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2-(4-{[3-(benzyloxy)phenyl]methyl}morpholin-2-yl)ethan-1-amine
N-{[4-(4-fluorophenyl)-5-(methylsulfanyl)-4H-1,2,4-triazol-3-yl]methyl}-3-(4-methylphenyl)propanamide
(2S,4S)-N-ethyl-4-(2-methylfuran-3-amido)-1-(oxan-4-yl)pyrrolidine-2-carboxamide
(2,1,3-benzoxadiazol-5-ylmethyl)[1-(2-methoxyphenyl)propan-2-yl]amine
3-(propan-2-yl)-1-[(1-{[5-(1H-pyrazol-3-yl)furan-2-yl]methyl}pyrrolidin-3-yl)methyl]urea
N-(3-aminopropyl)-2-[(2,6-dichlorophenyl)methyl]-4-hydroxypyrimidine-5-carboxamide
1-{3-[(1S,5R)-3-(pyridine-3-carbonyl)-3,6-diazabicyclo[3.2.2]nonane-6-carbonyl]phenyl}ethan-1-one
methyl({4-methyl-5-[(2-phenoxyethyl)sulfanyl]-4H-1,2,4-triazol-3-yl}methyl)(quinolin-6-ylmethyl)amine
(2R,6R)-4-(pyridin-3-ylmethyl)-8-oxa-4-azatricyclo[7.4.0.02,6]trideca-1(13),9,11-triene-6-carboxylic acid
2-amino-N-{1H,4H,5H,6H,7H,8H-cyclohepta[c]pyrazol-3-ylmethyl}-N-methyl-6-(propan-2-yl)pyrimidine-4-carboxamide
1-(dimethylamino)-2-[4-(5-phenyl-1,2-oxazole-3-carbonyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-7-yl]propan-2-ol
1-(3-methoxypropyl)-4-(2,3,4,5-tetrahydro-1-benzoxepin-4-ylmethyl)piperazine
1-(2-methoxyphenyl)-3-{1-[1-(3-methoxypropyl)piperidin-4-yl]-1H-pyrazol-5-yl}urea
1-[4-(2-cyclobutyl-5-fluoro-1H-1,3-benzodiazol-1-yl)piperidin-1-yl]-2-(2,5-dimethoxyphenyl)ethan-1-one
[3-ethyl-1-(2-propylpyridine-4-carbonyl)piperidin-3-yl]methanol
N-({1-[(5-chloro-1,3-dimethyl-1H-pyrazol-4-yl)sulfonyl]piperidin-3-yl}methyl)pyridine-3-carboxamide
4-tert-butyl-6-[3-(2-hydroxypropan-2-yl)pyrrolidine-1-carbonyl]-1,2-dihydropyrimidin-2-one
4-{[3-(2-hydroxyethoxy)phenyl]methyl}-1-(3-methoxyphenyl)piperazin-2-one
N-(2-{[(1S,9aR)-octahydro-1H-quinolizin-1-ylmethyl]amino}ethyl)pyridine-4-carboxamide
2-(2-hydroxyethyl)-6-{[5-(oxan-2-yl)furan-2-yl]methyl}-1H,2H,3H,4H,5H,6H,7H-pyrazolo[3,4-c]pyridin-3-one
(2R,6R)-11-methoxy-4-{[3-(methylsulfanyl)phenyl]methyl}-8-oxa-4-azatricyclo[7.4.0.02,6]trideca-1(13),9,11-triene-6-carboxylic acid
2-methoxy-1-[1'-(2-methylbenzoyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-5-yl]ethan-1-one
{1-[(4-fluoro-3-methoxyphenyl)methyl]-4-[(4-methoxyphenyl)methyl]piperidin-4-yl}methanol
N-[(3-hydroxy-4-methoxyphenyl)methyl]-N-methylimidazo[1,2-a]pyrimidine-2-carboxamide
8-[2-(2-oxopyrrolidin-1-yl)acetyl]-2-(pyridin-4-ylmethyl)-2,8-diazaspiro[5.5]undecan-3-one
