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7-(3-chlorophenyl)-4-(2,2-difluorocyclopropanecarbonyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
methyl({[1-(2-phenylethyl)-2-(propane-2-sulfonyl)-1H-imidazol-5-yl]methyl})(pyridin-2-ylmethyl)amine
2-[4-(1-ethyl-1H-imidazol-2-yl)piperidine-1-carbonyl]-3,4,7-trimethyl-1H-indole
N-{2H,4H,5H,6H-cyclopenta[c]pyrazol-3-ylmethyl}-N-methyl-5-(2-methylpropyl)-1,2-oxazole-3-carboxamide
3-{[(1R,3S,5S)-3-hydroxy-8-azabicyclo[3.2.1]octan-8-yl]methyl}-N-(2-methoxypyridin-3-yl)benzamide
4-(1-{imidazo[2,1-b][1,3]thiazole-6-carbonyl}pyrrolidin-2-yl)-3,5-dimethyl-1,2-oxazole
3-{2-[4-(methoxymethyl)piperidin-1-yl]-2-oxoethyl}-4-(naphthalen-1-ylmethyl)piperazin-2-one
N-[2-(azepane-1-carbonyl)phenyl]-2,2-dimethyl-4-oxo-3,4-dihydro-2H-pyran-6-carboxamide
N-methyl-N-(2-methylpropyl)-2-[3-(trifluoromethyl)phenoxymethyl]-1,3-oxazole-4-carboxamide
(4aS,7aR)-1-[(2-methyl-1,3-oxazol-4-yl)methyl]-4-(pyrimidin-2-yl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
2-(1,3-thiazol-2-yl)-1-(thiophen-3-ylmethyl)piperidine
2-(4-{[4-(furan-2-yl)phenyl]methyl}-1-(thiophen-2-ylmethyl)piperazin-2-yl)ethan-1-ol
6-{6-[(2-methoxyethyl)amino]-1H-pyrrolo[2,3-b]pyridin-4-yl}-3,4-dihydroquinazolin-4-one
2-(2,3-difluorophenoxymethyl)-N-[(5-methyl-1H-pyrazol-3-yl)methyl]-1,3-oxazole-4-carboxamide
4-{3-[2-(3-fluorophenyl)ethyl]piperidin-1-yl}pyrimidin-2-amine
8-methyl-3-{1-[3-(pyridin-3-yl)-1,2,4-oxadiazol-5-yl]ethyl}-3,4-dihydroquinazolin-4-one
1,2-dimethyl-3-[1-(pyridin-2-yl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indole-2-carbonyl]-1H-indol-5-ol
1-{2-[(1-methanesulfonylpiperidin-4-yl)amino]pyrimidin-4-yl}pyrrolidin-3-ol
methyl 1-[(3R,5S)-5-{[2-(3-chlorophenyl)ethyl]carbamoyl}-1-[(4-ethylphenyl)methyl]pyrrolidin-3-yl]-1H-1,2,3-triazole-4-carboxylate
methyl 3-(3-methylbenzamido)-6-(piperidin-1-ylmethyl)thieno[2,3-b]pyridine-2-carboxylate
2-[2-(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)ethyl]-2,9-diazaspiro[5.5]undecan-3-one
3-[1-(1-methyl-6-oxo-1,4,5,6-tetrahydropyridazine-3-carbonyl)piperidin-4-yl]-N-(3-methylphenyl)propanamide
N-benzyl-2-ethyl-N-[(3-methylpyridin-2-yl)methyl]pyrimidine-5-carboxamide
3-[(3aR,7aS)-2,3,3a,4,7,7a-hexahydro-1H-isoindol-2-yl]-N-[(4-fluorophenyl)methyl]propanamide
