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6-[8-(2-methoxyethyl)-9-oxo-2,8-diazaspiro[5.5]undecan-2-yl]pyridine-3-carbonitrile
{4-[(4-chlorophenyl)methyl]-1-(quinolin-6-ylmethyl)piperidin-4-yl}methanol
6-{3-[2-methyl-4-(2-methylphenyl)piperazin-1-yl]-3-oxopropyl}-2,3-dihydropyridazin-3-one
1-[2-hydroxy-3-(4-methoxy-2-{[(1-phenylcyclopropyl)amino]methyl}phenoxy)propyl]piperidin-4-ol
1-{[1-benzyl-2-(ethanesulfonyl)-1H-imidazol-5-yl]methyl}-N,N-dimethylpyrrolidin-3-amine
(4aR,6R,8aS)-8a-(methoxymethyl)-2-[(3-methyl-1,2-oxazol-5-yl)methyl]-6-(morpholin-4-yl)-decahydroisoquinoline
5,6-dimethyl-N-[2-(4-methyl-1,3-thiazol-2-yl)ethyl]pyrimidin-4-amine
1-[3-(2-methylpropyl)-1,2-oxazole-5-carbonyl]-4-(3-phenylpropyl)-1,4-diazepane
5-(2-fluorophenoxymethyl)-N-[(4-methyl-1H-1,3-benzodiazol-2-yl)methyl]-1H-pyrazole-3-carboxamide
1-[(4-chlorophenyl)methyl]-N-{[1-(4-methoxyphenyl)cyclopentyl]methyl}-1H-1,2,3-triazole-4-carboxamide
ethyl 1-{[2-(dimethylamino)-1,3-thiazol-5-yl]methyl}-3-[(2-fluorophenyl)methyl]piperidine-3-carboxylate
N,N-bis(1,3-oxazol-4-ylmethyl)-2-oxo-6-phenyl-1,2-dihydropyridine-3-carboxamide
(3S,5S,9R)-5-{[(2-fluoro-5-methylphenyl)methyl]amino}-1,7-diazatricyclo[7.3.0.03,7]dodecane-2,8-dione
1-(5-methyl-1,3-oxazole-4-carbonyl)-4-{[4-(trifluoromethyl)phenyl]methyl}piperazine
N-[(5-{[2-(cyclopentyloxy)phenyl]methyl}-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl)methyl]acetamide
2,2-dimethylpropyl 8-[2-(1H-imidazol-4-yl)ethyl]-9-oxo-2,8-diazaspiro[5.5]undecane-2-carboxylate
2-{4-[5-(oxolan-2-yl)thiophene-2-carbonyl]piperazin-1-yl}pyridine-3-carbonitrile
4-{2-[(2R,3R,6R)-3-(4-fluorophenyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]-2-oxoethyl}piperazin-2-one
4,4,4-trifluoro-1-{3-[2-(3-fluorophenyl)ethyl]piperidin-1-yl}butan-1-one
(2R,6R)-4-(2,5-dimethylfuran-3-carbonyl)-10-methoxy-8-oxa-4-azatricyclo[7.4.0.02,6]trideca-1(13),9,11-triene-6-carboxylic acid
1-[4-(5-methyl-1,3,4-oxadiazol-2-yl)phenyl]-3-[1-(pyrazin-2-yl)piperidin-3-yl]urea
(3aS,6aS)-2-cyclopentyl-5-[6-(methoxymethyl)pyrimidin-4-yl]-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
2-[4-(6-methoxypyridazin-3-yl)-1H-pyrazol-1-yl]-N-[1-(thiophen-2-ylmethyl)-1H-pyrazol-5-yl]acetamide
4-[(2H-1,3-benzodioxol-5-ylmethyl)amino]-N-(2-hydroxybutyl)-5-methylthieno[2,3-d]pyrimidine-6-carboxamide
5-({5-cyclopropanecarbonyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-yl}carbonyl)-3,4-dihydropyrimidin-4-one
