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ethyl 3-[(2-fluorophenyl)methyl]-1-(4-methyl-1,2,3-thiadiazole-5-carbonyl)piperidine-3-carboxylate
2-(4-{[3-(3-fluorophenyl)-1-(3-methylphenyl)-1H-pyrazol-4-yl]methyl}piperazin-1-yl)pyrimidine
1-benzyl-5-cyclobutyl-3-(oxan-4-yl)-1H-1,2,4-triazole
N-[(3-ethyl-1,2-oxazol-5-yl)methyl]-5-[3-(phenoxymethyl)-1,2,4-oxadiazol-5-yl]pyridin-2-amine
(2S,4S)-1-[(2-chlorophenyl)methyl]-4-[(1-ethylpiperidin-4-yl)amino]-N-(propan-2-yl)pyrrolidine-2-carboxamide
2-{4-[4-(3-methylpyridin-4-yl)-1,4-diazepan-1-yl]quinazolin-2-yl}ethan-1-amine
4-(1-butyl-1H-imidazol-2-yl)-1-[4-(trifluoromethyl)benzoyl]piperidine
2-{2-[2-(2-methyl-1H-imidazol-1-yl)ethyl]piperidine-1-carbonyl}-1H-indole
2-(6-methoxy-1,2,3,4-tetrahydronaphthalen-1-yl)-2,9-diazaspiro[5.5]undecan-3-one
1-(1H-indazol-5-yl)-4-{2-oxo-1-oxaspiro[4.4]nonane-4-carbonyl}piperazin-2-one
1-methyl-N-{[4-(5-methyl-1,2,4-oxadiazol-3-yl)phenyl]methyl}-6-propyl-1H-pyrazolo[3,4-d]pyrimidin-4-amine
2-[(cyclopropylmethyl)sulfanyl]-N-methyl-N-[(1-phenylpyrrolidin-3-yl)methyl]acetamide
1-(3,4-difluorophenyl)-3-(3-methoxypropyl)-3-(1-methylpiperidin-4-yl)urea
2-[4-(3-methoxy-5-methylthiophene-2-carbonyl)piperazin-1-yl]-4,6-dimethylpyrimidine
[(6-methoxy-2H-1,3-benzodioxol-5-yl)methyl](methyl)[2-(methylsulfanyl)ethyl]amine
7-{[1-(3-methoxyphenyl)-1H-pyrazol-4-yl]methyl}-2-oxa-7-azaspiro[4.5]decan-8-one
6-[3-(2H-1,3-benzodioxol-5-yl)propanoyl]-N-phenyl-6-azaspiro[2.5]octane-1-carboxamide
N,2,7,8-tetramethyl-N-[2-(4-methyl-1,3-thiazol-5-yl)ethyl]quinoline-4-carboxamide
N-ethyl-7,8-dimethyl-N-(pyridin-4-ylmethyl)-2-(pyrimidin-5-yl)quinoline-4-carboxamide
3,5-dimethyl-N-(3-methyl-1-{7-[(5-methylthiophen-2-yl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}butyl)benzamide
4-(but-2-ynoyl)-1-(4-methoxyphenyl)-6,6-dimethylpiperazin-2-one
1-methyl-4-[5-(propan-2-yl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-2-carbonyl]piperazin-2-one
1-[2-(3-fluorophenyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl]-2-(pyrrolidin-1-yl)propan-1-one
N-(3,5-dimethyl-1-propyl-1H-pyrazol-4-yl)-3-propoxypiperidine-1-carboxamide
2-(2,4-dimethoxyphenyl)-N-[(3R,4R)-3-hydroxypiperidin-4-yl]acetamide
5-[3-({5-phenyl-5H,6H,7H-pyrrolo[3,2-d]pyrimidin-2-yl}amino)propyl]-1,3,4-thiadiazol-2-amine
N-({2-[cyclohexyl(methyl)amino]pyridin-3-yl}methyl)-2-(2-methyl-6-oxo-1,6-dihydropyrimidin-5-yl)acetamide
1-[(3-fluorophenyl)methyl]-3-{[5-(2-methylpropyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl]methyl}urea
8-[(2-fluorophenyl)methyl]-1-oxa-8-azaspiro[4.6]undecan-9-one
2-{3-oxo-9-[(1R,2S)-2-propylcyclopropanecarbonyl]-2,9-diazaspiro[5.5]undecan-2-yl}acetamide
(3aS,6aS)-2-cyclopentyl-5-(2,3,4-trifluorobenzoyl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
4-ethyl-2-methyl-6-{3-[1-(1,3-thiazol-4-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}pyrimidine
[(2S)-1-[(3-phenyl-1,2,4-oxadiazol-5-yl)methyl]pyrrolidin-2-yl]methanol
4-[(2R,5S)-2,5-dimethylpyrrolidine-1-carbonyl]-1-{2-phenyl-5H,6H,7H-cyclopenta[d]pyrimidin-4-yl}piperidine
5-{4-[(3-fluorophenyl)methyl]piperazine-1-carbonyl}-4-propylpyrimidine
[4-(2-phenoxyethyl)-1-[(2,4,6-trimethoxyphenyl)methyl]piperidin-4-yl]methanol
1-{3-[(3R,4R)-3-hydroxy-3,4-dimethylpyrrolidine-1-carbonyl]phenyl}imidazolidin-2-one
1-{1'-[4-(trifluoromethyl)pyrimidin-2-yl]-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-5-yl}ethan-1-one
(1R,5R)-6-[(5-chloro-3-ethyl-1-methyl-1H-pyrazol-4-yl)methyl]-3-cyclobutanecarbonyl-3,6-diazabicyclo[3.2.2]nonane
(3S)-3-ethyl-4-(2-ethylpyridine-4-carbonyl)morpholine
1-{[2-(benzylamino)pyrimidin-5-yl]methyl}-3-phenylpyrrolidin-3-ol
4-benzyl-3-{1-[(1-ethyl-1H-1,2,4-triazol-5-yl)methyl]piperidin-4-yl}-4,5-dihydro-1H-1,2,4-triazol-5-one
4-(2-methyl-1-{4-[(2-methyl-1H-imidazol-1-yl)methyl]piperidin-1-yl}propan-2-yl)morpholine
2-[5-({2-[2-(1H-imidazol-1-yl)ethyl]piperidin-1-yl}methyl)furan-2-yl]benzonitrile
2-(2-methylphenyl)-5-{[1-(pyridin-2-yl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-2-yl]methyl}pyrimidine
(1S,5R)-6-(dimethyl-1,2-oxazole-4-carbonyl)-3-(pyrazin-2-yl)-3,6-diazabicyclo[3.2.2]nonane
3-(dimethyl-1,2-oxazol-4-yl)-1-(3-{[4-(hydroxymethyl)phenyl]methyl}pyrrolidin-1-yl)propan-1-one
{4-[({5-propylpyrazolo[1,5-a]pyrimidin-7-yl}amino)methyl]phenyl}methanol
N-[(3R,4S)-4-cyclopropyl-1-[(3-methoxyphenyl)methyl]pyrrolidin-3-yl]-3-methoxypropanamide
2-{4-[(2-fluoro-5-methoxyphenyl)methyl]-1-[1-(propan-2-yl)piperidin-4-yl]piperazin-2-yl}ethan-1-ol