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(4aS,8aR)-N-(5-acetamido-2-methoxyphenyl)-decahydroisoquinoline-2-carboxamide
(2S)-2-(2,3-difluorophenyl)-2-[2-(1-propylpiperidin-4-yl)acetamido]acetic acid
methyl N-(2-{4-[(2-fluorophenyl)methyl]-1,4-diazepan-1-yl}-2-oxoethyl)carbamate
2-{1-[1-(1-ethylpiperidin-4-yl)piperidin-4-yl]-1H-1,2,3-triazol-4-yl}propan-2-amine
ethyl 3-benzyl-1-{[2-(dimethylamino)-1,3-thiazol-5-yl]methyl}piperidine-3-carboxylate
(3aS,6aS)-1-[3-(trifluoromethyl)benzenesulfonyl]-octahydropyrrolo[2,3-c]pyrrole
1-(4-methylphenyl)-4-{2-[4-(propan-2-yl)morpholin-2-yl]acetyl}piperazin-2-one
8-(6-methylpyridazin-3-yl)-2-(pyridin-4-ylmethyl)-2,8-diazaspiro[5.5]undecan-3-one
N-{[1-(2,3-dihydro-1H-inden-2-yl)piperidin-4-yl]methyl}-N-[3-(dimethylamino)propyl]-1-methyl-1H-pyrazole-5-carboxamide
4-({4-hydroxy-4-[3-(trifluoromethyl)phenyl]piperidin-1-yl}methyl)-1,5-dimethyl-1H-pyrrole-2-carbonitrile
4-[(3R,4R)-3-(hydroxymethyl)-4-[(4-methyl-1,4-diazepan-1-yl)methyl]pyrrolidine-1-carbonyl]phenol
(1S,5R)-6-(1-ethyl-1H-pyrazole-5-carbonyl)-3-(3-phenylpropyl)-3,6-diazabicyclo[3.2.2]nonane
4-[1-(3-methylbutanoyl)piperidine-4-carbonyl]-1-phenylpiperazin-2-one
(1S,6R)-9-(1,2-oxazole-5-carbonyl)-3,9-diazabicyclo[4.2.1]nonan-4-one
3-(4,5-dimethyl-1H-pyrazol-3-yl)-1-{5-hydroxy-1-oxa-9-azaspiro[5.5]undecan-9-yl}propan-1-one
2-[4-({3-[(4-fluorophenyl)methyl]-3-(hydroxymethyl)piperidin-1-yl}methyl)phenoxy]ethan-1-ol
3-[({1-[2-(1H-1,2,4-triazol-1-yl)benzoyl]piperidin-4-yl}oxy)methyl]pyridine
1-{3-[1-(cyclobutylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}-3-(3-methoxyphenyl)propan-1-one
5-methoxy-3-{2-[2-(2-methyl-1H-imidazol-1-yl)ethyl]piperidine-1-carbonyl}-1H-indazole
7-cyclopentyl-2-(3-phenoxypropanoyl)-2,7-diazaspiro[4.5]decan-6-one
5-[(benzylsulfamoyl)amino]-N,N-dimethyl-1-benzothiophene-2-carboxamide
N-{1-[4-methyl-2-(pyridin-4-yl)pyrimidin-5-yl]ethyl}-2H,3H-thieno[3,4-b][1,4]dioxine-5-carboxamide
[(2S)-1-{[7-chloro-2-(2-methoxyphenyl)quinolin-3-yl]methyl}pyrrolidin-2-yl]methanol
2-methoxy-4-(4-phenyl-1H-imidazol-5-yl)-6-(prop-2-en-1-yl)phenol
1-[(3S,7S)-3-(hydroxymethyl)-9-oxa-5-azatricyclo[8.4.0.03,7]tetradeca-1(10),11,13-trien-5-yl]-3-(pyridin-3-yl)propan-1-one
