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1-[(6-methoxypyridin-3-yl)methyl]-4-(2-methylpyridin-4-yl)piperazine
N-methyl-N-[(5-phenyl-1H-pyrazol-4-yl)methyl]oxolane-2-carboxamide
6-fluoro-4-[2-(3-methyl-1,2,4-oxadiazol-5-yl)pyrrolidine-1-carbonyl]-2-(1-methyl-1H-pyrazol-4-yl)quinoline
(5S,9aS,9bS)-2-[(3-chlorophenyl)methyl]-5-(1H-indol-2-yl)-octahydro-1H-pyrrolo[3,4-h]pyrrolizin-1-one
(4aS,8aR)-6-{[3-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}-decahydro-1,6-naphthyridine-4a-carboxylic acid
N-(3-methoxy-1,5-dimethyl-1H-pyrazol-4-yl)thiomorpholine-4-carboxamide
2-(2H-1,3-benzodioxol-5-yl)-N-{[2-(morpholin-4-yl)pyridin-3-yl]methyl}acetamide
5-(methanesulfonylmethyl)-2-{[1-(pyrrolidin-1-yl)hex-5-en-2-yl]oxy}pyridine
3-[4-(1-butyl-1H-imidazol-2-yl)piperidine-1-carbonyl]-1-methyl-4,5,6,7-tetrahydro-1H-indazole
2-(1-benzyl-2-methyl-4-oxo-4,5,6,7-tetrahydro-1H-indol-3-yl)-N,N-diethylacetamide
4-[1-(pyridin-4-ylmethyl)piperidin-3-yl]pyrimidine
3,5-dimethoxy-N-{[1-(4-methoxypyrimidin-2-yl)piperidin-3-yl]methyl}benzamide
N-(1,3-benzothiazol-2-ylmethyl)-1-(prop-2-en-1-yl)-3-(thiomorpholine-4-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
3-({[2-(cyclohex-1-en-1-yl)ethyl]amino}methyl)-5,6,7-trimethoxy-N,N-dimethylquinolin-2-amine
4-[(2,3-dimethyl-1H-indol-7-yl)methyl]-3-methyl-1-(2-methylpropyl)piperazin-2-one
2-(3-fluorophenoxy)-1-[3-(1H-imidazol-2-yl)piperidin-1-yl]ethan-1-one
5-(1-{[2-(butylsulfanyl)pyrimidin-5-yl]methyl}pyrrolidin-2-yl)thiophene-2-carboxamide
N-[1-(1H-indol-2-yl)ethyl]-1-(2-methoxyethyl)-N-methylpiperidine-4-carboxamide
2-{3-[(3R,4R)-3-[(dimethylamino)methyl]-4-(hydroxymethyl)pyrrolidine-1-carbonyl]phenoxy}acetamide
N-(1-{1-[(2E)-2-methylbut-2-en-1-yl]piperidin-4-yl}-1H-pyrazol-5-yl)-4-phenylbutanamide
N-[2-(4-ethylmorpholin-2-yl)ethyl]-2,3-dihydro-1-benzofuran-7-carboxamide
1-{1H-pyrrolo[2,3-b]pyridin-6-yl}-3-{[1,2,4]triazolo[4,3-a]pyridin-3-yl}piperidine
N-(1-hydroxybutan-2-yl)-N-[(5-methylthiophen-2-yl)methyl]-2-(morpholin-4-yl)pyridine-3-carboxamide
(4aS,7aR)-1-(5-methyl-1,2-oxazole-3-carbonyl)-4-(3-methylbutanoyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
3-{4-[2-(1,2-benzoxazol-3-yl)acetyl]piperazin-1-yl}-1,2-dihydropyrazin-2-one
N-{[(2S,4S)-4-fluoropyrrolidin-2-yl]methyl}-2,3-dimethylquinoxaline-6-carboxamide
4-(4-chloro-3-methyl-1H-pyrazol-5-yl)-3-methyl-1-(2-methylphenyl)-1H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one
3-[3-(6-hydroxy-2-methylpyrimidin-4-yl)piperidine-1-carbonyl]-2-methyl-4,5,6,7-tetrahydro-1H-indol-4-one
2-amino-4-{methyl[2-(pyridin-2-yl)ethyl]amino}quinazoline-6-carboxylic acid
8-(3-hydroxypyridine-2-carbonyl)-3-(2-phenylethyl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
7-chloro-3-[1-(6-methylpyridin-2-yl)propan-2-yl]-3,4-dihydroquinazolin-4-one
ethyl 3-(2-phenoxyethyl)-1-(4,4,4-trifluorobutyl)piperidine-3-carboxylate
2-[(2R,3R,6R)-3-(2-methoxyphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecane-5-carbonyl]benzonitrile
1-(1-{[2,5-dimethoxy-4-(methylsulfanyl)phenyl]methyl}piperidin-4-yl)piperidin-3-ol
1-cyclopentyl-N-{[1-methyl-2-(methylsulfanyl)-1H-imidazol-5-yl]methyl}piperidine-3-carboxamide
5-methoxy-N-[(2,3,5-trimethyl-1H-indol-7-yl)methyl]furan-2-carboxamide
4-{3-[4-(2-aminopyrimidin-4-yl)piperidine-1-carbonyl]phenyl}-2-methylbut-3-yn-2-ol
4-(2-methyl-5-propylpyrimidin-4-yl)-N-(pyridin-4-ylmethyl)-1H-pyrrolo[2,3-b]pyridin-6-amine
1-methyl-N-[1-(pyridin-2-ylmethyl)piperidin-3-yl]-1H-indole-3-carboxamide
N-ethyl-3,5-dimethyl-N-[2-(2-methylphenoxy)ethyl]-1H-pyrrole-2-carboxamide
1-({4-methyl-5-[1-(oxan-4-yl)piperidin-4-yl]-4H-1,2,4-triazol-3-yl}methyl)piperidin-4-ol
(2R,3S,6R)-N-(furan-2-ylmethyl)-3-(2-methoxyphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecane-5-carboxamide
2-[5-(1H-1,3-benzodiazol-1-ylmethyl)-3-methyl-1H-1,2,4-triazol-1-yl]acetic acid
2-[4-(3,6-dimethylpyrazin-2-yl)-1-[(4-methoxy-2,3-dimethylphenyl)methyl]piperazin-2-yl]ethan-1-ol
5-(furan-3-yl)-4-phenyl-1-[4-(pyrrolidin-1-yl)butyl]-1H-imidazole
2-amino-6-(1-propyl-1H-1,2,3-benzotriazol-5-yl)-4-(pyridin-4-yl)pyridine-3-carbonitrile
N-[(3R,4S)-4-cyclopropyl-1-(pyrimidin-5-ylmethyl)pyrrolidin-3-yl]-3-methanesulfonylpropanamide
ethyl 3-benzyl-1-{[3-(methylsulfanyl)phenyl]carbamoyl}piperidine-3-carboxylate
N-[(2-chloro-6-fluorophenyl)methyl]-1-cyclopropyl-N-ethyl-6-oxopiperidine-3-carboxamide
9-[(1-ethyl-1H-pyrazol-5-yl)sulfonyl]-2-(propan-2-yl)-2,9-diazaspiro[5.5]undecan-3-one