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8-(1,3-benzothiazol-2-ylmethyl)-1-(2-methoxyethyl)-3-(pyridin-3-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
5-[2-(4-fluorophenyl)azetidine-1-carbonyl]-2-(pyridin-2-yl)pyrimidin-4-ol
N-[(1R,2R)-2-acetamido-2,3-dihydro-1H-inden-1-yl]-1-(propan-2-yl)piperidine-4-carboxamide
3-{1-[2-(diphenylmethyl)-1H-imidazol-1-yl]ethyl}-4-methyl-4H-1,2,4-triazole
N-[2-(2-ethyl-1H-imidazol-1-yl)ethyl]-3-(pyrrolidin-3-yl)benzamide
(4aS,7aR)-1-(1-methylcyclopropanecarbonyl)-4-(pyridin-4-ylmethyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
N-[(2,2-dimethyl-2,3-dihydro-1-benzofuran-5-yl)methyl]-3-(4,5,6,7-tetrahydro-2H-indazol-3-yl)propanamide
2-(4-{[4-(1H-pyrazol-1-yl)butan-2-yl]amino}piperidin-1-yl)pyridine-3-carbonitrile
1-(1,3-benzothiazol-2-ylmethyl)-5-(2-{[(4-methoxyphenyl)methyl]amino}ethyl)pyrrolidin-2-one
(1R,5R)-6-(2,3-difluoro-4-methylbenzoyl)-N,N-dimethyl-3,6-diazabicyclo[3.2.2]nonane-3-carboxamide
N-methyl-N-[(3-methyl-1,2-oxazol-5-yl)methyl]-2-(3-phenylpropyl)-1,3-benzoxazole-5-carboxamide
6-[(2E)-3-(2,3-difluorophenyl)prop-2-enoyl]-N-(furan-2-ylmethyl)-6-azaspiro[2.5]octane-1-carboxamide
5-(methoxymethyl)-N-({5-[3-(trifluoromethoxy)phenyl]-2,3-dihydro-1-benzofuran-2-yl}methyl)furan-2-carboxamide
1-[4-(1-methyl-1H-pyrazol-4-yl)phenyl]-2-(morpholin-4-yl)ethan-1-ol
1-[6-(1-hydroxyethyl)pyridin-2-yl]-4-[3-(trifluoromethyl)phenyl]piperidin-4-ol
1-{[(1R,5S)-6,6-dimethylbicyclo[3.1.1]hept-2-en-2-yl]methyl}-N-[3-(1H-pyrazol-5-yl)phenyl]piperidine-4-carboxamide
ethyl 3-(2-phenylethyl)-1-[3-(1H-pyrazol-1-ylmethyl)benzoyl]piperidine-3-carboxylate
2-[3-({3-[methyl(2-phenylethyl)amino]piperidin-1-yl}methyl)phenoxy]ethan-1-ol
6-(3-chlorophenyl)-N-[(1-ethyl-5-oxopyrrolidin-3-yl)methyl]-N-methylimidazo[2,1-b][1,3]thiazole-3-carboxamide
(2S,4R)-N-ethyl-1-(naphthalen-1-ylmethyl)-4-({[2-(trifluoromethyl)phenyl]methyl}amino)pyrrolidine-2-carboxamide
3-(3-methoxypropyl)-1-[5-(propan-2-yl)thiophene-3-carbonyl]piperidine-3-carboxylic acid
4-{5-[3-(oxan-4-yl)-1H-1,2,4-triazol-5-yl]pyrimidin-2-yl}morpholine
1-[(2-methoxyphenyl)methyl]-6-oxo-N-[4-(pyridin-2-yl)butyl]piperidine-3-carboxamide
(2R,6R)-4-[2-(2-methyl-1,3-thiazol-4-yl)acetyl]-8-oxa-4-azatricyclo[7.4.0.02,6]trideca-1(13),9,11-triene-6-carboxylic acid
