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N-[(3R,4S)-1-acetyl-4-phenylpyrrolidin-3-yl]-3-(azepan-1-yl)propanamide
2-methyl-5-(3-{[(6-methyl-2-propylpyrimidin-4-yl)amino]methyl}pyrrolidin-1-yl)-2,3-dihydropyridazin-3-one
3-hydroxy-1-(2-phenylethyl)-3-{[(1H-1,2,4-triazol-3-ylmethyl)amino]methyl}piperidin-2-one
4-chlorophenyl (7S,9aR)-7-benzyl-8-methyl-6,9-dioxo-octahydro-1H-pyrazino[1,2-a]piperazine-2-carboxylate
5-methyl-1-(4-methylphenyl)-4-[2-(trifluoromethyl)benzoyl]piperazin-2-one
1-[(4-fluorophenyl)methyl]-3-hydroxy-3-({methyl[(3-methyl-1,2-oxazol-5-yl)methyl]amino}methyl)piperidin-2-one
N-{[(3S,4S)-3-hydroxypiperidin-4-yl]methyl}-2-phenylacetamide
2-(cyclohex-1-en-1-yl)-1-{3-[5-(2-methylphenyl)-2-(pyridin-4-yl)pyrimidin-4-yl]piperidin-1-yl}ethan-1-one
(3R,5S)-1-benzyl-N3-(2,3-dihydro-1H-inden-5-yl)-N5-[(3,5-dimethylphenyl)methyl]piperidine-3,5-dicarboxamide
(4aR,7aS)-N,N-dimethyl-6,6-dioxo-4-[2-(2-oxo-1,2-dihydropyridin-1-yl)acetyl]-octahydro-6λ6-thieno[3,4-b]piperazine-1-carboxamide
1-[(5-cyano-1H-pyrrol-3-yl)methyl]-N-[3-(4-fluorophenyl)phenyl]piperidine-3-carboxamide
3-[(1R,5R)-6-(cyclopropylmethyl)-3,6-diazabicyclo[3.2.2]nonane-3-carbonyl]-4-phenyl-1H-pyrazol-5-amine
ethyl 4-oxo-5-phenoxy-1-{[3-(propan-2-yl)-4,5-dihydro-1,2-oxazol-5-yl]methyl}-1,4-dihydropyridine-3-carboxylate
2-{4-cyclopentyl-1-[(4-methoxy-2,3-dimethylphenyl)methyl]piperazin-2-yl}ethan-1-ol
3-(aminomethyl)-4-[(1R)-1-(4-fluorophenyl)ethyl]-4,5-dihydro-1H-1,2,4-triazol-5-one
1-{2-methylimidazo[1,2-a]pyrimidine-3-carbonyl}-4-[(3-methylphenyl)sulfanyl]piperidine
1-{4-[(3-methylphenyl)methyl]piperazin-1-yl}-3-(1H-pyrazol-1-yl)propan-1-one
N-[3-(1H-imidazol-1-yl)-1-phenylpropyl]-1-[4-(morpholine-4-carbonyl)phenyl]piperidin-4-amine
N-[2-({2,3-dimethyl-5-phenylpyrazolo[1,5-a]pyrimidin-7-yl}amino)ethyl]methanesulfonamide
2-[4-(2-methoxyphenyl)-3-oxopiperazine-1-carbonyl]pyrrolidine-1-carboxamide
3-(2-chlorophenyl)-N-methyl-N-[(4-methyl-1H-imidazol-2-yl)methyl]-3-phenylpropanamide
[(3R,4R)-4-(piperidin-1-ylmethyl)-1-[3-(propan-2-yl)-1H-pyrazole-5-carbonyl]pyrrolidin-3-yl]methanol
N-[1-(5-methyl-1-phenyl-1H-pyrazol-4-yl)ethyl]-3-(3-phenyl-1,2,4-oxadiazol-5-yl)propanamide
[(3R,4R)-1-(5-fluoro-2-methoxybenzoyl)-4-(pyrrolidin-1-ylmethyl)pyrrolidin-3-yl]methanol
