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N,N-dimethyl-1-[4-(1H-pyrazol-3-yl)benzoyl]azepan-4-amine
3-(1H-1,2,3-benzotriazol-1-yl)-1-{3-tert-butyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl}propan-1-one
8-methoxy-N-[1-(methoxymethyl)cyclopentyl]-2-oxo-1,2,3,4-tetrahydroquinoline-4-carboxamide
1-(1H-1,3-benzodiazole-5-carbonyl)-4-(4-methyl-1H-pyrazol-1-yl)piperidine-4-carboxylic acid
2-{[4-(1,3-dimethyl-1H-pyrazol-5-yl)-5-[(2-fluorophenyl)methyl]-4H-1,2,4-triazol-3-yl]sulfanyl}acetic acid
7-[2-(pyridin-2-ylsulfanyl)ethyl]-2-oxa-7-azaspiro[4.5]decan-8-one
N-[(2,4-dimethoxyphenyl)methyl]-4-{5-[(4-methylpiperidin-1-yl)methyl]-1H-1,2,3,4-tetrazol-1-yl}butanamide
1-methyl-N-{2-[(1-methyl-1H-1,2,3,4-tetrazol-5-yl)sulfanyl]ethyl}-6-propyl-1H-pyrazolo[3,4-d]pyrimidin-4-amine
N-[2-(dimethylamino)pentyl]-4-(propan-2-yl)pyrimidin-2-amine
2-methyl-7-[4-methyl-2-(propan-2-yl)pyrimidine-5-carbonyl]-2,7-diazaspiro[4.5]decane
N-{2-[(4-ethyl-5-methyl-4H-1,2,4-triazol-3-yl)sulfanyl]ethyl}-5,6-dimethylpyridine-3-carboxamide
1-methyl-4-{4-[1-(2-methylphenyl)-3-(2-methylpropyl)-1H-1,2,4-triazol-5-yl]butan-2-yl}piperazine
2-[(5-methyl-1,3,4-oxadiazol-2-yl)sulfanyl]-1-[(1S,5R)-3-(pyridine-2-carbonyl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]ethan-1-one
[(5-ethylpyridin-2-yl)methyl][(6-methoxypyridin-3-yl)methyl]methylamine
(2S,4R)-1-cyclopentanecarbonyl-N-ethyl-4-(2-fluorobenzamido)pyrrolidine-2-carboxamide
1-(4-methoxyphenyl)-5-(1-propoxyethyl)-1H-1,2,4-triazole
4-(2-methoxyphenoxy)-1-(6-methylpyridazin-3-yl)piperidine-4-carboxylic acid
1-(3-ethyl-5-methyl-1,2-oxazole-4-carbonyl)-3-(4-methylphenoxymethyl)piperidine
8-[2-(4-chlorophenoxy)ethyl]-2-(2-hydroxyethyl)-2,8-diazaspiro[5.5]undecan-3-one
2-{5-[2-(azocan-1-yl)ethyl]-3-(furan-2-yl)-1H-1,2,4-triazol-1-yl}acetic acid
2-{2-[1-(2-methyl-2,3-dihydro-1-benzofuran-5-yl)-1H-imidazol-2-yl]phenoxy}ethan-1-ol
1-[(1R,3S)-1,3-dihydroxy-7-azaspiro[3.5]nonan-7-yl]-2-(2-ethyl-1H-imidazol-1-yl)ethan-1-one
N-[(2S,4R,6S)-2-(2,3-dimethyl-1H-indol-7-yl)-6-(2-methylpropyl)oxan-4-yl]acetamide
N-(1-carbamoylcyclopentyl)-1-(piperidin-3-ylmethyl)-1H-1,2,3-triazole-4-carboxamide
1-[(3R,4S)-3-amino-4-(4-methoxyphenyl)pyrrolidin-1-yl]-3-(thiophen-3-yl)propan-1-one
6-(morpholine-4-sulfonyl)-2-(1H-pyrrole-2-carbonyl)-1,2,3,4-tetrahydroisoquinoline
2-tert-butyl-N-[3-(dimethyl-1,2-oxazol-4-yl)propyl]-4-hydroxypyrimidine-5-carboxamide
1-[(1,5-dimethyl-1H-pyrazol-4-yl)methyl]-4-[3-(trifluoromethyl)phenyl]piperidin-4-ol
(1R,5S)-3-({5-[(4-methylphenyl)sulfanyl]furan-2-yl}methyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
1-(1-{[2,4-dimethyl-6-(1H-pyrazol-1-yl)phenyl]methyl}piperidin-4-yl)pyrrolidin-2-one
N-{[(2S,4S)-4-fluoropyrrolidin-2-yl]methyl}-2-(1,1,2,2-tetrafluoroethoxy)benzamide
5-{[4-(3-methoxyphenyl)-3,3-dimethylpiperazin-1-yl]methyl}-N,N-dimethylpyrimidin-2-amine
3-[(3R,4S)-1-[(1-ethyl-1H-pyrazol-4-yl)methyl]-4-(morpholin-4-yl)piperidin-3-yl]propan-1-ol
2-{1-[(3,4-difluorophenyl)methyl]-4-{[4-(pyrimidin-2-yloxy)phenyl]methyl}piperazin-2-yl}ethan-1-ol
7-[(3,4-difluorophenyl)methyl]-2-(propan-2-yl)-2,7-diazaspiro[4.5]decan-6-one
2-[4-hydroxy-4-(5-methylpyridin-2-yl)piperidine-1-carbonyl]thiophene-3-sulfonamide
N-{[5-fluoro-7-(pyrimidin-5-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}-2-(methylsulfanyl)benzamide
3-butyl-4-({7-chloro-4-oxo-4H-pyrido[1,2-a]pyrimidin-2-yl}methyl)-1-methylpiperazin-2-one
2-(5-acetylthiophen-3-yl)-N-(1-cycloheptylpiperidin-3-yl)acetamide
1-{1-[1-(1,3-benzothiazol-2-yl)piperidin-4-yl]-1H-1,2,3-triazol-4-yl}ethan-1-ol
8-[(5-ethylpyridin-2-yl)methyl]-2-(3-methoxypropyl)-2,8-diazaspiro[4.5]decan-3-one
5-[(3R,4S)-4-(dimethylamino)-3-(3-hydroxypropyl)piperidine-1-carbonyl]-1-methyl-1,2,3,4-tetrahydropyrimidine-2,4-dione
N-{[1-methyl-2-(methylsulfanyl)-1H-imidazol-5-yl]methyl}-3-(1-methylpiperidin-3-yl)propanamide
methyl 4-({7-[(2-fluorophenyl)methyl]-2,7-diazaspiro[4.5]decan-2-yl}methyl)benzoate
2-(4-chloro-2-methylphenoxy)-1-{2-[2-(dimethylamino)ethyl]morpholin-4-yl}ethan-1-one
3-{imidazo[1,2-a]pyridin-2-yl}-N-[(5-methylfuran-2-yl)methyl]propanamide
N,N-diethyl-5-{1-[3-(1H-1,2,3,4-tetrazol-1-yl)propanoyl]pyrrolidin-2-yl}thiophene-2-carboxamide
1-ethyl-3-{1-[4-(1H-1,2,3,4-tetrazol-5-yloxy)phenyl]-1H-imidazol-2-yl}piperidine
4-[(3-fluorophenyl)methyl]-3-{2-oxo-2-[4-(pyrimidin-2-yl)piperazin-1-yl]ethyl}piperazin-2-one
({4-[(3,5-dimethyl-1H-pyrazol-1-yl)methyl]phenyl}methyl)(2-methoxyethyl)methylamine