1-[2-({[2-(2-methyl-1H-imidazol-1-yl)phenyl]methyl}amino)pyrimidin-4-yl]piperidin-3-ol
{1-[(4-fluoro-3-methylphenyl)methyl]-3-(2-methoxyethyl)piperidin-3-yl}methanol
N-[2-(morpholin-4-yl)ethyl]-4-(4-{4H,5H,6H,7H-thieno[3,2-c]pyridin-5-yl}piperidin-1-yl)benzamide
4-phenyl-1-{5-[3-(trifluoromethyl)phenoxymethyl]-1,2-oxazole-3-carbonyl}piperidine
1-[(2-methyl-1,3-thiazol-5-yl)methyl]-N-[4-(2-methyl-1H-imidazol-1-yl)phenyl]piperidine-3-carboxamide
2-{3-[(4-fluoropiperidin-1-yl)methyl]phenyl}-6-(pyridin-4-yl)-3,4-dihydropyrimidin-4-one
N,3-dimethyl-N-[1-(2-phenylethyl)piperidin-3-yl]thiophene-2-carboxamide
4-{2-[4-(2-phenylpropyl)-1H-1,2,3-triazol-1-yl]ethyl}morpholine
3-[4-(1-benzothiophen-3-ylmethyl)piperazin-1-yl]-1λ6-thiolane-1,1-dione
(3S,4S)-1-[(5-tert-butyl-1H-pyrazol-3-yl)methyl]-4-(4,4-difluoropiperidin-1-yl)pyrrolidin-3-ol
N-{[1-(1H-imidazol-4-ylmethyl)piperidin-3-yl]methyl}-1-phenylmethanesulfonamide
3-cyano-5-fluoro-N-methyl-N-[(2-methyl-1,2,3,4-tetrahydroisoquinolin-3-yl)methyl]benzamide
2-(5-fluoro-2-methylphenyl)-N-[2-(1-oxo-1,2-dihydrophthalazin-2-yl)ethyl]acetamide
N-[(3R,4S)-1-(1H-imidazol-4-ylmethyl)-4-propylpyrrolidin-3-yl]-2-(2-oxopyrrolidin-1-yl)acetamide
4-{1-[1-(furan-3-ylmethyl)piperidin-4-yl]piperidine-4-carbonyl}morpholine
2-ethyl-6-[4-(2-methylphenyl)benzoyl]-5H,6H,7H-pyrrolo[3,4-d]pyrimidine
5-{2-methyl-4-oxo-3H,4H,5H,6H,7H,8H,9H-pyrimido[4,5-d]azepine-7-carbonyl}-2-phenyl-2,3-dihydro-1H-pyrazol-3-one
11-(4-hydroxy-3,5-dimethoxyphenyl)-4,6,10,12-tetraazatricyclo[7.3.0.03,7]dodeca-1,3(7),8,10-tetraen-5-one
4-(3-methyl-1H-1,2,4-triazol-5-yl)-1-[2-(methylsulfanyl)-1,3-thiazole-4-carbonyl]piperidine
1-(4-fluorophenyl)-N-(2-hydroxyethyl)-N-[(1-methyl-1H-imidazol-2-yl)methyl]cyclopropane-1-carboxamide
3-{2-[3-(propan-2-yl)-[1,2,4]triazolo[3,4-b][1,3,4]thiadiazol-6-yl]ethyl}pyridine
N,N-dimethyl-1-({5-methyl-2-[3-(trifluoromethyl)phenyl]-1,3-oxazol-4-yl}methyl)pyrrolidin-3-amine
N-[2-(3,4-dimethylphenoxy)ethyl]-6-(methoxymethyl)-1-methyl-1H-pyrazolo[3,4-d]pyrimidin-4-amine
N,2-dimethyl-6-(piperidin-3-yl)-N-(4,5,6,7-tetrahydro-1,2-benzoxazol-3-ylmethyl)pyrimidin-4-amine
3-(2,1,3-benzoxadiazol-5-ylmethyl)-1-[2-(2-ethoxyethoxy)phenyl]-3-methylurea
4-(3-cyclopropyl-1H-1,2,4-triazol-5-yl)-6-fluoro-1,2-dihydroquinolin-2-one