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6-{3-[1-(cyclobutylmethyl)-1H-imidazol-2-yl]piperidine-1-carbonyl}-1,3-dimethyl-1,2,3,4-tetrahydropyrimidine-2,4-dione
N-{2-[(1-methyl-1H-1,2,3,4-tetrazol-5-yl)sulfanyl]ethyl}-3-(1H-pyrazol-1-ylmethyl)benzamide
3-(2-fluoro-5-methoxyphenyl)pyridin-2-ol
(3S,4S)-1-[(6-hydroxy-2-methylpyrimidin-4-yl)methyl]-4-propylpyrrolidine-3-carboxylic acid
1-methyl-4-[2-(phenylsulfanyl)ethyl]-1,4,9-triazaspiro[5.6]dodecan-10-one
5-chloro-4,6-dimethyl-2-oxo-N-(thiolan-3-yl)-1,2-dihydropyridine-3-carboxamide
N-(furan-3-ylmethyl)-N-methyl-2-{[(3-methylthiophen-2-yl)methyl]amino}benzamide
(3R,4S)-4-cyclopropyl-1-(3-phenylbenzoyl)pyrrolidin-3-amine
N-({2-methylimidazo[2,1-b][1,3]thiazol-6-yl}methyl)-3-(pyridin-3-yl)propanamide
2-ethyl-N-[2-(pyridin-2-ylsulfanyl)ethyl]pyrimidine-5-carboxamide
6-phenyl-2-{2-phenyl-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-6-yl}pyridine-3-carboxylic acid
N-{[7-(5-acetylthiophen-2-yl)-5-fluoro-2,3-dihydro-1-benzofuran-2-yl]methyl}-2,2-dimethyloxane-4-carboxamide
(3aR,6aS)-5-[(1S,9aR)-octahydro-1H-quinolizin-1-ylmethyl]-2-methyl-octahydropyrrolo[3,4-c]pyrrole-1,3-dione
2-(2-methoxybutanoyl)-N-(5-methyl-1,3,4-thiadiazol-2-yl)-1,2,3,4-tetrahydroisoquinoline-7-sulfonamide
N-(4-methoxy-2-methylphenyl)-3-[1-(quinolin-2-yl)piperidin-3-yl]propanamide
N-{2-[(4-ethyl-5-methyl-4H-1,2,4-triazol-3-yl)sulfanyl]ethyl}pyrazolo[1,5-a]pyridine-7-carboxamide
2-(cyclopropylmethyl)-9-[3-(2-methyl-1H-imidazol-1-yl)propanoyl]-2,9-diazaspiro[5.5]undecan-3-one
2-methyl-8-[1-(thiophene-2-carbonyl)piperidin-4-yl]-1,3,8-triazaspiro[4.5]dec-1-en-4-one
2-(adamantan-1-yl)-N-[2-(pyrazin-2-yl)ethyl]acetamide
N-benzyl-5-{[(furan-2-ylmethyl)(prop-2-en-1-yl)amino]methyl}pyrimidin-2-amine
(3aR,6aR)-2-cyclopropanecarbonyl-5-{[1-(prop-2-en-1-yl)-1H-pyrazol-4-yl]methyl}-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
(3S,4R)-4-(3-methoxyphenyl)-1-[(2-methyl-1,3-oxazol-4-yl)methyl]pyrrolidine-3-carboxylic acid
1-(2,3-dihydroxypropyl)-6-methyl-4-(trifluoromethyl)-1,2-dihydropyridin-2-one
4-[(3-{[4-(hydroxymethyl)phenyl]methyl}pyrrolidin-1-yl)methyl]-1,5-dimethyl-2-phenyl-2,3-dihydro-1H-pyrazol-3-one
N3-(cyclohexylmethyl)-N5-[2-(1-methyl-1H-1,3-benzodiazol-2-yl)ethyl]-4-oxo-1-(propan-2-yl)-1,4-dihydropyridine-3,5-dicarboxamide