N-(furan-2-ylmethyl)-N-methyl-5-{[2-(propan-2-yl)-1H-imidazol-1-yl]methyl}-1H-pyrazole-3-carboxamide
4-[3-oxo-2-(pyridin-3-ylmethyl)-2,9-diazaspiro[5.5]undecane-9-carbonyl]oxane-4-carbonitrile
2-(benzyloxy)-N-(butan-2-yl)-N-(pyridin-3-ylmethyl)acetamide
N-(4-fluoro-2-methylphenyl)-3-{1-[3-(2-methylphenyl)propanoyl]piperidin-3-yl}propanamide
(4aR,7aS)-1-propanoyl-4-(quinoline-3-carbonyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
N-(6-methoxy-2H-1,3-benzodioxol-5-yl)-3-(pyrrolidine-1-carbonyl)piperidine-1-carboxamide
(1r,4r)-4-({[3-(2-chlorophenyl)-1-(4-methoxyphenyl)-1H-pyrazol-4-yl]methyl}amino)cyclohexan-1-ol
3-(8-methylquinolin-5-yl)-1-[(3R)-piperidin-3-yl]urea
N-{[5-(methoxymethyl)-1H-pyrazol-3-yl]methyl}-N,1,5-trimethyl-1H-indole-2-carboxamide
[4-(2-phenoxyethyl)-1-(1-phenoxypropan-2-yl)piperidin-4-yl]methanol
2-(pyridin-4-ylmethyl)-4-[3-(thiomorpholine-4-carbonyl)piperidin-1-yl]-2,3-dihydro-1H-isoindole-1,3-dione
(2S,4S)-N-{2-azatricyclo[9.4.0.03,8]pentadeca-1(11),3,5,7,12,14-hexaen-5-yl}-1-[(2-fluorophenyl)methyl]-4-(pyrimidin-2-ylsulfanyl)pyrrolidine-2-carboxamide
1-ethyl-5-methyl-4-[8-(trifluoromethyl)-[1,2,4]triazolo[4,3-a]pyridin-3-yl]-1H-pyrazole
(2R)-2-amino-2-cyclohexyl-1-(4-{1-[3-(dimethylamino)propyl]-1H-imidazol-2-yl}piperidin-1-yl)ethan-1-one
1-[(2-butyl-1H-imidazol-4-yl)methyl]-4-(1H-imidazol-1-yl)piperidine-4-carboxylic acid
1-{[3-(furan-2-yl)-1,2,4-oxadiazol-5-yl]methyl}-2-[2-(1-methyl-1H-imidazol-2-yl)ethyl]piperidine
(4aR,7aS)-1-[2-(2-chloro-6-fluoro-3-methylphenoxy)acetyl]-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
2-(3-cyclohexyl-5-oxo-4,5-dihydro-1H-1,2,4-triazol-4-yl)propanoic acid
1-{3-[2-(3-ethenylphenyl)-1H-imidazol-1-yl]phenyl}-5-methyl-1H-1,2,3,4-tetrazole
[(1-cyclopentylpiperidin-4-yl)methyl](furan-2-ylmethyl)(oxolan-2-ylmethyl)amine
3,3-dimethyl-1-[(5-{[(1s,4s)-4-aminocyclohexyl]methyl}-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl)methyl]urea
(3aR,7aS)-5-methyl-2-[2-(4H-1,2,4-triazol-4-yl)pyridine-4-carbonyl]-2,3,3a,4,7,7a-hexahydro-1H-isoindole
8-(3-fluoropyridin-4-yl)-2-(3-methoxypropyl)-2,8-diazaspiro[5.5]undecan-3-one
9-[(2-ethylpyrimidin-4-yl)methyl]-1-oxa-9-azaspiro[5.5]undecan-5-ol
1-{1-[(6-methylpyridin-2-yl)methyl]piperidin-3-yl}-4-[3-(trifluoromethyl)phenyl]piperazine
N-[(3-ethyl-1,2-oxazol-5-yl)methyl]-2-{3-oxo-1-[(3-phenoxyphenyl)methyl]piperazin-2-yl}acetamide