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3-(2,4-difluorophenyl)-5-(2,3-dihydro-1-benzofuran-5-ylmethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine
2-methoxy-1-(4-{2-[4-(methoxymethyl)piperidine-1-carbonyl]phenoxy}piperidin-1-yl)ethan-1-one
4-methyl-2-(propan-2-yl)-N-{[3-(thiophen-2-yl)-1H-pyrazol-4-yl]methyl}-1,3-thiazole-5-carboxamide
N-ethyl-N-{[5-(2-methylpropyl)-1,2,4-oxadiazol-3-yl]methyl}-1H-1,2,4-triazole-5-carboxamide
2-[({5-[1-(2-ethylpyridine-4-carbonyl)piperidin-4-yl]-4-methyl-4H-1,2,4-triazol-3-yl}methyl)(methyl)amino]ethan-1-ol
1-(2-chloropyridin-3-yl)-3-[(1-propyl-1H-pyrazol-4-yl)methyl]urea
N-cyclopropyl-5-(morpholin-4-ylmethyl)-N-propyl-1,2-oxazole-3-carboxamide
2-methoxy-N-({1-[(2-methylphenyl)methyl]piperidin-4-yl}methyl)-N-(pyridin-3-ylmethyl)acetamide
(1R,5S)-6-methyl-3-{2-[(4-methyl-6-oxo-1,6-dihydropyrimidin-2-yl)sulfanyl]acetyl}-3,6-diazabicyclo[3.2.2]nonan-7-one
N-[2-methyl-3-(pyrrolidin-1-yl)phenyl]-4-(thiomorpholin-4-yl)piperidine-1-carboxamide
(1S,5R)-3-methanesulfonyl-6-(pyridine-3-sulfonyl)-3,6-diazabicyclo[3.2.2]nonane
4-hydroxy-2-{2-oxo-1,2-dihydrospiro[indole-3,3'-piperidine]-1'-ylmethyl}quinoline-6-carboxamide
(3aR,6aR)-2-methanesulfonyl-5-[(3-methyl-1H-indol-2-yl)methyl]-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
5-(methoxymethyl)-N-[2-(4-methoxyphenyl)ethyl]pyrazolo[1,5-a]pyrimidin-7-amine
4-{1-[1-(2-methoxyphenyl)-1H-pyrazole-4-carbonyl]pyrrolidin-2-yl}-3,5-dimethyl-1,2-oxazole
5-[({dimethyl-1H-pyrazolo[3,4-d][1,3]thiazol-5-yl}amino)methyl]-N-methyl-1,2,4-oxadiazole-3-carboxamide
1-(2-fluorophenyl)-N-{2H,3H-imidazo[2,1-b][1,3]thiazol-6-ylmethyl}-2,2-dimethylcyclopropane-1-carboxamide
3-(2-{4-[(dimethylamino)methyl]phenyl}piperidine-1-carbonyl)-5-fluorobenzonitrile
N,6-dimethyl-2-{3-[4-methyl-5-(1H-pyrazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}pyrimidin-4-amine
4-{[1-(2-methoxyacetyl)piperidin-4-yl]oxy}-N-(1H-1,2,3,4-tetrazol-5-ylmethyl)benzamide
5-acetyl-N-methyl-N-(pyridin-3-ylmethyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-2-carboxamide
2-ethyl-9-(3-hydroxynaphthalene-2-carbonyl)-2,9-diazaspiro[5.5]undecan-3-one
methyl 2-{[(3-chlorophenyl)methyl]sulfamoyl}-6-cyclopentanecarbonyl-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
ethyl 1-[(2-hydroxy-3-methoxyphenyl)methyl]-4-{[2-(trifluoromethyl)phenyl]methyl}piperidine-4-carboxylate
{imidazo[1,2-a]pyridin-3-ylmethyl}(methyl){[2-(propan-2-yl)-1,3-oxazol-4-yl]methyl}amine
N-[(1,4-dimethylpiperazin-2-yl)methyl]-10-oxa-5,7-diazatricyclo[9.4.0.03,8]pentadeca-1(11),3,5,7,12,14-hexaen-4-amine
1-(2,3-dimethylphenyl)-N-{[2-(2-methylphenyl)pyrimidin-5-yl]methyl}-4,5,6,7-tetrahydro-1H-indazol-4-amine
N-[3-(3-methoxypyrazin-2-yl)phenyl]acetamide
2-{5-[2-amino-6-(propan-2-yloxy)pyrimidin-4-yl]-1H,4H,5H,6H-pyrrolo[3,4-c]pyrazol-1-yl}ethan-1-ol
N-(4-tert-butyl-1,3-thiazol-2-yl)-2-[(pyridin-4-ylmethyl)amino]acetamide
4-(4-ethyl-2-methyl-1,3-thiazole-5-carbonyl)-2-[1-(2-methoxyethyl)-1H-1,2,3,4-tetrazol-5-yl]morpholine
4-{[1-(furan-2-ylmethyl)piperidin-4-yl]methyl}thiomorpholine
1-cyclopentyl-N3-ethyl-4-oxo-N5-{[4-(trifluoromethoxy)phenyl]methyl}-1,4-dihydropyridine-3,5-dicarboxamide
1-methyl-5-[3-(2-phenylacetyl)piperidine-1-carbonyl]-1,2-dihydropyridin-2-one
1-[(1-ethyl-3-methyl-1H-pyrazol-4-yl)methyl]-N-[4-(2-fluorophenoxy)phenyl]piperidine-4-carboxamide
4-{[1-(2-propyl-1,3-thiazole-4-carbonyl)piperidin-2-yl]methyl}morpholine
5-cyclobutanecarbonyl-1'-[(2E)-3-phenylprop-2-en-1-yl]-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
3-{1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-5-carbonyl}-2-methyl-1,2,3,4-tetrahydroisoquinoline
N-[(3S)-1-benzylpyrrolidin-3-yl]-3-{imidazo[1,2-a]pyridin-2-yl}-N-methylpropanamide
(1S,6R)-9-{[4-(1H-pyrazol-1-ylmethyl)phenyl]methyl}-3,9-diazabicyclo[4.2.1]nonane
6-[1-(cyclohex-3-en-1-ylmethyl)piperidin-4-yl]-2-methylpyrimidin-4-ol
2-(dimethylamino)-2-(2-fluorophenyl)-N-{[2-(morpholin-4-yl)pyridin-3-yl]methyl}acetamide
3-{2-[2-(morpholin-4-yl)ethyl]piperidine-1-carbonyl}pyridin-2-ol
N-[(1-ethylpyrrolidin-2-yl)methyl]-4-(4-methylphenoxy)piperidine-4-carboxamide
5-(3-acetylphenyl)-N-(prop-2-en-1-yl)furan-2-carboxamide
N-[2-(cyclohex-1-en-1-yl)ethyl]-5-(3-hydroxypiperidine-1-carbonyl)-1-[(2-methoxyphenyl)methyl]-4-oxo-1,4-dihydropyridine-3-carboxamide
2-methyl-5-[(4-{octahydropyrrolo[1,2-a]piperazine-2-carbonyl}-1,3-oxazol-2-yl)methoxy]-1,3-benzothiazole
3-(2-chlorophenyl)-3-phenyl-N-[3-(1H-1,2,4-triazol-1-yl)propyl]propanamide
1-tert-butyl-N-methyl-N-{[2-(thiophen-2-yl)-1,3-thiazol-4-yl]methyl}-1H-pyrrole-3-carboxamide
2-[(isoquinolin-5-yloxy)methyl]-N-methyl-N-(prop-2-en-1-yl)-1,3-oxazole-4-carboxamide