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2-[2-methyl-4-(2-methylphenyl)piperazin-1-yl]acetic acid
ethyl 1-[2-(2,4-dioxo-1,3-thiazolidin-3-yl)acetyl]-4-(3-phenylpropyl)piperidine-4-carboxylate
N-[2-(2-fluorophenyl)ethyl]-2-(oxan-3-yl)acetamide
2-[(6-{1-methyl-1H-pyrrolo[2,3-b]pyridin-4-yl}pyrimidin-4-yl)amino]ethan-1-ol
N-({1-[2-(4-chlorophenyl)ethyl]piperidin-3-yl}methyl)-3-methoxy-N-methylpropanamide
2-[1-(2,2-dimethylpropyl)-3-oxopiperazin-2-yl]-N-[(4-ethylphenyl)methyl]-N-methylacetamide
5-ethyl-2-{1-[(5-methyl-1,3,4-oxadiazol-2-yl)methyl]-4-phenyl-1H-imidazol-5-yl}pyridine
[(1S,9aR)-octahydro-1H-quinolizin-1-ylmethyl]({[4-(pyrrolidine-1-carbonyl)phenyl]methyl})amine
(3S,4R)-3-methoxy-1-(2-phenoxybenzoyl)piperidin-4-amine
N-(1-methoxypropan-2-yl)-2-methyl-7-(5-methyl-1,3-oxazole-4-carbonyl)-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
1-(2-amino-4-methylpyrimidine-5-carbonyl)-4-benzyl-3-ethyl-1,4-diazepan-5-one
(1R,3S)-3-[6-(methylsulfanyl)-1,2,3,4-tetrahydroisoquinoline-2-carbonyl]cyclopentane-1-carboxylic acid
1-{3-[(3,4-dimethylphenyl)amino]piperidin-1-yl}-2-(methylsulfanyl)ethan-1-one
1-[4-(2-methoxyphenoxy)piperidin-1-yl]-2-(morpholin-4-yl)butan-1-one
1-{[3-(1-benzofuran-2-yl)-1-benzyl-1H-pyrazol-4-yl]methyl}-4-methoxypiperidine
(1S,6R)-9-(quinolin-4-yl)-3,9-diazabicyclo[4.2.1]nonan-4-one
1-ethyl-4-({5-methyl-2-[3-(trifluoromethyl)phenyl]-1,3-oxazol-4-yl}methyl)piperazine
2-methoxy-5-{1-[1-phenyl-2-(1H-pyrazol-1-yl)ethyl]-1H-imidazol-2-yl}pyrimidine
1-(difluoromethyl)-N-(1-methylpiperidin-4-yl)-N-(2-phenylethyl)-1H-pyrazole-3-carboxamide
3-[2-(4-cyclopentylpiperazin-1-yl)-2-oxoethyl]-4-(2,2-dimethylpropyl)piperazin-2-one
2-{[3-({[1-(3-methoxypropyl)pyrrolidin-3-yl]methyl}carbamoyl)phenyl]amino}acetic acid
3-[4-(4-methoxybenzoyl)piperazine-1-carbonyl]-6-(propan-2-yl)-1,2-dihydropyridin-2-one
N-[2-(4-benzylpiperazin-1-yl)ethyl]-5-cyclopropyl-1,3,4-oxadiazol-2-amine
3-{2-oxo-2-[3-(pyridin-3-ylmethoxy)piperidin-1-yl]ethyl}-1,3-oxazolidin-2-one
methyl[2-(1-methyl-1H-pyrazol-4-yl)ethyl]{[5-(1H-pyrazol-3-yl)thiophen-2-yl]methyl}amine
5-fluoro-2-[(2-methoxyphenyl)methyl]-1-{1-[(1-methyl-1H-pyrazol-4-yl)methyl]piperidin-4-yl}-1H-1,3-benzodiazole
N-({7-[3-(3,4-dimethoxyphenyl)propanoyl]-3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl}methyl)-5-methylthiophene-2-carboxamide
(3S,5S)-1-benzyl-5-(pyrrolidine-1-carbonyl)piperidine-3-carboxylic acid
5-(1-{2-[5-fluoro-2-(1H-pyrazol-1-yl)phenyl]-1H-imidazol-1-yl}ethyl)-3-methyl-1,2,4-oxadiazole
N-ethyl-N-{[5-(2-methylpropyl)-1,2,4-oxadiazol-3-yl]methyl}-5H,6H,7H,8H-imidazo[1,2-a]pyrazine-2-carboxamide
1-cyclopentyl-4-[(1-methyl-1H-indol-5-yl)methyl]piperazin-2-one
1-{1-[(3-fluorophenyl)methyl]-5-oxopyrrolidin-3-yl}-3-(propan-2-yl)urea
4-{1-[(4-fluorophenyl)methyl]-1H,4H,5H,6H-pyrrolo[3,4-c]pyrazol-5-yl}-2-methoxypyridine-3-carbonitrile
4-(1-{[4-ethoxy-3-(hydroxymethyl)phenyl]methyl}piperidin-3-yl)benzoic acid
N-({1-[2-(azepan-1-yl)acetyl]piperidin-3-yl}methyl)thiophene-2-sulfonamide
N-(2-{[2-(pyridin-2-yl)pyrrolidin-1-yl]methyl}quinolin-6-yl)acetamide
N-{[2-(4-acetylpiperazin-1-yl)pyridin-3-yl]methyl}-5-propyl-1,2-oxazole-3-carboxamide
2-(4-{3-methyl-3H-[1,2,3]triazolo[4,5-b]pyridine-6-carbonyl}piperazin-1-yl)-1,3-benzothiazole
N-[2-methyl-1-(5-methyl-1H-1,3-benzodiazol-2-yl)propyl]-2-[3-oxo-1-(propan-2-yl)piperazin-2-yl]acetamide
(2R,3R,6R)-5-[(1-ethyl-1H-imidazol-5-yl)methyl]-3-(4-methoxyphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
1-ethyl-5-(1-ethyl-1H-pyrazole-4-carbonyl)-N-[(4-methoxyphenyl)methyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
N-[(3R,4S)-4-(propan-2-yl)-1-[2-(pyridin-2-yl)ethyl]pyrrolidin-3-yl]oxane-4-carboxamide
N'-(2,4-dimethylphenyl)-N-(3-hydroxy-3-methylbutyl)-N-methylethanediamide
4-{5-[2-(methylsulfanyl)benzoyl]-1-(pyridin-2-ylmethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carbonyl}morpholine
(1S,5R)-3-(1-acetylpiperidine-4-carbonyl)-6-benzyl-3,6-diazabicyclo[3.2.2]nonan-7-one
N-{[3-(pyridin-3-yl)-1,2,4-oxadiazol-5-yl]methyl}pyrimidin-4-amine
methyl[(1-methyl-1H-imidazol-5-yl)methyl]{[5-(propan-2-yl)-1,2,4-oxadiazol-3-yl]methyl}amine
2-(2,5-dioxoimidazolidin-1-yl)-N-{[4-(3-fluorophenyl)oxan-4-yl]methyl}acetamide
(1R,3S,5S)-8-{5-[(4H-1,2,4-triazol-3-ylsulfanyl)methyl]furan-2-carbonyl}-8-azabicyclo[3.2.1]octan-3-ol
1-{1-[(4-methylphenyl)amino]cyclopentanecarbonyl}piperidin-4-ol