2-[3-({3-[2-(2,6-difluorophenyl)ethyl]piperidin-1-yl}methyl)phenoxy]acetic acid
3-({4-[3-(4-ethylpiperidine-1-carbonyl)piperidin-1-yl]piperidin-1-yl}methyl)pyridine
N-(2-{[(3-chlorophenyl)methyl]sulfanyl}ethyl)-1-ethyl-5-oxopyrrolidine-3-carboxamide
1-{4-[3-(cyclopropylmethyl)-1-methyl-1H-1,2,4-triazol-5-yl]piperidin-1-yl}ethan-1-one
2-(2,4-dioxo-1,3-diazinan-1-yl)-N-[1-(pyridin-4-yl)propyl]benzamide
(1S,6R)-9-[6-(piperidine-1-carbonyl)pyrazin-2-yl]-3,9-diazabicyclo[4.2.1]nonane
N-ethyl-4-hydroxy-N-{[5-(2-methylpropyl)-1,2,4-oxadiazol-3-yl]methyl}-2-(pyridin-2-yl)pyrimidine-5-carboxamide
5-{1,8-dioxa-4,11-diazaspiro[5.6]dodecane-4-carbonyl}-N,N,4-trimethylpyrimidin-2-amine
2-[4-(pyrrolidine-1-sulfonyl)piperazin-1-yl]-4-(3,3,3-trifluoropropyl)pyrimidine
N-{[5-(methoxymethyl)-1H-pyrazol-3-yl]methyl}-6-methyl-2-(piperidin-1-yl)pyrimidin-4-amine
4-[(2R)-3,4-dihydro-2H-1-benzopyran-2-ylmethyl]-8-thia-4,6,11-triazatricyclo[7.4.0.02,7]trideca-1(9),2(7),5-trien-3-one
N,2,5-trimethyl-N-[1-(pyridin-3-yl)ethyl]-[1,3]oxazolo[5,4-d]pyrimidin-7-amine
1-methyl-4-({1-[4-(methylsulfanyl)phenyl]-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-2-yl}methyl)-1H-pyrazole
N,N-dimethyl-2-(4H-1,2,4-triazol-4-yl)ethane-1-sulfonamide
(3aS,6aR)-3-[3-(4-fluorophenyl)propyl]-5-(1,3-thiazole-5-carbonyl)-hexahydro-2H-pyrrolo[3,4-d][1,3]oxazol-2-one
4-cyclobutyl-6-methyl-2-[3-(2-methylpiperidin-1-yl)azetidin-1-yl]pyrimidine
ethyl 1-[2-(4,6-dimethylpyrimidin-2-yl)ethyl]-4-oxo-5-phenoxy-1,4-dihydropyridine-3-carboxylate
(3R,4R)-4-(azepan-1-yl)-1-(quinolin-8-ylmethyl)piperidin-3-ol
1-{4-[(3,5-dimethyl-1H-pyrazol-1-yl)methyl]phenyl}-3-[2-(furan-2-ylmethyl)-3-hydroxypropyl]urea
1-methyl-N-[(5-phenyl-1,2,4-oxadiazol-3-yl)methyl]azepane-2-carboxamide
4-(2-{1-methyl-1H,2H,3H,4H-pyrrolo[1,2-a]pyrazin-2-yl}-2-oxoethyl)-1,2,3,6-tetrahydropyridazine-3,6-dione
N-{1-[4-methyl-2-(pyridin-4-yl)pyrimidin-5-yl]ethyl}pyridine-4-carboxamide
N-(2,3-dihydro-1,4-benzodioxin-6-yl)-3-[1-(pyridin-4-ylmethyl)piperidin-4-yl]propanamide
ethyl 4-[5-(2,6-difluorophenoxymethyl)-1,2-oxazole-3-carbonyl]piperazine-1-carboxylate
(4aR,7aS)-1-{2-[(cyclopentylmethyl)(methyl)amino]pyrimidin-4-yl}-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione