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2-(2,5-dioxoimidazolidin-1-yl)-N-[1-(1-methyl-1H-pyrazol-5-yl)propyl]acetamide
N-(cyclobutylmethyl)-4-[5-(morpholin-4-ylmethyl)-1H-1,2,3,4-tetrazol-1-yl]-N-(oxolan-2-ylmethyl)butanamide
N-({5-[(3-methyl-1-benzofuran-2-yl)methyl]-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)cyclobutanecarboxamide
1-[4-(3-ethyl-1,2,4-oxadiazol-5-yl)phenyl]-3-[2-(4-ethyl-4H-1,2,4-triazol-3-yl)ethyl]urea
5-(3-methyl-1,2,4-oxadiazol-5-yl)-2-[4-(pyrrolidine-1-carbonyl)piperidin-1-yl]pyridine
N-[2-(1H-1,3-benzodiazol-2-yl)ethyl]-6-(4H-1,2,4-triazol-4-yl)pyridine-3-carboxamide
2,3,4-trifluoro-N-(1,4-oxazepan-6-ylmethyl)benzene-1-sulfonamide
3-cyclopropyl-5-[(4,5-dimethyl-1H-imidazol-1-yl)methyl]-1-[(2-methylphenyl)methyl]-1H-1,2,4-triazole
3-[(4-methoxyphenyl)methyl]-1-methyl-8-{1-[3-(trifluoromethyl)phenyl]propan-2-yl}-1,3,8-triazaspiro[4.5]decane-2,4-dione
9-(cyclopropylmethyl)-4-[5-fluoro-4-(methylamino)pyrimidin-2-yl]-1-methyl-1,4,9-triazaspiro[5.6]dodecan-10-one
2-(propan-2-yl)-7-{[4-(propan-2-yl)phenyl]methyl}-2,7-diazaspiro[4.5]decan-6-one
2-methyl-5-(propan-2-yl)-N-[3-(1H-pyrazol-1-yl)propyl]pyrazolo[1,5-a]pyrimidin-7-amine
N-[(5-{[(2-fluorophenyl)methyl]sulfanyl}-4-(2-methylpropyl)-4H-1,2,4-triazol-3-yl)methyl]-2-(5-methyl-1H-pyrazol-1-yl)acetamide
3-(5-amino-1H-1,2,4-triazol-3-yl)-N-[(3-chlorophenyl)methyl]-N-propylpropanamide
propyl 3-{[2-(4-methoxyphenyl)phenyl]carbamoyl}piperidine-1-carboxylate
1-[4-(1,3-benzothiazol-2-yl)piperazin-1-yl]-3-(3-chloro-1H-1,2,4-triazol-5-yl)propan-1-one
4-(1H-imidazol-1-yl)-1-[5-oxo-1-(prop-2-en-1-yl)pyrrolidine-3-carbonyl]piperidine-4-carboxylic acid
1-{1-[(2-chlorophenyl)methyl]-1H-1,2,3-triazole-4-carbonyl}-4-methylpiperazine
N-[2-(3-methoxyphenyl)ethyl]-5-methylpyrazolo[1,5-a]pyrimidin-7-amine
N-cyclopentyl-N'-[3-(4-hydroxypiperidin-1-yl)propyl]butanediamide
N-(1,3-dihydroxypropan-2-yl)-5-(3-methoxyphenoxymethyl)-1H-pyrazole-3-carboxamide
N-methyl-2-{1-oxo-1H,2H-pyrrolo[1,2-d][1,2,4]triazin-2-yl}-N-{[5-(propan-2-yl)-1,2-oxazol-3-yl]methyl}acetamide
1-{2-cyclopentyl-3-oxo-2,9-diazaspiro[5.5]undecan-9-yl}-4-phenylbutane-1,4-dione
(2R,3R,6R)-3-(3-methoxyphenyl)-5-[(2-methyl-1,3-thiazol-4-yl)methyl]-1,5-diazatricyclo[5.2.2.02,6]undecane
