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N-{[1-(1H-imidazol-1-ylmethyl)cyclopropyl]methyl}-3,6,7-trimethyl-1-benzofuran-2-carboxamide
2-ethyl-1-{[5-methyl-2-(2-methylphenyl)-1,3-oxazol-4-yl]methyl}piperidine
9-{[2-(methoxymethyl)pyrimidin-5-yl]methyl}-2-methyl-4-phenyl-2,9-diazaspiro[5.5]undecane
N-(1-benzylpyrrolidin-3-yl)-3-{1-[2-(methylamino)acetyl]piperidin-4-yl}propanamide
2-[4-(4-oxo-3,4-dihydro-2H-1-benzopyran-7-yl)-1H-pyrazol-1-yl]-N-[2-(propan-2-yl)-2H-1,2,3-triazol-4-yl]acetamide
1-{2-methyl-5-[3-(pyridin-4-yl)-1,2,4-oxadiazol-5-yl]phenyl}imidazolidin-2-one
1,2-dimethyl-4-{[1-(2-phenylethyl)-2-(propane-2-sulfonyl)-1H-imidazol-5-yl]methyl}piperazine
3-({[2-(5-cyclopentyl-1,2,4-oxadiazol-3-yl)ethyl]carbamoyl}amino)-4-fluorobenzamide
1-{[3,5-dimethyl-1-(propan-2-yl)-1H-pyrazol-4-yl]methyl}-N-(4-methoxyphenyl)piperidin-3-amine
N-({2,3-dimethylimidazo[2,1-b][1,3]thiazol-6-yl}methyl)-7-(propan-2-yl)-[1,2,4]triazolo[1,5-a]pyrimidine-5-carboxamide
1-{1-methyl-6-propyl-1H-pyrazolo[3,4-d]pyrimidin-4-yl}-4-(1H-1,2,3,4-tetrazol-5-yl)piperidine
2-(dimethylamino)-2-(3-fluorophenyl)-1-{4-[(3-methyl-1,2,4-oxadiazol-5-yl)methyl]piperidin-1-yl}ethan-1-one
3-{[(4-fluorophenyl)methyl]sulfanyl}-N-methyl-N-[(1-methyl-1H-imidazol-2-yl)methyl]propanamide
N-[(3S,4R)-1-(2,3-dihydro-1H-indene-5-carbonyl)-4-(4-methylphenyl)pyrrolidin-3-yl]acetamide
4-{[2-(cyclopentylmethyl)-1H-imidazol-4-yl]methyl}-2-ethyl-1-(propan-2-yl)piperazine
2-[(1-methyl-1H-indol-3-yl)sulfanyl]-N-[(3-methylthiophen-2-yl)methyl]acetamide
[(3R,5R)-5-{[(2-methoxyethyl)(methyl)amino]methyl}-1-(3-methylpyrazin-2-yl)piperidin-3-yl]methanol
N-{1-[2-(4-methoxyphenyl)ethyl]-5-oxopyrrolidin-3-yl}-3-methylthiophene-2-carboxamide
7-methoxy-3-({methyl[3-(1H-pyrazol-1-yl)propyl]amino}methyl)-1,2-dihydroquinolin-2-one
2-(1-{1-[(6-methoxypyridin-3-yl)methyl]piperidin-4-yl}-1H-1,2,3-triazol-4-yl)propan-2-ol
N-[(1S,2R)-1-hydroxy-1-(4-hydroxyphenyl)propan-2-yl]-3-methoxy-5-methylthiophene-2-carboxamide
N-methyl-2-[5-(morpholin-4-ylmethyl)-1H-1,2,3,4-tetrazol-1-yl]-N-[(3-phenyl-1,2,4-oxadiazol-5-yl)methyl]acetamide
3-[3-(2,5-dimethoxyphenyl)pyrrolidine-1-carbonyl]pyridine
1-(cyclohex-1-ene-1-carbonyl)-N-[4-(3,5-dimethyl-1H-pyrazol-1-yl)phenyl]piperidine-2-carboxamide
