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2-benzyl-8-{[3-(phenoxymethyl)-1,2,4-oxadiazol-5-yl]methyl}-2,8-diazaspiro[5.5]undecane
3-[(dimethylamino)methyl]-1-[(1-propyl-1H-imidazol-2-yl)methyl]pyrrolidin-3-ol
N-{5-[4-(2-hydroxyethyl)-1H-pyrazol-1-yl]pyridin-2-yl}cyclopropanecarboxamide
3-methoxy-5-methyl-N-[4-(pyrrolidin-1-yl)butyl]thiophene-2-carboxamide
methyl (2S)-3-methyl-2-{3-[5-(thiophen-3-yl)-1,3,4-oxadiazol-2-yl]propanamido}butanoate
N-{2-[(2-amino-5,6,7,8-tetrahydroquinazolin-4-yl)amino]ethyl}-N-methylmethanesulfonamide
ethyl 1-[(5-methylfuran-2-yl)methyl]-4-(2-phenoxyethyl)piperidine-4-carboxylate
2-cyclopentyl-2-phenyl-1-{4-[2-(1H-1,2,4-triazol-1-yl)ethyl]piperazin-1-yl}ethan-1-one
{[1-(2-methoxyethyl)piperidin-4-yl]methyl}({[5-(2-methylpropyl)-1H-pyrazol-3-yl]methyl})(pyridin-4-ylmethyl)amine
3-{5-[4-(3,5-dimethyl-1H-pyrazol-1-yl)butanoyl]-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}propanoic acid
2-[(1S,5R)-3-benzoyl-3,6-diazabicyclo[3.2.2]nonane-6-carbonyl]-5-methoxyphenol
4-{4-[4-ethyl-5-(pyrrolidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}-2-methylpyridine
(1S,6R)-9-[1-(2-phenylacetyl)piperidine-4-carbonyl]-3,9-diazabicyclo[4.2.1]nonan-4-one
2-(1-ethyl-3-oxopiperazin-2-yl)-N-(1,2,3,4-tetrahydronaphthalen-1-yl)acetamide
1-[(3-phenyloxolan-3-yl)methyl]-4-(pyrrolidin-1-ylmethyl)piperidin-4-ol
4-[4-(3-hydroxypiperidine-1-carbonyl)piperidin-1-yl]-2-(thiophen-2-ylmethyl)-2,3-dihydro-1H-isoindole-1,3-dione
1-methyl-N-[2-(4-methyl-1,3-thiazol-2-yl)ethyl]-6-propyl-1H-pyrazolo[3,4-d]pyrimidin-4-amine
{[5-methyl-2-(naphthalen-2-yl)-1,3-oxazol-4-yl]methyl}(prop-2-en-1-yl)(prop-2-yn-1-yl)amine
1-(2-{[(1-benzothiophen-2-ylmethyl)amino]methyl}phenoxy)-3-(thiomorpholin-4-yl)propan-2-ol
3-[3-hydroxy-3-(hydroxymethyl)piperidine-1-carbonyl]-4,5,6,7-tetrahydro-1-benzofuran-4-one
[4-({[2-amino-6-(cyclopropylamino)pyrimidin-4-yl](methyl)amino}methyl)oxan-4-yl]methanol
2-methoxy-N,N-dimethyl-5-({[2-(1H-1,2,3-triazol-5-ylsulfanyl)ethyl]carbamoyl}amino)benzamide
2-ethyl-9-(4-methylpyridine-3-carbonyl)-4-phenyl-2,9-diazaspiro[5.5]undecane
6-amino-1-[3-(diphenylmethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]hexan-1-one
N-[(1-{[4-(trifluoromethyl)phenyl]carbamoyl}piperidin-3-yl)methyl]pyridine-3-carboxamide
N-[(3S,7S,8aS)-3-(4-aminobutyl)-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-4-bromobenzamide
2-amino-4-(2-chloro-4-hydroxyphenyl)-6-(4-hydroxy-3-methoxyphenyl)pyridine-3-carbonitrile
2,4-difluoro-N-{5H,6H,7H,8H-imidazo[1,2-a]pyridin-3-yl}-3-methoxybenzamide
(2S,4R)-1-(furan-2-ylmethyl)-N-methyl-4-[2-(2-oxo-1,2-dihydropyridin-1-yl)acetamido]pyrrolidine-2-carboxamide
1-[(4-methylphenyl)methyl]-4-[3-(pyridin-4-yl)-1H-pyrazole-5-carbonyl]piperazin-2-one
(3S,4S)-4-(3-methoxyphenyl)-1-(thian-4-yl)piperidin-3-ol
(3aR,5S,6S,7aS)-2-[(4-chloro-1-methyl-1H-indazol-3-yl)methyl]-octahydro-1H-isoindole-5,6-diol
1-(2-oxo-2-{4-[1-(pyridin-4-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}ethyl)imidazolidine-2,4-dione
3-[5-(methoxymethyl)-3-methyl-1H-pyrazol-4-yl]-N,N-dimethylaniline
N-[cyclopropyl(1-ethyl-1H-1,2,4-triazol-5-yl)methyl]-3-(4-methyl-1,3-thiazol-5-yl)propanamide
N-{[7-(4-methanesulfonylphenyl)-2,3-dihydro-1-benzofuran-2-yl]methyl}-2-methylpropanamide
4-{4-[(2Z)-2-chloro-3-phenylprop-2-en-1-yl]piperazin-1-yl}-2-(2,3-dihydro-1,4-benzodioxin-2-ylmethyl)-2,3-dihydro-1H-isoindole-1,3-dione
6-(3-fluorophenyl)-N-methyl-N-[(trimethyl-1H-pyrazol-4-yl)methyl]imidazo[2,1-b][1,3]thiazole-3-carboxamide
3-(2H-1,3-benzodioxol-5-yl)-N-methyl-N-[2-(2-methyl-1H-imidazol-1-yl)ethyl]-3-phenylpropanamide
1-(2-chlorophenyl)-4-{[5-(1,5-dimethyl-1H-pyrrol-2-yl)-1,3,4-oxadiazol-2-yl]methyl}piperazin-2-one
1-methyl-4-{2-[4-(trifluoromethyl)phenyl]-1,3-thiazole-4-carbonyl}-1,4-diazepane
N-tert-butyl-2-{3'-oxo-3',4'-dihydro-1'H-spiro[piperidine-4,2'-quinoxaline]-1-yl}butanamide
2-(1-{2-methylpyrido[2,3-d]pyrimidin-4-yl}piperidin-4-yl)-1,3-benzoxazole
4-{[6-(5-fluoro-2-methylphenyl)pyridin-3-yl]methyl}morpholine
[1-(1-cyclopropanecarbonylpiperidin-4-yl)-3-(3-methoxypropyl)piperidin-3-yl]methanol
N,5-dimethyl-N-{[2-(methylamino)pyrimidin-5-yl]methyl}-4,5,6,7-tetrahydro-1-benzothiophene-2-carboxamide
4-oxo-N,N-bis(propan-2-yl)-2-(pyridin-3-yl)-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidine-7-carboxamide
2-(2,3-dimethoxy-5-methylphenyl)-5-(piperidin-1-ylmethyl)pyridine
N-[7,7-dimethyl-2-(morpholin-4-yl)-5,6,7,8-tetrahydroquinazolin-5-yl]-2,6-dioxo-1,2,3,6-tetrahydropyrimidine-4-carboxamide
5-chloro-N-cyclopentyl-N-{[4-methoxy-3-(propan-2-yloxy)phenyl]methyl}thiophene-2-sulfonamide