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6-chloro-2-methyl-N-{1-[3-(2-methylpropyl)-1,2,4-oxadiazol-5-yl]ethyl}imidazo[1,2-a]pyridine-3-carboxamide
1-methyl-2-[1-(3-propyl-1H-pyrazole-4-carbonyl)pyrrolidin-2-yl]-1H-1,3-benzodiazole
N-[3-(2-ethyl-1H-imidazol-1-yl)propyl]-1-{thieno[3,2-d]pyrimidin-4-yl}piperidin-4-amine
(2S,4R)-1-(2,2-diphenylethyl)-N-(propan-2-yl)-4-[(propan-2-yl)amino]pyrrolidine-2-carboxamide
N-ethyl-N-[2-(2-fluorophenoxy)ethyl]-3-[(5-methyl-1,3,4-thiadiazol-2-yl)sulfanyl]propanamide
1-benzoyl-N-[(2-propyl-1,3-thiazol-4-yl)methyl]piperidin-4-amine
N-({5-[(2-ethylphenyl)methyl]-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)cyclobutanecarboxamide
(3R,4S)-3,4-dimethyl-1-[4-(pyrrolidin-1-yl)benzoyl]piperidin-4-ol
6,6-dimethyl-1-(2-methylphenyl)-N-[(6-methylpyridin-2-yl)methyl]-4,5,6,7-tetrahydro-1H-indazol-4-amine
3-(2-chlorophenyl)-3-(3-hydroxyphenyl)-N-methyl-N-(pyrazin-2-ylmethyl)propanamide
2-[(5-methylpyrazin-2-yl)methyl]-8-(3-methylpyridin-4-yl)-2,8-diazaspiro[5.5]undecan-3-one
N-[2-(pyridin-4-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-yl]piperidin-4-amine
(3S,4S)-1-(3,5-dichloro-4-methylbenzoyl)-4-(propan-2-yloxy)pyrrolidin-3-ol
8-(6-methyl-4-oxo-4H-pyran-2-carbonyl)-1-oxa-3,8-diazaspiro[4.6]undecan-2-one
2-[(4-hydroxyquinazolin-2-yl)sulfanyl]-N-[(2-methyl-1,3-thiazol-4-yl)methyl]acetamide
1-(5-acetyl-2-methoxyphenyl)-3-{[2-(dimethylamino)-1,3-thiazol-4-yl]methyl}urea
5-(4-cyclohexylpiperazin-1-yl)-3-(morpholine-4-carbonyl)-1-propyl-4,5,6,7-tetrahydro-1H-indazole
2-butyl-4-{[3-(2,6-dimethylphenoxy)azetidin-1-yl]methyl}-1H-imidazole
3-methyl-8-[3-(5-methylthiophen-2-yl)-1H-pyrazole-5-carbonyl]-1-oxa-3,8-diazaspiro[4.6]undecan-2-one
benzyl(cyclopropylmethyl){[2-(2,3-difluorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}amine
2-methyl-N-[(3R)-pyrrolidin-3-yl]-1,3-benzothiazole-6-carboxamide
2-[4-(1H-pyrazol-1-yl)phenyl]pyridine-4-carboxamide
4-benzyl-3-butyl-1-[2-(1,4-oxazepan-4-yl)-2-oxoethyl]-4,5-dihydro-1H-1,2,4-triazol-5-one
N-{[4-(3-fluorophenyl)-5-(pyridin-2-yl)-1H-imidazol-2-yl]methyl}-1,4-dioxane-2-carboxamide
5-{2-[2-(morpholin-4-yl)ethyl]piperidine-1-carbonyl}-1H-1,2,3-benzotriazole
3-(1H-indazol-4-yl)-1-methyl-1-[3-(1-methyl-1H-pyrazol-4-yl)propyl]urea
(3S,4S)-1-(2-methyl-1H-1,3-benzodiazole-5-carbonyl)-4-(pyridin-2-yl)pyrrolidine-3-carboxylic acid
2-(dimethylamino)-2-(3-fluorophenyl)-N-methyl-N-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]acetamide
N-{[3-(ethoxymethyl)-4-methoxyphenyl]methyl}-3,4-dihydro-2H-1-benzopyran-3-amine
6-methoxy-2-oxo-N-[3-(4H-1,2,4-triazol-4-yl)propyl]-1,2,3,4-tetrahydroquinoline-4-carboxamide
1-[2-(3-hydroxypiperidin-1-yl)acetyl]-3',4'-dihydro-1'H-spiro[piperidine-4,2'-quinoxaline]-3'-one
5-[3-(1-ethyl-1H-imidazol-2-yl)piperidine-1-carbonyl]-4-propylpyrimidine
{[3-(2-chlorophenyl)-1-(4-methoxyphenyl)-1H-pyrazol-4-yl]methyl}[2-(1H-1,2,3-triazol-5-ylsulfanyl)ethyl]amine
N-(5-{[4-(4-benzyl-2,5-dioxoimidazolidin-4-yl)piperidin-1-yl]methyl}thiophen-2-yl)acetamide
4-{1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl}-2-methylquinoline
N-cyclohexyl-3-({2,5-dimethylpyrazolo[1,5-a]pyrimidin-7-yl}amino)propanamide
3-[2-(dimethyl-1H-1,2,4-triazol-1-yl)ethyl]-1-(6-methyl-2H-1,3-benzodioxol-5-yl)urea
1-{2-[methyl({[4-(1H-pyrazol-1-ylmethyl)phenyl]methyl})amino]ethyl}cyclopentan-1-ol
N-(2-methoxyethyl)-N-(pyridin-4-ylmethyl)-2-(pyrrolidin-3-yl)acetamide
6-methyl-2-oxo-N-{[1-(1H-pyrazol-1-ylmethyl)cyclopropyl]methyl}-4-(thiophen-2-yl)-1,2,3,4-tetrahydropyrimidine-5-carboxamide
8-(1-methyl-1H-pyrazole-5-carbonyl)-2-propyl-2,8-diazaspiro[4.5]decane-3-carboxylic acid
6-{8-[(5-methylpyrazin-2-yl)methyl]-9-oxo-2,8-diazaspiro[5.5]undecan-2-yl}pyridine-3-carbonitrile
(4S)-3,3,4-trimethyl-1-[3-(trifluoromethyl)-1H-pyrazole-5-carbonyl]piperidin-4-ol
4-[(3-methoxyphenyl)methyl]-1-{1-[3-(trifluoromethyl)phenyl]propan-2-yl}-1,4-diazepan-5-one
N-{2-[(1R,5S)-6,6-dimethylbicyclo[3.1.1]hept-2-en-2-yl]ethyl}-3-[2-(furan-2-ylmethyl)-5-oxopyrrolidin-2-yl]propanamide
N-({4-[4-(2-methoxyphenyl)piperazin-1-yl]quinazolin-2-yl}methyl)-2-(piperidin-1-yl)acetamide
(1S,5R)-3-(pyridin-2-ylmethyl)-6-(thiophene-2-sulfonyl)-3,6-diazabicyclo[3.2.2]nonane
2-(4-{[1-(5-chloropyridin-2-yl)-1H-pyrrol-2-yl]methyl}-2,3,4,5-tetrahydro-1,4-benzoxazepin-7-yl)-1-(dimethylamino)propan-2-ol
2-[1-(dimethyl-1,2-oxazole-4-carbonyl)piperidin-2-yl]-5-fluoro-1H-1,3-benzodiazole
2-cyclopropyl-9-(2-methoxy-5-methylbenzoyl)-2,9-diazaspiro[5.5]undecan-3-one