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2-{[(2-chlorophenyl)methyl]sulfanyl}-N-[(3-ethyl-1,2,4-oxadiazol-5-yl)methyl]acetamide
2-[1-(2,2-diphenylethyl)-3-oxopiperazin-2-yl]-N-[(1-ethyl-1H-imidazol-2-yl)methyl]acetamide
N,N-dimethyl-4-[2-(2,4,7-trimethyl-1H-indol-3-yl)acetyl]piperazine-1-carboxamide
(2R,3R)-3-amino-1'-(naphthalene-2-carbonyl)-2,3-dihydrospiro[indene-1,4'-piperidine]-2-ol
[(5,6-dimethyl-1H-1,3-benzodiazol-2-yl)methyl]({[3-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl})amine
ethyl 5-[3,5-bis(trifluoromethyl)benzoyl]-1-(prop-2-en-1-yl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylate
2-(dimethyl-1,2-oxazol-4-yl)-1-[3-(3-{[methyl(quinolin-6-ylmethyl)amino]methyl}phenoxymethyl)piperidin-1-yl]ethan-1-one
(4-methoxyphenyl)[3-methyl-1-(pyridin-2-yl)-1H-1,2,4-triazol-5-yl]methanol
{1-[(2-cyclohexylpyrimidin-5-yl)methyl]-3-(cyclopropylmethyl)piperidin-3-yl}methanol
N-[5-oxo-1-(2-phenylethyl)pyrrolidin-3-yl]but-3-enamide
5-(methoxymethyl)-N-[(2,3,5-trimethyl-1H-indol-7-yl)methyl]furan-2-carboxamide
2-(2H-1,2,3-benzotriazol-2-yl)-1-[2-(3-phenylpropyl)morpholin-4-yl]ethan-1-one
N-(2-methyl-2H-1,2,3-triazol-4-yl)-2-{4-[4-methyl-6-(methylamino)pyrimidin-2-yl]-1H-pyrazol-1-yl}acetamide
4-{1-[4-(4-methoxypyrimidin-2-yl)piperazin-1-yl]-2-methylpropan-2-yl}morpholine
N-[(2-phenyl-1,3-oxazol-4-yl)methyl]-2-propyl-1,3-thiazole-4-carboxamide
4-[3-(1H-1,2,3,4-tetrazol-1-yl)-5-(2,3,4-trimethoxyphenyl)benzoyl]thiomorpholine
N-{2-[(4-methyl-6-oxo-1,6-dihydropyrimidin-2-yl)amino]ethyl}-2-(pyridin-3-yl)-2-(pyrrolidin-1-yl)acetamide
4-{4-[2-(2,5-dimethyl-1H-pyrrol-1-yl)ethyl]piperazin-1-yl}-5-ethyl-2-methylpyrimidine
(3S,4R)-4-(2H-1,3-benzodioxol-5-yl)-1-(1-methylpiperidine-4-carbonyl)pyrrolidine-3-carboxylic acid
3-[(3R,4R)-3-(hydroxymethyl)-4-{[(2-methoxyethyl)(methyl)amino]methyl}pyrrolidine-1-carbonyl]-2-methyl-4,5,6,7-tetrahydro-1-benzofuran-4-one
4-{1-[(4-fluorophenyl)methyl]-1H,4H,5H,6H-pyrrolo[3,4-c]pyrazol-5-yl}-6-methoxypyrimidine
4-[5-methyl-4-(4-methylphenyl)-1H-imidazol-2-yl]-1-(propan-2-yl)pyrrolidin-2-one
1-methyl-1'-(6-oxo-1,6-dihydropyridine-3-carbonyl)-1,2-dihydrospiro[indole-3,3'-piperidine]-2-one
N-cyclopropyl-3-{[3-(3-oxopiperazin-1-yl)propyl]sulfamoyl}benzamide
2-amino-N-[(5-tert-butyl-1,3-benzoxazol-2-yl)methyl]-2-(3,5-dimethyl-1H-pyrazol-4-yl)acetamide
5-{[(2R,3R)-3-[ethyl(methyl)amino]-2-hydroxy-2,3-dihydrospiro[indene-1,4'-piperidine]-1'-yl]carbonyl}-1,2-dihydropyridin-2-one
ethyl 3-(2-methoxyethyl)-1-[(2E)-3-(4-methoxyphenyl)prop-2-en-1-yl]piperidine-3-carboxylate
N-(oxan-4-yl)-2,3,4,5-tetrahydro-1-benzoxepine-4-carboxamide
(2R,3R,6R)-3-(4-methoxyphenyl)-5-(1-methylpiperidine-4-carbonyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
N-{[5-(2-methoxyethyl)-1,2,4-oxadiazol-3-yl]methyl}-10-oxa-5,7-diazatricyclo[9.4.0.03,8]pentadeca-1(11),3,5,7,12,14-hexaen-4-amine
2-(3-hydroxypiperidin-1-yl)-N-[(3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl)methyl]acetamide
4-{4-[(4-methanesulfonyl-1,4-diazepan-1-yl)methyl]phenyl}-2-methylbutan-2-ol
3-butyl-1-methyl-4-(6-oxo-1,6-dihydropyridine-3-carbonyl)piperazin-2-one
1-(2-chlorophenyl)-4-[1-(2-methoxyethyl)piperidine-3-carbonyl]piperazin-2-one
3-(1-{[2-(methylsulfanyl)phenyl]methyl}piperidin-3-yl)propanoic acid
2-(2,3-dimethoxyphenyl)-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-4-one
(4aS,8aR)-1-[2-(1H-imidazol-4-yl)ethyl]-6-(4,4,4-trifluorobutanoyl)-decahydro-1,6-naphthyridin-2-one
1-[3-(hydroxymethyl)-3-(2-methoxyethyl)piperidin-1-yl]-2-(2,3,6-trimethylphenoxy)ethan-1-one
2-[2-(3-ethyl-1,2-oxazol-5-yl)-1H-imidazol-1-yl]-3-phenylpropanoic acid
N-{1-[(3-fluorophenyl)methyl]-5-oxopyrrolidin-3-yl}-3-methoxypropanamide
N-(prop-2-en-1-yl)-4-{3-[(pyridin-3-ylmethyl)carbamoyl]piperidin-1-yl}piperidine-1-carboxamide
N-(4-fluoro-2-methylphenyl)-2-{[1-(2-methylpropyl)piperidin-4-yl]amino}acetamide
1-[(2-ethylpyrimidin-4-yl)methyl]-4-(2-methylquinolin-6-yl)piperidin-4-ol
3-[(1,1-dioxo-1λ6-thiolan-3-yl)methyl]-1-[4-ethoxy-3-(1H-pyrrol-1-yl)phenyl]urea
1-[2-(4-chloro-2-methylphenoxy)ethyl]-4-(oxane-4-carbonyl)piperazine
N-(2-{7-[2-(2-oxo-4-phenylpyrrolidin-1-yl)acetyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}ethyl)cyclohexanecarboxamide
3-(4-methyl-1,3-thiazol-5-yl)-1-[3-(1-methyl-1H-imidazole-2-carbonyl)piperidin-1-yl]propan-1-one
3-{2-[4-(6-chloropyridazin-3-yl)piperazin-1-yl]ethyl}-2,3-dihydro-1,3-benzoxazol-2-one
2-{[(7-methoxynaphthalen-2-yl)oxy]methyl}-4-(2-phenylazetidine-1-carbonyl)-1,3-oxazole
6-fluoro-4-[4-(1H-pyrrole-2-carbonyl)piperazine-1-carbonyl]-1,2,3,4-tetrahydroquinolin-2-one