2-(5-acetylthiophen-3-yl)-N-(1-methylpiperidin-4-yl)-N-(pyridin-4-ylmethyl)acetamide
N-{[5,8-dimethoxy-2-(morpholin-4-yl)quinolin-3-yl]methyl}-3-(3,5-dimethyl-1H-pyrazol-1-yl)-N-(furan-2-ylmethyl)propanamide
(3S,4S)-4-(dimethylamino)-1-({4-[2-(4-ethylpiperazin-1-yl)ethoxy]phenyl}methyl)pyrrolidin-3-ol
N-cyclohexyl-4-(1H-pyrazol-4-yl)-N-(pyridin-2-ylmethyl)butanamide
5-chloro-N-[(3R,5S)-5-(diethylcarbamoyl)-1-methylpyrrolidin-3-yl]-6-oxo-1,6-dihydropyridine-3-carboxamide
N-[(1R,3R)-3-aminocyclopentyl]-6-methoxy-4-oxo-1,4-dihydroquinoline-3-carboxamide
4-{2,7-diazaspiro[4.5]decane-7-carbonyl}-1,2-dihydroquinazolin-2-one
(1S,5R)-6-(3-methylbut-2-en-1-yl)-3-[3-(pyridin-3-yl)propanoyl]-3,6-diazabicyclo[3.2.2]nonan-7-one
N-butyl-N,5-dimethyl-4-[(oxolan-2-ylmethyl)amino]thieno[2,3-d]pyrimidine-6-carboxamide
1-{[2-cyclohexylmethanesulfonyl-1-(2-methoxyethyl)-1H-imidazol-5-yl]methyl}-2-(2-methoxyethyl)piperidine
(3S,4R)-N,N-dimethyl-1-(2-methyl-1,3-benzothiazole-5-carbonyl)-4-propylpyrrolidin-3-amine
2-(4-acetylpiperazin-1-yl)-2-(5-chloro-2-methoxyphenyl)acetic acid
ethyl 4-[3-(azepane-1-carbonyl)-1-methyl-4,5,6,7-tetrahydro-1H-indazol-5-yl]piperazine-1-carboxylate
propyl (1R,5S,6R)-6-{[(1,1-dioxo-1λ6-thian-4-yl)(methyl)amino]methyl}-3-azabicyclo[3.1.0]hexane-3-carboxylate
5-(3-methoxy-5-methylthiophen-2-yl)-3-(oxolan-3-yl)-1,2,4-oxadiazole
N-methyl-N-[(5-propylfuran-2-yl)methyl]thian-4-amine
3-{2-[(3-ethyl-1H-1,2,4-triazol-5-yl)sulfanyl]acetamido}-N-(1,3-thiazol-2-yl)propanamide
4-(3-cyclopropyl-1H-1,2,4-triazol-5-yl)pyridin-2-amine
N4-[(2-ethoxypyridin-3-yl)methyl]-6-(morpholin-4-yl)pyrimidine-2,4-diamine
N-(2,3-dihydro-1H-inden-2-yl)-2-[3-methyl-5-oxo-4-(2-phenylethyl)-4,5-dihydro-1H-1,2,4-triazol-1-yl]acetamide
2-methyl-9-[(3E)-pent-3-enoyl]-4-phenyl-2,9-diazaspiro[5.5]undecan-3-one
N-{[(2S,4S)-4-fluoropyrrolidin-2-yl]methyl}-5-methoxy-1H-indole-2-carboxamide
[(3R,4R)-1-[5-(methoxymethyl)thiophene-2-carbonyl]-4-(morpholin-4-ylmethyl)pyrrolidin-3-yl]methanol
methyl (2S,4R)-1-methyl-4-[(2E)-3-phenylprop-2-enamido]pyrrolidine-2-carboxylate
1-ethyl-3-(4-methyl-1,4-diazepane-1-carbonyl)-N-[(1-phenylcyclopentyl)methyl]-4,5,6,7-tetrahydro-1H-indazol-5-amine
(1R,5R)-3-benzoyl-6-(1H-imidazol-2-ylmethyl)-3,6-diazabicyclo[3.2.2]nonane