carboxamide