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1-({3-[(1S,5R)-1,3,3-trimethyl-6-azabicyclo[3.2.1]octane-6-carbonyl]-1H-pyrazol-5-yl}methyl)-1H-1,3-benzodiazole
N-{[(2S)-5-oxopyrrolidin-2-yl]methyl}-5-(propan-2-yl)-N-(pyridin-4-ylmethyl)-1,2-oxazole-3-carboxamide
2-{1-[(2-chloro-6-fluorophenyl)methyl]-3-oxopiperazin-2-yl}-N-methyl-N-[(3-methyl-1,2-oxazol-5-yl)methyl]acetamide
2-(2-amino-6-methylpyrimidin-4-yl)-7-(oxan-4-yl)-2,7-diazaspiro[4.5]decan-6-one
N-[3-(4-methoxyphenyl)propyl]-1-methyl-2-oxo-1,2-dihydroquinoline-4-carboxamide
2-{[(4-fluorophenyl)methyl](methyl)amino}-1-[(3R,4R)-3-(hydroxymethyl)-4-(piperidin-1-ylmethyl)pyrrolidin-1-yl]ethan-1-one
(4aR,8aS)-6-(furan-2-carbonyl)-1-(quinoline-6-carbonyl)-decahydro-1,6-naphthyridine
1-[5-(4-methylphenyl)-1H-pyrazole-3-carbonyl]-4-(pyridin-4-yl)piperazine
2-(3-benzyl-1-methyl-2-oxo-2,3-dihydro-1H-indol-3-yl)-N-(2-methoxyethyl)acetamide
1-[(3-methoxyphenyl)methyl]-4-[3-(2-methyl-5-oxopyrrolidin-2-yl)propanoyl]piperazin-2-one
3-[1-({4-[methyl(phenyl)amino]phenyl}methyl)piperidin-3-yl]-1-(pyrrolidin-1-yl)propan-1-one
1-[(2-methyl-1,3-thiazol-4-yl)methyl]-4-{[3-(2-phenylethyl)-1,2,4-oxadiazol-5-yl]methyl}piperazine
4-({[6-(azepan-1-yl)-[1,2,5]oxadiazolo[3,4-b]pyrazin-5-yl]amino}methyl)-1-ethylpyrrolidin-2-one
2-ethyl-4-phenyl-9-(pyridine-3-carbonyl)-2,9-diazaspiro[5.5]undecane
(2-{1-[(2,3-difluoro-6-methoxyphenyl)methyl]piperidin-2-yl}ethyl)dimethylamine
methyl 4-(4-{[(1,1-dioxo-1λ6-thiolan-3-yl)(prop-2-en-1-yl)amino]methyl}-5-methyl-1,3-oxazol-2-yl)benzoate
N-{2-[2-methyl-5-(morpholine-4-sulfonyl)-1H-1,3-benzodiazol-1-yl]ethyl}cyclopropanecarboxamide
N-[3-(dimethyl-1H-1,2,4-triazol-1-yl)propyl]-5-hydroxy-1,2-dimethyl-1H-indole-3-carboxamide
1-{[2-(6-chloro-2H-1,3-benzodioxol-5-yl)-5-methyl-1,3-oxazol-4-yl]methyl}-4-(furan-2-carbonyl)-1,4-diazepane
1-{2-[(2R,3R,6R)-3-(4-fluorophenyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]-2-oxoethyl}piperidin-2-one
1-(2-methylpropyl)-3-(morpholine-4-carbonyl)-N-{[4-(trifluoromethoxy)phenyl]methyl}-4,5,6,7-tetrahydro-1H-indazol-5-amine
1-[2-(4-chlorophenyl)ethyl]-5-(morpholine-4-carbonyl)piperidin-2-one
3-{2-[1-(1,3-thiazol-4-ylmethyl)piperidin-2-yl]ethyl}phenol
3-(3-hydroxy-3-methylbutyl)-N-[1-(2-hydroxyphenyl)ethyl]benzamide