2-benzyl-N-{[2-(1H-imidazol-1-yl)phenyl]methyl}-1,3-thiazole-4-carboxamide
8-[(1,5-dimethyl-1H-pyrazol-4-yl)methyl]-2-(pyridin-3-ylmethyl)-2,8-diazaspiro[5.5]undecan-3-one
3-{1-[2-(3-chlorophenyl)acetyl]piperidin-3-yl}-N-methyl-N-(1-methylpiperidin-4-yl)propanamide
8-[(1,3-dimethyl-1H-pyrazol-4-yl)methyl]-1-(2-phenylethyl)-3-(pyridin-3-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
3-[(3R,4S)-4-(4-methylpiperazin-1-yl)-1-[2-(methylsulfanyl)-1,3-thiazole-4-carbonyl]piperidin-3-yl]propan-1-ol
N-{[4-(difluoromethoxy)phenyl]methyl}-1-(2-fluorophenyl)-4,5,6,7-tetrahydro-1H-indazol-4-amine
N2,N2,5,6-tetramethyl-N4-{[2-(pyrazin-2-yl)-1,3-thiazol-4-yl]methyl}pyrimidine-2,4-diamine
2-(5-methyl-2H-1,2,3,4-tetrazol-2-yl)-N-[1-methyl-3-(pyridin-2-yl)-1H-pyrazol-5-yl]acetamide
4-[4-(2-chlorophenyl)piperidin-4-yl]-2-(propan-2-yl)pyrimidine
(1R,3S,5S)-8-(furan-3-carbonyl)-3-(4-methoxyphenyl)-8-azabicyclo[3.2.1]octane
N1,N1,N3-trimethyl-N3-[3-(1-methyl-1H-pyrazol-4-yl)propyl]piperidine-1,3-dicarboxamide
1-[(3-fluorophenyl)methyl]-4-{[3-(pyridin-2-yl)phenyl]methyl}piperazine
6-[(6-ethoxyquinolin-2-yl)methyl]-2-(2-hydroxyethyl)-1H,2H,3H,4H,5H,6H,7H-pyrazolo[3,4-c]pyridin-3-one
1'-benzyl-5-methanesulfonyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
4-chloro-1-methyl-N-[(1-methylpiperidin-4-yl)methyl]-N-(2-phenylethyl)-1H-pyrrole-2-carboxamide
8-[6-(propan-2-yl)-2-(trifluoromethyl)pyrimidin-4-yl]-1-oxa-3,8-diazaspiro[4.6]undecan-2-one
4-{4-oxo-4H-pyrido[1,2-a]pyrimidine-3-amido}-N-phenylpiperidine-1-carboxamide
N-{[2-(4-fluorophenyl)-3-methyl-1H-indol-5-yl]methyl}-2,6-dioxo-1,2,3,6-tetrahydropyrimidine-4-carboxamide
(4aR,7aS)-1-benzyl-4-(2-methoxyacetyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
8-{[4-(3-hydroxy-3-methylbut-1-yn-1-yl)phenyl]methyl}-1-methyl-3-(propan-2-yl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
(2R,3R,6R)-3-(2H-1,3-benzodioxol-5-yl)-5-(1H-pyrazole-3-carbonyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
(2S,4R)-4-amino-1-(2,6-dichlorobenzoyl)-N-(propan-2-yl)pyrrolidine-2-carboxamide
1-(1-{5H,6H-benzo[h]quinazolin-2-yl}-5-methyl-1H-pyrazole-4-carbonyl)-4-(furan-2-carbonyl)piperazine
N-{2-cyclobutyl-7-[4-(2-fluorophenoxy)piperidine-1-carbonyl]-1-methyl-1H-1,3-benzodiazol-5-yl}-2-methoxyacetamide
6-{1-ethyl-1H,2H,3H,4H-pyrrolo[1,2-a]pyrazine-2-carbonyl}-1,3-benzothiazole