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5-{[(3aS,6aS)-1-[(2-fluorophenyl)methyl]-octahydropyrrolo[3,4-b]pyrrol-5-yl]methyl}-1H-indole
N-[(2,6-difluorophenyl)methyl]-1-[4-(2,5-dimethylthiophen-3-yl)pyrimidin-2-yl]-5-(methoxymethyl)-1H-pyrazole-4-carboxamide
4-[4-(2-aminopropan-2-yl)-1H-1,2,3-triazol-1-yl]-N-(2H-1,3-benzodioxol-5-yl)piperidine-1-carboxamide
N-[2-(5-methyl-1,3,4-thiadiazol-2-yl)ethyl]-2-(pyridin-3-yl)acetamide
2-(2-chlorophenyl)-2-[3-(4-methyl-1,3-thiazol-5-yl)propanamido]acetic acid
methyl N-({1-[(3R,5S)-5-(ethylcarbamoyl)pyrrolidin-3-yl]-1H-1,2,3-triazol-4-yl}methyl)-N-methylcarbamate
N-({5-[(2-chloroprop-2-en-1-yl)sulfanyl]-4-(4-methoxyphenyl)-4H-1,2,4-triazol-3-yl}methyl)thiophene-2-sulfonamide
4-({2-[1-(2-methyl-1,3-thiazole-4-carbonyl)piperidin-4-yl]-1H-imidazol-1-yl}methyl)pyridine
4-methanesulfonyl-N-(2,3,4,5-tetrahydro-1-benzoxepin-4-ylmethyl)benzamide
4-[4-hydroxy-4-(pyridin-3-yl)piperidine-1-carbonyl]benzene-1-sulfonamide
7-[3-(hydroxymethyl)-3-(2-methoxyethyl)piperidine-1-carbonyl]-1,2,3,4-tetrahydroquinoxalin-2-one
6-methyl-N-[(1-methyl-1H-pyrazol-4-yl)methyl]-10-oxa-5,7-diazatricyclo[9.4.0.03,8]pentadeca-1(11),3,5,7,12,14-hexaen-4-amine
(4aR,8aS)-1-(pyridin-3-ylmethyl)-6-(thiophene-2-carbonyl)-decahydro-1,6-naphthyridin-2-one
1-[2-(5-fluoro-1H-1,3-benzodiazol-2-yl)piperidin-1-yl]-2-(1H-1,2,4-triazol-1-yl)ethan-1-one
N-butyl-1-cyclohexyl-5-[3-(diethylamino)pyrrolidine-1-carbonyl]-4-oxo-1,4-dihydropyridine-3-carboxamide
3-fluoro-5-methyl-N-(1,2-oxazol-3-ylmethyl)imidazo[1,2-a]pyridine-2-carboxamide
ethyl 1-(pyridin-2-ylmethyl)-5-(4,4,4-trifluorobutan-2-yl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylate
6-{6-[(piperidin-4-yl)amino]-1H-pyrrolo[2,3-b]pyridin-4-yl}pyridine-3-carboxylic acid
5-fluoro-2-{4-[3-(pyrrolidine-1-carbonyl)piperidin-1-yl]piperidin-1-yl}pyrimidine
N-[(4-methanesulfonylmorpholin-2-yl)methyl]-7-(propan-2-yl)-[1,2,4]triazolo[1,5-a]pyrimidine-5-carboxamide
(2-ethoxy-5-{[({1-[(2-fluorophenyl)methyl]piperidin-4-yl}methyl)(2-methoxyethyl)amino]methyl}phenyl)methanol
3-methoxy-5-{methyl[1-(methylcarbamoyl)propan-2-yl]carbamoyl}benzoic acid
(2S,4S)-4-amino-N-ethyl-1-[4-(hydroxymethyl)benzoyl]pyrrolidine-2-carboxamide
N-(2,3-dihydro-1,4-benzodioxin-2-ylmethyl)-2-(2-phenyl-1H-imidazol-1-yl)acetamide
8-[2-(2-chlorophenoxy)acetyl]-1-methyl-2-oxo-1,8-diazaspiro[4.5]decane-4-carboxylic acid
