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N-(1H-1,3-benzodiazol-2-yl)-2-[({8-methylimidazo[1,2-a]pyridin-3-yl}methyl)amino]acetamide
4-methyl-N-{[2-(2-methyl-1H-imidazol-1-yl)phenyl]methyl}-2-(propan-2-yl)-1,3-thiazole-5-carboxamide
2-[4-({5-[(4-methyl-4H-1,2,4-triazol-3-yl)sulfanyl]furan-2-yl}methyl)-1-(propan-2-yl)piperazin-2-yl]ethan-1-ol
N-[2-(2,5-dimethylphenoxy)ethyl]-N-methyl-2-[4-(5-methyl-1H-1,2,3,4-tetrazol-1-yl)phenyl]acetamide
3-[4-(2-amino-5-methylpyrimidin-4-yl)piperazin-1-yl]propan-1-ol
1-(4-{[(1,3-benzoxazol-2-ylmethyl)amino]methyl}-2-methoxyphenoxy)-3-[methyl(propan-2-yl)amino]propan-2-ol
4-({2-oxo-3-phenyl-1,8-diazaspiro[4.5]decan-8-yl}methyl)benzoic acid
2-(ethylamino)-N-[1-(4-fluorophenyl)-2-hydroxyethyl]pyrimidine-5-carboxamide
[4-(2-fluoro-5-methoxyphenyl)pyridin-2-yl]methanol
ethyl 1,5-bis[(4-methoxyphenyl)methyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylate
2-[1-(2-propyl-1,3-thiazole-4-carbonyl)piperidin-4-yl]-1,3-benzoxazole
2-[8-(cyclopropylmethyl)-9-oxo-2,8-diazaspiro[5.5]undecan-2-yl]-1,3-thiazole-4-carboxamide
3-benzyl-8-(2,2-dimethylpropyl)-1-(2-phenylethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
N-(4-chloro-2-fluorophenyl)-2-{[2-(4-hydroxyphenyl)ethyl]amino}acetamide
5-[4-(2-ethoxyphenyl)piperazine-1-carbonyl]-1-(propan-2-yl)piperidin-2-one
4-{[4-(4-methoxypyrimidin-2-yl)piperazin-1-yl]methyl}benzoic acid
2-methyl-N-(3-{4-[(4-phenyl-1,2,3,6-tetrahydropyridin-1-yl)methyl]phenoxy}propyl)-1,2,3,4-tetrahydroisoquinoline-3-carboxamide
2-(1,2,3,4-tetrahydroisoquinolin-2-yl)-N-{[2-(1H-1,2,4-triazol-1-yl)phenyl]methyl}propanamide
N5-{[1-(3-methoxyphenyl)-1H-pyrazol-4-yl]methyl}-N5,N6,N6-trimethyl-[1,2,5]oxadiazolo[3,4-b]pyrazine-5,6-diamine
3-(azepane-1-carbonyl)-1-ethyl-N-[2-(thiophen-2-yl)ethyl]-4,5,6,7-tetrahydro-1H-indazol-5-amine
(3aS,6aS)-2-[2-(dimethylamino)acetyl]-5-(5-methoxypyrimidin-2-yl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
1-({1-[(3-ethoxy-2-hydroxyphenyl)methyl]piperidin-3-yl}methyl)-N,N-diethyl-1H-1,2,3-triazole-4-carboxamide
2,6-dimethyl-4-({[2-(pyrrolidine-1-sulfonyl)ethyl]amino}methyl)phenyl acetate
N-[(1R,2S)-2-hydroxy-2,3-dihydro-1H-inden-1-yl]-2-phenylimidazo[1,2-a]pyridine-6-carboxamide
2-(2-{[1-(3-methoxyphenyl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-2-yl]methyl}-1H-pyrrol-1-yl)pyrimidine
1-{3-[2-(3-methoxyphenyl)ethyl]piperidin-1-yl}-2-methylpropan-1-one
4-chloro-1-methyl-N-[1-(3-methylpyridin-2-yl)propan-2-yl]-3-(trifluoromethyl)-1H-pyrazole-5-carboxamide
N-(1-{imidazo[1,2-a]pyrimidin-2-yl}propyl)-3-(1-methyl-1H-pyrrol-2-yl)-1H-pyrazole-5-carboxamide
4-chloro-3-({[1-(5-methyl-1H-1,2,4-triazol-3-yl)ethyl]carbamoyl}amino)-N-propylbenzamide
2-(adamantan-1-yl)-N-methyl-N-[(2-methylpyridin-4-yl)methyl]acetamide
6-{4-[3-(3,5-dimethylphenyl)propanoyl]piperazin-1-yl}pyridine-3-carbonitrile
1-(4-methylphenyl)-4-[5-(propan-2-yl)-1,2-oxazole-3-carbonyl]piperazin-2-one
1-[3-(4-chlorophenyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]but-3-en-1-one
1-methyl-3-{[1-(1,3-oxazole-5-carbonyl)piperidin-4-yl]methyl}-4-phenyl-4,5-dihydro-1H-1,2,4-triazol-5-one
2-ethyl-1-{[2-(4-methoxy-3-methylphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}piperidine
(3S,4S)-1-(6-fluoro-4-hydroxyquinoline-3-carbonyl)-4-methylpiperidine-3,4-diol
1-[3-(2-chlorophenoxy)azetidin-1-yl]-3-[methyl(1-methylpyrrolidin-3-yl)amino]propan-1-one
2-(1-{5-[(3,5-dimethyl-1H-pyrazol-1-yl)methyl]-1H-pyrazole-3-carbonyl}pyrrolidin-2-yl)pyridine
2-{4-[5-(propan-2-yl)pyrazolo[1,5-a]pyrimidin-7-yl]piperazin-1-yl}benzonitrile
3-({2-[(4aS,8aR)-decahydroisoquinolin-2-ylmethyl]-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-5-yl}methyl)benzonitrile
(3R,5S)-N3-(2,3-dihydro-1H-inden-5-yl)-1-[(3,4-dimethoxyphenyl)methyl]-N5-[(1-ethylpyrrolidin-2-yl)methyl]piperidine-3,5-dicarboxamide
5-[2-(3,3-diphenylpiperidin-1-yl)-2-oxoethyl]-2,6-dimethyl-3,4-dihydropyrimidin-4-one
[1-({methyl[(4-methyl-1H-imidazol-5-yl)methyl]amino}methyl)cyclopentyl]methanol
4-[3-(3-methoxyphenoxymethyl)piperidine-1-carbonyl]-1λ6-thiane-1,1-dione
2-{2-[(1R,3R,5S)-3-(4-fluoro-3-methylphenyl)-8-azabicyclo[3.2.1]octan-8-yl]-2-oxoethyl}-5,6-dimethyl-2,3-dihydropyridazin-3-one
N-{[2-(2,3-difluoro-4-methylphenoxy)pyridin-3-yl]methyl}-2-oxo-1,3-oxazolidine-4-carboxamide
N-(2-{1-[(1-ethyl-1H-pyrazol-4-yl)sulfonyl]piperidin-2-yl}ethyl)acetamide
(1S,5R)-3-[(4-fluoro-3-methoxyphenyl)methyl]-6-(3-methylbut-2-en-1-yl)-3,6-diazabicyclo[3.2.2]nonan-7-one
1-[9-methoxy-7-(6-methoxypyridin-2-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]-2-(3,4,5-trimethoxyphenyl)ethan-1-one
N4-{[1-(methoxymethyl)cyclopentyl]methyl}-5-methylpyrimidine-2,4-diamine