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4-({[(5-fluoro-1H-indol-2-yl)methyl](methyl)amino}methyl)-1H-pyrazole-3-carboxylic acid
N-[2-(3,5-dimethyl-1H-pyrazol-1-yl)ethyl]-N-methyl-1-[2-(morpholin-4-yl)ethyl]-6-oxopiperidine-3-carboxamide
1-methyl-N-[3-(2-propoxyphenyl)propyl]piperidine-2-carboxamide
7-{[(2R,6S)-2,6-dimethylmorpholin-4-yl]methyl}-4-[3-(5-methylthiophen-2-yl)-1H-pyrazole-5-carbonyl]-2,3,4,5-tetrahydro-1,4-benzoxazepine
4-chloro-3-{2-[2-(1H-pyrazol-1-yl)ethyl]piperidine-1-carbonyl}-1H-pyrazol-5-amine
1-{thieno[3,2-d]pyrimidin-4-yl}-N-[3-(1H-1,2,3-triazol-1-yl)propyl]piperidin-4-amine
3-(5-oxo-1-propylpyrrolidin-3-yl)-1-{3-[(trifluoromethyl)sulfanyl]phenyl}urea
1-[2-(1H-pyrazol-1-yl)benzoyl]-4-(thian-4-yl)piperazine
4-acetyl-N-{3-[(2-methoxyethyl)carbamoyl]-2-methylphenyl}piperazine-1-carboxamide
2-oxo-N-[2-(pyridin-3-yl)ethyl]-1-[(1r,4r)-4-hydroxycyclohexyl]-2,3-dihydro-1H-1,3-benzodiazole-5-carboxamide
3-(oxan-4-yl)-1-(4-{[2-(pyridin-2-yl)ethyl]sulfanyl}phenyl)urea
{[(1R,5S,6S)-3-[(2-ethylpyrimidin-4-yl)methyl]-3-azabicyclo[3.1.0]hexan-6-yl]methyl}dimethylamine
6-cyclopentyl-1-methyl-N-[2-(piperidin-2-yl)ethyl]-1H-pyrazolo[3,4-d]pyrimidin-4-amine
(1R,5S)-3-{[5-(2-methylpropyl)thiophen-2-yl]methyl}-3,6-diazabicyclo[3.2.2]nonan-7-one
2-acetamido-N-ethyl-N-{[3-(methoxymethyl)-1,2,4-oxadiazol-5-yl]methyl}-3-methylbutanamide
(2S,4S)-N-ethyl-4-[2-(pyridin-2-yl)acetamido]-1-(thiophen-2-ylmethyl)pyrrolidine-2-carboxamide
2,5-dioxo-6-[2-(pyrrolidine-1-sulfonyl)ethyl]-1,2,5,6-tetrahydro-1,6-naphthyridine-3-carbonitrile
(2S,4R)-4-amino-N-(propan-2-yl)-1-{4H,5H,6H,7H-pyrazolo[1,5-a]pyridine-3-carbonyl}pyrrolidine-2-carboxamide
N-(2-methoxyethyl)-N-[(1-methyl-1H-pyrazol-4-yl)methyl]-2-(methylsulfanyl)pyridine-3-carboxamide
N-[(5-ethylpyridin-2-yl)methyl]-N-methyl-2,8-diazaspiro[4.5]decane-3-carboxamide
3-chloro-4-fluoro-N-{[7-fluoro-5-(pyridin-3-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}benzamide
N-benzyl-6-methyl-N-[(4-methyl-1,3-thiazol-5-yl)methyl]-2-oxo-1,2-dihydropyridine-3-carboxamide
2-(4-fluorophenoxy)-1-[(3R,4R)-3-(hydroxymethyl)-4-[(4-methylpiperazin-1-yl)methyl]pyrrolidin-1-yl]ethan-1-one
N-{1-[1-(3-aminopropanoyl)piperidin-4-yl]-1H-pyrazol-5-yl}-3-fluorobenzamide