2-{[(3aS,6aS)-1-methyl-octahydropyrrolo[3,4-b]pyrrol-5-yl]methyl}-1-(4-methoxyphenyl)-1H-imidazole
2-[(2,6-dichlorophenyl)methyl]-4-hydroxy-N-[(2-methyl-1,3-thiazol-4-yl)methyl]pyrimidine-5-carboxamide
3-cyclobutyl-4-pentyl-4,5-dihydro-1H-1,2,4-triazol-5-one
5-(2-cyclopentylacetamido)-N-[2-(furan-2-yl)ethyl]-1-methyl-2-(oxolan-2-yl)-1H-1,3-benzodiazole-7-carboxamide
N-[2-chloro-5-(pyrrolidine-1-carbonyl)phenyl]-4-ethylpiperazine-1-carboxamide
2-methyl-N-[(4-{3-oxa-9-azaspiro[5.5]undecane-9-carbonyl}phenyl)methyl]propanamide
N-[3-(4-{[(4-methyl-1,2,5-oxadiazol-3-yl)methyl]amino}piperidin-1-yl)phenyl]-3-(trifluoromethyl)benzamide
methyl 4-({[(5-cyclobutyl-1,2,4-oxadiazol-3-yl)methyl](ethyl)carbamoyl}amino)benzoate
methyl 4-(3-ethoxyphenyl)-1-methyl-1H-pyrazole-5-carboxylate
4-(3-chloro-4-methylphenyl)-3-[2-(3,5-dimethyl-1H-pyrazol-4-yl)ethyl]-4,5-dihydro-1H-1,2,4-triazol-5-one
4-(3-{5-[(dimethylamino)methyl]-4-methyl-4H-1,2,4-triazol-3-yl}piperidine-1-carbonyl)piperidin-4-amine
2-{1-methyl-4-[4-(1-methyl-1H-pyrazol-4-yl)pyrimidin-2-yl]piperazin-2-yl}ethan-1-ol
1-(2-chlorophenyl)-4-(2-{imidazo[1,2-a]pyridin-3-yl}acetyl)-5-methylpiperazin-2-one
4-{2-cyclopropyl-4-phenyl-2,9-diazaspiro[5.5]undecan-9-yl}pyrimidin-2-amine
3-(5-methylfuran-2-yl)-N-[3-(pyridin-3-yloxy)propyl]-1H-pyrazole-5-carboxamide
1-(2-cyclohexylethyl)-3-({[(1-ethyl-1H-imidazol-2-yl)methyl]amino}methyl)-3-hydroxypiperidin-2-one
1-(4-methylquinazolin-2-yl)-N-{spiro[bicyclo[2.2.1]heptane-7,1'-cyclopropan]-2-en-6-ylmethyl}piperidine-4-carboxamide
1-(3-oxo-3-{2-[2-(1H-pyrazol-1-yl)ethyl]piperidin-1-yl}propyl)azepan-2-one
2-(dimethylamino)-7-[4-(1H-pyrazol-3-yl)benzoyl]-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
5-[2-(4-fluorophenyl)piperidine-1-carbonyl]-7H-[1,3]thiazolo[3,2-a]pyrimidin-7-one
3-methyl-1-{2-[2-(3-methyl-1,2-oxazol-5-yl)pyrrolidin-1-yl]-2-oxoethyl}-1,2-dihydroquinoxalin-2-one
4-(2,4-dimethoxyphenyl)pyridin-2-amine
1-{6-chloroimidazo[1,2-a]pyridine-2-carbonyl}-4-[(4-methyl-4H-1,2,4-triazol-3-yl)methyl]piperidine
[(1-benzyl-1H-pyrazol-4-yl)methyl](benzylsulfamoyl)amine
5-(5-ethylfuran-2-yl)-1-(1H-imidazol-2-ylmethyl)-4-phenyl-1H-imidazole
3-fluoro-N-{[3-methoxy-4-(oxolan-3-yloxy)phenyl]methyl}-N-(pyridin-3-ylmethyl)benzamide