1-(cyclopropylmethyl)-4-{5,7-dimethylpyrazolo[1,5-a]pyrimidine-3-carbonyl}-2-(propan-2-yl)-1,4-diazepane
methyl 4-{3-[1-(pyrrolidin-1-yl)ethyl]phenyl}-1H-pyrrole-2-carboxylate
(1R,2S,6R,7S)-4-{3-methyl-5H,6H-imidazo[2,1-b][1,3]thiazole-2-carbonyl}-4-azatricyclo[5.2.2.02,6]undecane
1-[(3R,4R)-3-(hydroxymethyl)-4-[(4-methylpiperazin-1-yl)methyl]pyrrolidine-1-carbonyl]cyclopropane-1-carboxamide
N-({7-[(2-ethoxyphenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}methyl)pyridine-2-carboxamide
N-[(2,2-dimethyl-1-phenylcyclopropyl)methyl]-1H,4H,5H,6H-cyclopenta[c]pyrazole-3-carboxamide
N-[(3S,5S)-1-[(1,5-dimethyl-1H-pyrazol-4-yl)methyl]-5-(ethylcarbamoyl)pyrrolidin-3-yl]pyrazine-2-carboxamide
2-chloro-N-{2-[2-(2-methoxyphenyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]ethyl}benzamide
2,2-dimethyl-N-(3-{11-oxo-4,6,10,12-tetraazatricyclo[7.3.0.03,7]dodeca-1(9),2,4,7-tetraen-5-yl}pyridin-2-yl)propanamide
3-(dimethyl-1,3-thiazol-5-yl)-7-methyl-1H-indole
5-methanesulfonyl-4-(piperidin-3-yl)-N-(pyridin-4-ylmethyl)pyrimidin-2-amine
3-(azepane-1-carbonyl)-N-[2-(2-fluorophenyl)ethyl]-1-(prop-2-en-1-yl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
2-amino-N-[3-(furan-2-yl)propyl]-4-methyl-1,3-thiazole-5-carboxamide
N-methyl-N-(2-phenyl-1-{1-[(3-phenyl-1H-pyrazol-4-yl)methyl]piperidin-4-yl}ethyl)thiophene-2-carboxamide
2-[2-({methyl[(4-methyl-1H-imidazol-2-yl)methyl]amino}methyl)phenoxy]acetic acid
2-(2-{1-[2-(1H-indol-3-yl)acetyl]piperidin-3-yl}-1H-imidazol-1-yl)acetamide
3-(3-ethyl-1,4-dimethyl-1H-pyrazol-5-yl)-1-[(2-methoxy-4,6-dimethylpyridin-3-yl)methyl]urea
N-(oxolan-2-ylmethyl)-3-(2-phenylethyl)-N-propyl-1,2-oxazole-5-carboxamide
(3aR,6aR)-2-cyclopentyl-N-{[4-(hydroxymethyl)oxan-4-yl]methyl}-octahydropyrrolo[3,4-c]pyrrole-3a-carboxamide
3-[({1-[(5-chloro-3-ethyl-1-methyl-1H-pyrazol-4-yl)methyl]piperidin-4-yl}oxy)methyl]pyridine
1-[2-(3-methyl-1H-1,2,4-triazol-5-yl)pyrrolidin-1-yl]-3-(pyridin-3-yl)propan-1-one
3-(2-{2-azabicyclo[2.2.1]heptan-2-yl}-2-oxoethyl)-3-(3-fluorophenyl)-1-(pyridin-3-ylmethyl)pyrrolidine-2,5-dione
N-{[8-(propan-2-yl)-1-oxa-8-azaspiro[4.5]decan-2-yl]methyl}-2-(1H-1,2,4-triazol-3-yl)benzamide
3-{[1-(hydroxymethyl)-9-[(6-methylpyridin-2-yl)methyl]-3,9-diazaspiro[5.5]undecan-3-yl]methyl}phenol
N,5-dimethyl-N-(2-methylpropyl)-4-[(2-phenylethyl)amino]thieno[2,3-d]pyrimidine-6-carboxamide