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1-[2-(cyclopent-2-en-1-yl)acetyl]-4-(1H-imidazol-1-yl)piperidine-4-carboxylic acid
1-(4-benzylpiperazin-1-yl)-3-[1-(pyridin-2-ylmethyl)piperidin-3-yl]propan-1-one
3-[5-(4-methylphenoxymethyl)-1,3,4-thiadiazol-2-yl]-1-(pyridin-3-ylmethyl)urea
4-[3-(1H-1,3-benzodiazol-2-yl)azetidine-1-carbonyl]-N-methyl-1,3-thiazol-2-amine
2-{2-[(3aS,6aS)-1-methyl-octahydropyrrolo[3,4-b]pyrrol-5-yl]-2-oxoethyl}-3-phenylcyclopent-2-en-1-one
1-(piperidin-1-yl)-2-[4-(pyridin-4-yl)piperazin-1-yl]ethan-1-one
2-(4-chlorophenyl)-3-[(4-methylpiperazin-1-yl)methyl]-7-(methylsulfanyl)quinoline
N-[(6-fluoro-1H-1,3-benzodiazol-2-yl)methyl]-N-methyl-1-(oxan-4-yl)piperidine-3-carboxamide
N-{[2-(4-fluorophenyl)-3-methyl-1H-indol-5-yl]methyl}-2-(2-methyl-1,3-thiazol-4-yl)acetamide
{[2-(azepane-1-carbonyl)-7-methylimidazo[1,2-a]pyridin-3-yl]methyl}[2-(1H-imidazol-4-yl)ethyl]amine
2-(3-chloro-5-fluorophenyl)-1-[(3R,4R)-3-(hydroxymethyl)-4-(piperidin-1-ylmethyl)pyrrolidin-1-yl]ethan-1-one
2-methyl-4-[4-({4-[(3-methyl-1,2,4-oxadiazol-5-yl)methyl]piperidin-1-yl}methyl)phenyl]butan-2-ol
N-{1-[1-(3-chlorobenzoyl)piperidin-4-yl]-2-(3-methoxyphenyl)ethyl}-N-methyl-3-(methylsulfanyl)propanamide
1-[(3,5-dimethyl-1H-pyrazol-4-yl)methyl]-5-(3-ethoxy-4-methoxyphenyl)-4-phenyl-1H-imidazole
1-cyclopropyl-N-(3-hydroxy-2,2-dimethylpropyl)-5-oxopyrrolidine-3-carboxamide
N-{[4-(3-fluorophenyl)oxan-4-yl]methyl}-8-methoxy-3,4-dihydro-2H-1-benzopyran-3-carboxamide
N-(4-chlorophenyl)-3-{1-[(4-ethyl-4H-1,2,4-triazol-3-yl)methyl]piperidin-3-yl}propanamide
N-[2-(ethylsulfanyl)phenyl]-4-(thiophene-2-carbonyl)piperazine-1-carboxamide
2-{[(3S,4S)-3-hydroxy-4-(pyrrolidin-1-yl)pyrrolidin-1-yl]methyl}benzonitrile
2-{4-[(2,4-difluorophenyl)methyl]-1-[(5-methylfuran-2-yl)methyl]piperazin-2-yl}ethan-1-ol
2-{4-[(1-methyl-1H-indol-3-yl)methyl]-1-[1-(propan-2-yl)piperidin-4-yl]piperazin-2-yl}ethan-1-ol
5-{[4-benzyl-3-(2-hydroxyethyl)piperazin-1-yl]methyl}-1,2,4-oxadiazole-3-carboxamide
{4-[(2-chlorophenyl)methyl]-1-(4-methyl-1H-imidazole-5-carbonyl)piperidin-4-yl}methanol
5-{[benzyl(methyl)amino]methyl}-N-methyl-N-[(2-methyl-1,3-thiazol-4-yl)methyl]-1,2-oxazole-3-carboxamide
(2R)-2-amino-4-methyl-1-[4-(pyridin-3-ylmethoxy)piperidin-1-yl]pentan-1-one