(3R,4R)-3-cyclopropyl-4-methyl-1-{4-methyl-6H,7H,8H-cyclopenta[g]quinolin-2-yl}pyrrolidin-3-ol
1-[(2S,6S)-6-(hydroxymethyl)-8-oxa-4-azatricyclo[7.4.0.02,6]trideca-1(13),9,11-trien-4-yl]-5-phenylpentane-1,5-dione
N-(2,3-dihydro-1H-inden-5-yl)-4-(2-methoxyacetyl)-1,4-diazepane-1-carboxamide
1-(furan-2-ylmethyl)-N-(5-oxo-1-phenylpyrrolidin-3-yl)piperidine-4-carboxamide
4-(6-methylpyridazin-3-yl)-N-[3-(propan-2-yl)phenyl]morpholine-2-carboxamide
6-{3-[1-(cyclobutylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}-9H-purine
5-chloro-3-ethyl-4-{[3-(2-fluorophenoxy)azetidin-1-yl]methyl}-1-methyl-1H-pyrazole
(3S,9aR)-8-{[1-(2-methoxyphenyl)-1H-pyrazol-4-yl]methyl}-3-(propan-2-yl)-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
N-{2-[5-(oxolan-2-yl)-1,2,4-oxadiazol-3-yl]ethyl}-1-(propan-2-yl)piperidine-4-carboxamide
6-(4-{2-[(1-benzylpyrrolidin-3-yl)carbamoyl]ethyl}piperidin-1-yl)pyridine-3-carboxamide
2-{1-[(2-chlorophenyl)methyl]-1H-1,2,3-triazole-4-carbonyl}-1,2-oxazinane
2-hydroxy-3-methoxy-N-methyl-N-{[3-(1H-pyrazol-1-yl)phenyl]methyl}benzamide
N-(6-methoxypyridin-3-yl)-4-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]piperazine-1-carboxamide
2-[(2-butyl-1H-imidazol-4-yl)methyl]-7-cyclohexyl-2,7-diazaspiro[4.5]decan-6-one
(3S,4R)-1-(5-chloro-6-oxo-1,6-dihydropyridine-3-carbonyl)-4-phenylpyrrolidine-3-carboxylic acid
9-methoxy-7-(4-methoxyphenyl)-4-[(5-methylthiophen-2-yl)methyl]-2,3,4,5-tetrahydro-1,4-benzoxazepine
1-(5,6-dimethylpyrimidin-4-yl)-4-(2-fluorophenoxy)piperidine-4-carboxylic acid
1-{[3-(2H-1,3-benzodioxol-5-yl)-1,2,4-oxadiazol-5-yl]methyl}-N,N-diethylpiperidine-3-carboxamide
6-methyl-9-[3-(propan-2-yloxy)phenyl]-9H-purine
1-[(4-chlorophenyl)methyl]-N-[1-(2-methyl-1,3-thiazol-4-yl)ethyl]-1H-1,2,3-triazole-4-carboxamide
methyl 4-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-ylmethyl}piperazine-1-carboxylate
N-cyclopentyl-N-[(2-methoxyphenyl)methyl]-2-(1H-1,2,4-triazol-3-yl)benzamide
3-(1-ethyl-1H-1,2,3-triazol-4-yl)-1-{[1-methyl-2-(methylsulfanyl)-1H-imidazol-5-yl]methyl}urea
(1S,5R)-3-{[3-(furan-2-yl)phenyl]methyl}-6-(2-methoxyethyl)-3,6-diazabicyclo[3.2.2]nonane
2-[2-(dimethylamino)-2-(2-methylphenyl)ethyl]-2,9-diazaspiro[5.5]undecan-3-one
2-[(3,4-difluorophenyl)methyl]-8-(3-methylpyrazin-2-yl)-2,8-diazaspiro[4.5]decan-3-one