2-(morpholin-4-yl)-N-(1,2-oxazol-3-ylmethyl)-6-{8-thiatricyclo[7.4.0.02,7]trideca-1(9),2(7),3,5,10,12-hexaen-6-yl}pyridine-3-carboxamide
3-(3-fluorophenyl)-4-[1-(thiophen-2-ylmethyl)-1H,4H-pyrazolo[3,4-d]imidazol-5-yl]-1H-pyrazole
N-[(5-methoxy-1H-indol-2-yl)methyl]-2,5-dimethyl-[1,3]oxazolo[5,4-d]pyrimidin-7-amine
{1-[(5-tert-butyl-1H-pyrazol-3-yl)methyl]-4-[(dimethylamino)methyl]piperidin-4-yl}methanol
(2S)-2-{[(4-hydroxy-6,8-dimethylquinolin-2-yl)methyl]amino}-3-methylbutanamide
4-benzyl-1-{2-[3-(3,5-dimethyl-1H-pyrazol-1-yl)azetidin-1-yl]-2-oxoethyl}pyrrolidin-2-one
4,4-difluoro-1-({3-[3-(piperidin-1-yl)propoxy]phenyl}methyl)piperidine
1-methyl-2-[3-methyl-1-(pyridin-2-yl)-1H-1,2,4-triazol-5-yl]azepane
5-(4-{[4-(cyclopentyloxy)phenyl]methyl}piperazin-1-yl)-2-methyl-2,3-dihydropyridazin-3-one
{4-[3-(2-methoxyethyl)-1-(2-methoxyphenyl)-1H-1,2,4-triazol-5-yl]phenyl}methanol
N-[(3-chlorophenyl)methyl]-3-[3-(cyclopropylmethyl)-3-(hydroxymethyl)piperidin-1-yl]propanamide
N-(2-methyl-1-benzofuran-5-yl)-4-(2-methylpyridin-4-yl)-1,4-diazepane-1-carboxamide
3-(4,5,6,7-tetrahydro-1H-indazol-3-yl)-1-(thiomorpholin-4-yl)propan-1-one
(3R,4R)-3-cyclobutyl-1-[5-(methoxymethyl)thiophene-2-carbonyl]-4-methylpyrrolidin-3-ol
(2S,4R)-N-methyl-1-(propan-2-yl)-4-({[3-(trifluoromethyl)phenyl]methyl}amino)pyrrolidine-2-carboxamide
3-{3-[(1-methylpiperidin-4-yl)methyl]-1,2,4-oxadiazol-5-yl}quinoline
1-{5-[7-(2-phenylethyl)-2,7-diazaspiro[4.5]decane-2-carbonyl]thiophen-2-yl}ethan-1-one
4-(1H-imidazol-1-yl)-1-(morpholine-4-sulfonyl)piperidine-4-carboxylic acid
3-(dimethylamino)-N-[3-(3-methylphenyl)phenyl]piperidine-1-carboxamide
(2S)-1-acetyl-N-({5-[4-(methylsulfanyl)phenyl]-2,3-dihydro-1-benzofuran-2-yl}methyl)pyrrolidine-2-carboxamide
N-[2-(3,5-dimethyl-1H-pyrazol-4-yl)ethyl]-2-{1-[(4-fluorophenyl)methyl]-3-oxopiperazin-2-yl}-N-methylacetamide
ethyl[(5-ethyl-1,3,4-oxadiazol-2-yl)methyl]({3-phenylpyrazolo[1,5-a]pyrimidin-6-yl}methyl)amine
methyl 4-{[1-(2-methoxyethyl)-2,4-dioxo-3-[3-(pyridin-3-yl)propyl]-1,3,8-triazaspiro[4.5]decan-8-yl]methyl}benzoate
2-(4-{[2-methyl-4-(1H-pyrazol-1-yl)phenyl]methyl}-1-[(2-methylphenyl)methyl]piperazin-2-yl)ethan-1-ol
N-{[6-(thiophen-3-yl)-2H-[1,3]dioxolo[4,5-g]quinolin-7-yl]methyl}-1,2,3,4-tetrahydronaphthalen-1-amine
2-{4-[4-(3-fluorophenyl)-1H-pyrazol-5-yl]piperidin-1-yl}pyridine-4-carboxamide