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3-(3-fluorophenyl)-N-(2-oxooxolan-3-yl)benzamide
1-cyclopentyl-5-oxo-N-[2-(1-oxo-1,2-dihydrophthalazin-2-yl)ethyl]pyrrolidine-3-carboxamide
8-(3-cyclopropylpropanoyl)-3-(3-methylbutyl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
7-[(2,3-difluorophenyl)methyl]-6-oxo-N-(propan-2-yl)-2,7-diazaspiro[4.5]decane-2-carboxamide
2-amino-4-{[2-(dimethylamino)ethyl]amino}-N,N-dimethyl-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepine-7-sulfonamide
3-benzyl-8-methyl-1-(2-phenylethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
N-[(2,3-dimethyl-1H-indol-5-yl)methyl]-6-(morpholin-4-yl)pyrimidin-4-amine
2-(benzenesulfonamidomethyl)-N,N-dimethyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-5-carboxamide
N-({5-cyclobutanecarbonyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)pyrrolidine-1-carboxamide
1-{[3-(3-methoxyphenyl)-1,2,4-oxadiazol-5-yl]methyl}-1H-indazole
N3-(2-methylpropyl)-4-oxo-1-(propan-2-yl)-N5-(thiophen-2-ylmethyl)-1,4-dihydropyridine-3,5-dicarboxamide
2-(2-ethyl-4-methyl-6-oxo-1,6-dihydropyrimidin-5-yl)-N-[(3-phenyl-1H-1,2,4-triazol-5-yl)methyl]acetamide
N-methyl-3-[5-(morpholin-4-ylmethyl)-1H-1,2,3,4-tetrazol-1-yl]-N-{[1-(propan-2-yl)pyrrolidin-3-yl]methyl}propanamide
2-[2-(1H-imidazol-4-yl)ethyl]-9-[2-(3-methyl-1H-1,2,4-triazol-5-yl)acetyl]-2,9-diazaspiro[5.5]undecan-3-one
3-(4-methoxypyrimidin-2-yl)-5-methyl-1H-indole
2-{imidazo[2,1-b][1,3]thiazol-6-yl}-1-[3-(pyridin-4-yl)azetidin-1-yl]ethan-1-one
1-[1,3-dioxo-2-(thiophen-2-ylmethyl)-2,3-dihydro-1H-isoindol-4-yl]-N,N-dimethylpiperidine-4-carboxamide
5-{4-[4-ethyl-5-(1H-imidazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidine-1-carbonyl}-4-methylpyrimidine
4-(4-{1H-naphtho[2,3-d]imidazol-2-yl}-1H-1,2,3-triazol-1-yl)piperidine
3-(2,3-dihydro-1H-inden-4-yl)-1-[2-(4,6-dimethyl-2-oxo-1,2-dihydropyrimidin-1-yl)ethyl]urea
3-[5-(1-benzofuran-2-yl)-4-phenyl-1H-imidazol-1-yl]propan-1-ol
3-[(4-methoxyphenyl)methyl]-1-methyl-8-[(3-methylquinoxalin-2-yl)methyl]-1,3,8-triazaspiro[4.5]decane-2,4-dione
4-chloro-1-ethyl-N-[(2-fluorophenyl)methyl]-N-(1-methoxypropan-2-yl)-1H-pyrazole-3-carboxamide
3-(1-ethyl-1H-imidazol-2-yl)-1-[2-methyl-5-(trifluoromethyl)benzoyl]piperidine
8-(5-chloropyridin-2-yl)-2-[(dimethyl-1,2-oxazol-4-yl)methyl]-2,8-diazaspiro[4.5]decan-3-one
3-(azepan-1-ylmethyl)-3-hydroxy-1-[(3-methylphenyl)methyl]piperidin-2-one
4-hydroxy-N-{[4-(2-methoxyethyl)-4H-1,2,4-triazol-3-yl]methyl}-2-(2-methyl-1,3-thiazol-4-yl)pyrimidine-5-carboxamide
1-(4-{[3-(2-phenylethyl)-1H-1,2,4-triazol-5-yl]methyl}phenyl)-1H-1,2,3,4-tetrazole
N-[(2,3-dimethoxyphenyl)methyl]-2,3,5,6-tetramethylbenzamide
(1-{4-[4-({[3-(trifluoromethyl)phenyl]methyl}amino)piperidin-1-yl]benzoyl}piperidin-3-yl)methanol
1-[2-chloro-5-(morpholin-4-yl)phenyl]-3-[2-(1H-1,2,4-triazol-5-ylsulfanyl)ethyl]urea
3-{2-[4-(5-chloropyridin-2-yl)piperazin-1-yl]-2-oxoethyl}-4-(2-methylpropyl)piperazin-2-one
6-ethyl-1,5-dimethyl-N-[2-(1-methylpiperidin-3-yl)ethyl]-2-oxo-1,2-dihydropyridine-3-carboxamide
N-methyl-N-phenyl-2-{3-[3-(pyrimidin-5-yl)phenyl]-1H-pyrazol-1-yl}acetamide
4-[(5-cyclopropyl-1,3,4-oxadiazol-2-yl)methyl]-2-(trifluoromethyl)morpholine
4-(1-{1-[(3,5-dimethyl-1H-pyrazol-4-yl)methyl]piperidin-4-yl}piperidine-3-carbonyl)morpholine
2-{2-[(1R,5S,8R)-8-methoxy-3-azabicyclo[3.2.1]octan-3-yl]-2-oxoethyl}-2,3-dihydro-1,2-benzothiazol-3-one
(2R,3R)-3-({[4-(2-methoxyethyl)-4H-1,2,4-triazol-3-yl]methyl}(methyl)amino)-2,3-dihydrospiro[indene-1,4'-piperidine]-2-ol
6-fluoro-2-{[4-(piperidine-1-carbonyl)piperidin-1-yl]methyl}quinolin-4-ol
4-[(1E)-3-{3-benzyl-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-7-yl}prop-1-en-1-yl]-N,N-dimethylaniline
4-{4-[(1-acetyl-1H-indol-3-yl)methyl]piperazin-1-yl}-2-(thiophen-3-ylmethyl)-2,3-dihydro-1H-isoindole-1,3-dione
2-(4-methoxy-2-methylphenyl)-2-[4-(pyridin-2-yl)piperazin-1-yl]acetic acid
1-{4-[(4-{[4-(1-hydroxyethyl)-1H-1,2,3-triazol-1-yl]methyl}piperidin-1-yl)methyl]thiophen-2-yl}ethan-1-one
1-{[6-(dimethylamino)pyridin-3-yl]methyl}-4-(4-fluorophenyl)piperidin-4-ol
N-cyclooctyl-3-{[1-(1-methylpiperidin-4-yl)piperidin-4-yl]oxy}benzamide
2-amino-N-{1H,4H,5H,6H-cyclopenta[c]pyrazol-3-ylmethyl}-3-ethyl-3H-imidazo[4,5-b]pyridine-6-carboxamide
3-methyl-8-(2,3,4-trimethoxyphenyl)-2H,3H,5H,6H,7H,8H-[1,3]oxazolo[5,4-g]quinoline-2,6-dione
5-[(2H-1,3-benzodioxol-5-yloxy)methyl]-N-methyl-N-[1-(1,2-oxazol-3-yl)ethyl]-1H-pyrazole-3-carboxamide
1-tert-butyl-N-[2-(1-methyl-1H-1,2,4-triazol-5-yl)ethyl]-5-oxopyrrolidine-3-carboxamide
2-methyl-3-[1-(3-methylphenyl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indole-2-carbonyl]pyridine