1-benzyl-3-(2-methoxyethyl)-8-[(2-methyl-1H-imidazol-4-yl)methyl]-1,3,8-triazaspiro[4.5]decane-2,4-dione
1-[(1,2-dimethyl-1H-imidazol-5-yl)methyl]-3-phenylpiperidine
6-[1-butyl-3-(thiophen-2-ylmethyl)-1H-1,2,4-triazol-5-yl]-2-methyl-2H,3H,5H,6H,7H,8H-[1,2,4]triazolo[4,3-a]pyridin-3-one
1-[(3R,4S)-3-(dimethylamino)-4-phenylpyrrolidine-1-carbonyl]cyclopropane-1-carboxamide
5-[(1S,5R)-3-[(4-methyl-1H-imidazol-5-yl)methyl]-3,6-diazabicyclo[3.2.2]nonane-6-carbonyl]-1H-1,2,3-benzotriazole
4-(1-{[2-(3-methylphenyl)-1,3-thiazol-4-yl]methyl}-1H-imidazol-2-yl)pyridine
1-(4-benzylpiperazin-1-yl)-3-(1-cyclohexanecarbonylpiperidin-3-yl)propan-1-one
N-[(1,3-dimethyl-1H-pyrazol-5-yl)methyl]-4-(piperidin-1-yl)butanamide
N-[(3S,4R)-1-[6-(piperidine-1-carbonyl)pyrazin-2-yl]-4-(propan-2-yl)pyrrolidin-3-yl]acetamide
5-ethyl-4-(4-methoxy-4-phenylpiperidin-1-yl)pyrimidin-2-amine
2-ethyl-4-methyl-N-({2-methylimidazo[2,1-b][1,3,4]thiadiazol-6-yl}methyl)-1,3-oxazole-5-carboxamide
1'-[(6-hydroxy-1,4-oxazepan-6-yl)methyl]-1-methyl-1,2-dihydrospiro[indole-3,4'-piperidine]-2-one
2-[1-(2-chlorophenyl)-5-oxo-3-phenyl-4,5-dihydro-1H-1,2,4-triazol-4-yl]-N-(3-hydroxypropyl)acetamide
5-({3-[1-(4-chlorophenyl)cyclopentyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl}methyl)-2-methylpyrimidine
5-{1-[(3-chloropyridin-4-yl)methyl]piperidin-4-yl}-5-(pyridin-2-yl)imidazolidine-2,4-dione
(3S,4R)-1-(1-aminocyclopropanecarbonyl)-4-(4-fluorophenyl)pyrrolidine-3-carboxylic acid
ethyl 5-{[ethyl(2-hydroxyethyl)amino]methyl}-1-(4-phenyl-1,3-thiazol-2-yl)-1H-pyrazole-4-carboxylate
3-[2-({dimethyl-[1,2]oxazolo[5,4-d]pyrimidin-4-yl}amino)ethyl]-1,3-oxazinan-2-one
3-acetamido-N-(quinolin-6-yl)pyrrolidine-1-carboxamide
6-[4-(dimethylamino)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidine-7-carbonyl]-4-methyl-1,3-benzothiazol-2-amine
N-(butan-2-yl)-3-(5-methyl-1,2,4-oxadiazol-3-yl)-N-(pyridin-4-ylmethyl)benzamide
1-{4-[(6-chloropyridin-3-yl)methyl]piperazin-1-yl}-3-(1-methylpiperidin-2-yl)propan-1-one
(4aS,7aR)-1-(2-fluorobenzoyl)-4-methanesulfonyl-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
N-{3-[methyl(phenyl)amino]propyl}-3-(trifluoromethyl)-1H-pyrazole-5-carboxamide
N-methyl-5-(propan-2-yl)-N-{[2-(pyrrolidin-1-ylmethyl)phenyl]methyl}-1,2-oxazole-3-carboxamide
(3aR,5S,6S,7aS)-2-(5-phenyl-1,2,4-oxadiazol-3-yl)-octahydro-1H-isoindole-5,6-diol