N-(1-{1-[(2-chlorophenyl)methyl]piperidin-4-yl}-1H-pyrazol-5-yl)-2H-1,3-benzodioxole-5-carboxamide
2-{1-[4-(2,5-dimethylthiophen-3-yl)pyrimidin-2-yl]-5-methyl-1H-pyrazole-4-carbonyl}-2-azabicyclo[2.2.1]heptane
2-(2-fluoro-5-methoxyphenyl)-5-methyl-4-{octahydropyrrolo[1,2-a]piperazin-2-ylmethyl}-1,3-oxazole
7-[3-chloro-5-(trifluoromethyl)pyridin-2-yl]-4-[(2-fluoro-4-methoxyphenyl)methyl]-9-methoxy-2,3,4,5-tetrahydro-1,4-benzoxazepine
N,2-dimethyl-N-[(1-methyl-1H-1,3-benzodiazol-2-yl)methyl]-2-(thiophen-2-ylformamido)propanamide
(2S,4S)-N-ethyl-4-{[(3-phenoxyphenyl)methyl]amino}-1-(propan-2-yl)pyrrolidine-2-carboxamide
N-[2-(hydroxymethyl)-6-methylphenyl]-4-{[methyl(2-methylprop-2-en-1-yl)amino]methyl}benzamide
N-methyl-2-[3-oxo-1-(piperidin-4-yl)piperazin-2-yl]acetamide
1-[2-({[1-(pyridin-2-ylmethyl)piperidin-4-yl]amino}methyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-5-yl]ethan-1-one
4-{[3-(3-methoxyphenyl)-1,2-oxazol-5-yl]methyl}-1-[3-(methylsulfanyl)propyl]piperidin-4-ol
4-{6-cyclopentyl-1-methyl-1H-pyrazolo[3,4-d]pyrimidin-4-yl}-2-(trifluoromethyl)morpholine
6-ethyl-2-(3-{[(furan-2-ylmethyl)(methyl)amino]methyl}phenyl)-3,4-dihydropyrimidin-4-one
({5,7-dimethylpyrazolo[1,5-a]pyrimidin-3-yl}methyl)(methyl)[1-(pyridin-2-yl)ethyl]amine
5-[4-(3-hydroxypiperidin-1-yl)pyrimidin-2-yl]thiophene-2-carboxylic acid
N-(2-{7-[2-(2H-1,3-benzodioxol-5-ylmethyl)propyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}ethyl)-2-(4-fluorophenyl)acetamide
4-(piperidin-3-yl)-N-{[3-(pyridin-4-yl)-1H-1,2,4-triazol-5-yl]methyl}benzamide
1-(3-methoxyphenyl)-4-[4-(2-methylphenyl)benzoyl]piperazin-2-one
4-cyclobutaneamido-N-ethyl-N-[(1-ethyl-1H-pyrazol-4-yl)methyl]benzamide
1-{[1-benzyl-2-(ethanesulfonyl)-1H-imidazol-5-yl]methyl}-3-(pyrrolidin-1-ylmethyl)piperidine
5-oxo-N-[2-(2-oxo-1,3-oxazolidin-3-yl)ethyl]-1-[4-(propan-2-yl)phenyl]pyrrolidine-3-carboxamide
2-(cyclopropylmethyl)-8-[2-(3-fluorophenoxy)acetyl]-2,8-diazaspiro[5.5]undecan-3-one
N-(5-fluoro-2-oxo-2,3-dihydro-1H-indol-3-yl)-4-sulfamoylbutanamide
N-{[1-(3-acetamidopropanoyl)piperidin-3-yl]methyl}-4-phenylbenzamide
1-(2-hydroxyethyl)-5-[1-(4-methylphenyl)cyclopropanecarbonyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylic acid
methyl({[1-(2-phenylethyl)-2-(propane-2-sulfonyl)-1H-imidazol-5-yl]methyl})(pyrazin-2-ylmethyl)amine