(4aS,8aR)-1-(3-aminopropyl)-6-[(2E)-3-(4-fluorophenyl)prop-2-en-1-yl]-decahydro-1,6-naphthyridin-2-one
5-(2,4-difluorophenoxymethyl)-N-(2-hydroxyethyl)-1,2-oxazole-3-carboxamide
5-[2-(1-methylcyclopropyl)ethyl]-3-(oxolan-3-yl)-1H-1,2,4-triazole
6-(4-fluorophenyl)-2-[2-(2-methylpropyl)-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-6-yl]pyridine-3-carboxylic acid
4-{[2-(3-fluorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-1-methyl-1,4,9-triazaspiro[5.6]dodecan-10-one
2-(10-methoxy-3,4,5,6-tetrahydro-2H-1,5-benzoxazocin-5-yl)-3H,4H,5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-one
4-({[3-cyclopropyl-1-(2-phenylethyl)-1H-1,2,4-triazol-5-yl]methyl}sulfanyl)pyridine
3-(1-methyl-1H-pyrazol-4-yl)-1-{2-[4-methyl-6-(trifluoromethyl)pyrimidin-2-yl]ethyl}urea
1-(2-{1-[3-(difluoromethoxy)benzoyl]piperidin-4-yl}ethyl)pyrrolidin-2-one
N-(2-oxoazepan-3-yl)-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
1-(8-chloroquinolin-2-yl)-3',4'-dihydro-1'H-spiro[piperidine-4,2'-quinoxaline]-3'-one
N-{[7-fluoro-5-(3-fluoro-4-methylphenyl)-2,3-dihydro-1-benzofuran-2-yl]methyl}-3-(1H-1,2,4-triazol-1-yl)propanamide
N-{[3-(pyrazin-2-yl)-1H-1,2,4-triazol-5-yl]methyl}-1-[(1s,4s)-4-aminocyclohexyl]-1H-1,2,3-triazole-4-carboxamide
N-[(1,2-dimethyl-1H-1,3-benzodiazol-5-yl)methyl]-4-hydroxy-2-(pyridin-3-yl)pyrimidine-5-carboxamide
methyl 4-{[(3R,4R)-4-[4-(2-fluorophenyl)piperazin-1-yl]-3-hydroxypiperidin-1-yl]methyl}benzoate
1-{3-[({3-[2-hydroxy-3-(morpholin-4-yl)propoxy]phenyl}methyl)amino]propyl}pyrrolidin-2-one
4-{3-[2-(4-fluorophenyl)ethyl]piperidin-1-yl}-4-oxobutane-1-sulfonamide
2-[2-methyl-3-(1-methyl-1H-1,3-benzodiazol-2-yl)-1H-indol-1-yl]acetic acid
3-(3-chloro-1,2-oxazol-5-yl)-1-[4-(1-hydroxy-3-phenylpropyl)piperidin-1-yl]propan-1-one
6-[(diethylamino)methyl]-N-(1H-indol-5-yl)pyrazolo[1,5-a]pyrimidine-3-carboxamide
N-{1H,4H,5H,6H,7H,8H-cyclohepta[c]pyrazol-3-ylmethyl}-N,2,8-trimethylquinoline-4-carboxamide
(2R,6R)-11-methoxy-4-[(1-methyl-1H-pyrazol-4-yl)methyl]-8-oxa-4-azatricyclo[7.4.0.02,6]trideca-1(13),9,11-triene-6-carboxylic acid
N-{2-[5-(3-cyanophenyl)-4-phenyl-1H-imidazol-1-yl]ethyl}acetamide
2-[2-({[2-(1H-imidazol-1-yl)ethyl](methyl)amino}methyl)phenoxy]ethan-1-ol
3-(2-hydroxyphenyl)-N-(2-methoxyethyl)-N-(1-methylpiperidin-4-yl)-1H-pyrazole-5-carboxamide