(2S,4R)-1-cyclopentyl-N-ethyl-4-(4-ethyl-5-methylthiophene-3-amido)pyrrolidine-2-carboxamide
1-[1-(2,1,3-benzoxadiazol-4-ylmethyl)piperidin-4-yl]-N-(pyridin-2-ylmethyl)piperidine-4-carboxamide
3-{1-[3-(4-methylphenyl)propanoyl]piperidin-3-yl}-1-(pyrrolidin-1-yl)propan-1-one
N-[(3-methoxyphenyl)methyl]-3-{1-[(2-methyl-1,3-thiazol-5-yl)methyl]piperidin-3-yl}propanamide
2-(3-{4H,5H,6H,7H-thieno[3,2-c]pyridin-5-ylmethyl}phenyl)-3,4,5,6,7,8-hexahydroquinazolin-4-one
N-{1-[5-methyl-1-(naphthalen-1-yl)-1H-pyrazol-4-yl]ethyl}-3-(morpholin-4-yl)benzamide
6-tert-butyl-N-[(5-methylthiophen-2-yl)methyl]-2-oxo-2,3-dihydropyrimidine-4-carboxamide
2-{[4-(3-hydroxyprop-1-yn-1-yl)thiophen-2-yl]methyl}-1,2,3,4-tetrahydroisoquinoline-3-carboxamide
(1R,9S)-5-amino-12-methyl-3-[1-(prop-2-en-1-yl)-1H-pyrazol-4-yl]-6,12-diazatricyclo[7.2.1.02,7]dodeca-2,4,6-triene-4-carbonitrile
2-[(3-methyl-1-propyl-1H-pyrazol-4-yl)formamido]-2-[2-(trifluoromethyl)phenyl]acetic acid
(3aS,6aS)-2-[(2-methyl-1H-imidazol-4-yl)methyl]-5-(oxan-4-yl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
3-[4-(3-fluorophenyl)-1H-pyrazol-5-yl]-1-(2-methylpropyl)piperidine
5-(2-{8-methylimidazo[1,2-a]pyridin-3-yl}acetyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-6-carboxylic acid
3-cyclopropyl-5-[3-(3-methylphenyl)-1H-pyrazol-4-yl]-1H-1,2,4-triazole
1-[2-methoxy-5-({[2-(methylsulfanyl)ethyl]amino}methyl)phenoxy]-3-(piperidin-1-yl)propan-2-ol
(1S,9S)-11-{[2-(7-methoxy-2H-1,3-benzodioxol-5-yl)-5-methyl-1,3-oxazol-4-yl]methyl}-7,11-diazatricyclo[7.3.1.02,7]trideca-2,4-dien-6-one
{[5-chloro-3-methoxy-2-(propan-2-yloxy)phenyl]methyl}(methyl)[(3-methyl-1,2,4-oxadiazol-5-yl)methyl]amine
3-methyl-5-[1-(3-phenyl-1H-pyrazole-5-carbonyl)pyrrolidin-2-yl]-1,2-oxazole
1-ethyl-5-(2-{2-methylimidazo[1,2-a]pyridin-3-yl}acetyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylic acid
N-ethyl-2-[(isoquinolin-5-yloxy)methyl]-N-propyl-1,3-oxazole-4-carboxamide
ethyl 4-[(4-methoxyphenyl)methyl]-1-(2-methyl-1-benzofuran-5-carbonyl)piperidine-4-carboxylate
N,3-dimethyl-2-oxo-N-[(2-phenyl-1,3-thiazol-4-yl)methyl]-2,3-dihydro-1,3-benzoxazole-5-carboxamide
N-[(2R)-1-hydroxy-3-methylbutan-2-yl]-5-(phenoxymethyl)-1H-pyrazole-3-carboxamide
(5S,9aS,9bS)-5-(2,1,3-benzoxadiazol-4-yl)-2-(3-methoxyphenyl)-octahydro-1H-pyrrolo[3,4-h]pyrrolizin-1-one
ethyl 4-{3-[4-(trifluoromethyl)benzoyl]piperidin-1-yl}piperidine-1-carboxylate